8C13
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![BU of 8c13 by Molmil](/molmil-images/mine/8c13) | Crystal structure of pVHL:ElonginC:ElonginB complex bound to PROTAC JW48 | 分子名称: | (2~{S},4~{R})-1-[(2~{S})-2-[3-[2-[2-[2-(acetamidomethyl)-4-(6,7-dihydro-5~{H}-pyrrolo[1,2-a]imidazol-2-yl)phenoxy]ethoxy]ethoxy]propanoylamino]-3,3-dimethyl-butanoyl]-~{N}-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxidanyl-pyrrolidine-2-carboxamide, Elongin-B, Elongin-C, ... | 著者 | Kraemer, A, Weckesser, J, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2022-12-20 | 公開日 | 2022-12-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Tracking the PROTAC degradation pathway in living cells highlights the importance of ternary complex measurement for PROTAC optimization. Cell Chem Biol, 30, 2023
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2J9A
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![BU of 2j9a by Molmil](/molmil-images/mine/2j9a) | blLAP in Complex with Microginin FR1 | 分子名称: | (2S,3R)-3-AMINO-2-HYDROXYDECANOIC ACID, (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, ... | 著者 | Kraft, M, Schleberger, C, Weckesser, J, Schulz, G.E. | 登録日 | 2006-11-06 | 公開日 | 2006-12-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Binding Structure of the Leucine Aminopeptidase Inhibitor Microginin Fr1. FEBS Lett., 580, 2006
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1OKX
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![BU of 1okx by Molmil](/molmil-images/mine/1okx) | Binding Structure of Elastase Inhibitor Scyptolin A | 分子名称: | ELASTASE 1, SCYPTOLIN A | 著者 | Matern, U, Schleberger, C, Jelakovic, S, Weckesser, J, Schulz, G.E. | 登録日 | 2003-07-31 | 公開日 | 2003-10-24 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Binding Structure of Elastase Inhibitor Scyptolin A Chem.Biol., 10, 2003
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