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PDB: 12920 件

2JUV
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AbaA3-DKP-insulin
分子名称: Insulin A chain, Insulin B chain
著者Huang, K, Chan, S, Hua, Q, Chu, Y, Wang, R, Klaproth, B, Jia, W, Whittaker, J, De Meyts, P, Nakagawa, S.H, Steiner, D.F, Katsoyannis, P.G, Weiss, M.A.
登録日2007-09-05
公開日2007-10-16
最終更新日2021-10-20
実験手法SOLUTION NMR
主引用文献The A-chain of Insulin Contacts the Insert Domain of the Insulin Receptor: PHOTO-CROSS-LINKING AND MUTAGENESIS OF A DIABETES-RELATED CREVICE.
J.Biol.Chem., 282, 2007
2JMB
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Solution structure of the protein Atu4866 from Agrobacterium tumefaciens
分子名称: Hypothetical protein Atu4866
著者Ai, X, Semesi, A, Yee, A, Arrowsmith, C.H, Li, S.S.C, Choy, W, Ontario Centre for Structural Proteomics (OCSP)
登録日2006-11-01
公開日2007-10-16
最終更新日2023-12-20
実験手法SOLUTION NMR
主引用文献Solution structure of the protein Atu4866 from Agrobacterium tumefaciens
To be Published
2JPC
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SSRB DNA Binding Protein
分子名称: SsrB
著者Liao, X, Kenney, L, Sheng, W, Integrated Center for Structure and Function Innovation (ISFI)
登録日2007-05-03
公開日2007-07-03
最終更新日2023-12-20
実験手法SOLUTION NMR
主引用文献SSRB DNA Binding Protein
To be Published
2DW7
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BU of 2dw7 by Molmil
Crystal structure of D-tartrate dehydratase from Bradyrhizobium japonicum complexed with Mg++ and meso-tartrate
分子名称: Bll6730 protein, MAGNESIUM ION, S,R MESO-TARTARIC ACID
著者Fedorov, A.A, Fedorov, E.V, Yew, W.S, Wood, B.M, Gerlt, J.A, Almo, S.C.
登録日2006-08-07
公開日2006-12-19
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Evolution of Enzymatic Activities in the Enolase Superfamily: d-Tartrate Dehydratase from Bradyrhizobium japonicum
Biochemistry, 45, 2006
2DIP
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BU of 2dip by Molmil
Solution structure of the ZZ domain of Zinc finger SWIM domain containing protein 2
分子名称: ZINC ION, Zinc finger SWIM domain-containing protein 2
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the ZZ domain of Zinc finger SWIM domain containing protein 2
To be Published
3T2B
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BU of 3t2b by Molmil
Fructose-1,6-bisphosphate aldolase/phosphatase from Thermoproteus neutrophilus, ligand free
分子名称: Fructose-1,6-bisphosphate aldolase/phosphatase, MAGNESIUM ION
著者Du, J, Say, R, Lue, W, Fuchs, G, Einsle, O.
登録日2011-07-22
公開日2011-10-26
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.52 Å)
主引用文献Active-site remodelling in the bifunctional fructose-1,6-bisphosphate aldolase/phosphatase.
Nature, 478, 2011
3TA2
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A. fulgidus GlnK3, MgATP/2-OG complex
分子名称: 2-OXOGLUTARIC ACID, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Maier, S, Schleberger, P, Lue, W, Wacker, T, Pflueger, T, Litz, C, Andrade, S.L.A.
登録日2011-08-03
公開日2011-10-26
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Mechanism of disruption of the Amt-GlnK complex by P(II)-mediated sensing of 2-oxoglutarate.
Plos One, 6, 2011
2K20
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Solution structure of Par-3 PDZ3 in complex with PTEN peptide
分子名称: Partitioning-defective 3 homolog, Protein tyrosine phosphatase and tensin homolog
著者Feng, W, Wu, H, Chan, L, Zhang, M.
登録日2008-03-18
公開日2008-06-10
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of Par-3 PDZ3 in complex with PTEN peptide
To be Published
2DIR
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BU of 2dir by Molmil
Solution structure of the THUMP domain of THUMP domain-containing protein 1
分子名称: THUMP domain-containing protein 1
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the THUMP domain of THUMP domain-containing protein 1
To be Published
2DIQ
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BU of 2diq by Molmil
Solution structure of the TUDOR domain of Tudor and KH domain containing protein
分子名称: Tudor and KH domain-containing protein
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the TUDOR domain of Tudor and KH domain containing protein
To be Published
3T2G
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BU of 3t2g by Molmil
Fructose-1,6-bisphosphate aldolase/phosphatase from Thermoproteus neutrophilus, Y229F variant with DHAP
分子名称: 1,3-DIHYDROXYACETONEPHOSPHATE, Fructose-1,6-bisphosphate aldolase/phosphatase, MAGNESIUM ION
著者Du, J, Say, R, Lue, W, Fuchs, G, Einsle, O.
登録日2011-07-22
公開日2011-10-26
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Active-site remodelling in the bifunctional fructose-1,6-bisphosphate aldolase/phosphatase.
Nature, 478, 2011
2DIX
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BU of 2dix by Molmil
Solution structure of the DSRM domain of Protein activator of the interferon-induced protein kinase
分子名称: Interferon-inducible double stranded RNA-dependent protein kinase activator A
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the DSRM domain of Protein activator of the interferon-induced protein kinase
To be published
2DOO
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BU of 2doo by Molmil
The structure of IMP-1 complexed with the detecting reagent (DansylC4SH) by a fluorescent probe
分子名称: BETA-LACTAMASE IMP-1, N-[4-({[5-(DIMETHYLAMINO)-1-NAPHTHYL]SULFONYL}AMINO)BUTYL]-3-SULFANYLPROPANAMIDE, ZINC ION
著者Kurosaki, H, Yamaguchi, Y, Yasuzawa, H, Jin, W, Yamagata, Y, Arakawa, Y.
登録日2006-05-01
公開日2006-11-28
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献Probing, inhibition, and crystallographic characterization of metallo-beta-lactamase (IMP-1) with fluorescent agents containing dansyl and thiol groups
Chemmedchem, 1, 2006
2DIU
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BU of 2diu by Molmil
Solution structure of the RRM domain of KIAA0430 protein
分子名称: KIAA0430 protein
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the RRM domain of KIAA0430 protein
To be Published
2DNF
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BU of 2dnf by Molmil
Solution structure of RSGI RUH-062, a DCX domain from human
分子名称: Doublecortin domain-containing protein 2
著者Ohashi, W, Hirota, H, Nagashima, T, Hayashi, F, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-04-26
公開日2006-10-26
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RSGI RUH-062, a DCX domain from human
TO BE PUBLISHED
2E73
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BU of 2e73 by Molmil
Solution structure of the phorbol esters/diacylglycerol binding domain of protein kinase C gamma
分子名称: Protein kinase C gamma type, ZINC ION
著者Tanabe, W, Suzuki, S, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-01-05
公開日2007-12-18
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the phorbol esters/diacylglycerol binding domain of protein kinase C gamma
To be Published
2E22
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BU of 2e22 by Molmil
Crystal structure of xanthan lyase in complex with mannose
分子名称: Xanthan lyase, alpha-D-mannopyranose
著者Maruyama, Y, Mikami, B, Hashimoto, W, Murata, K.
登録日2006-11-07
公開日2007-01-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献A Structural Factor Responsible for Substrate Recognition by Bacillus sp. GL1 Xanthan Lyase that Acts Specifically on Pyruvated Side Chains of Xanthan
Biochemistry, 46, 2007
2E5S
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BU of 2e5s by Molmil
Solution structure of the zf-CCCHx2 domain of muscleblind-like 2, isoform 1 [Homo sapiens]
分子名称: OTTHUMP00000018578, ZINC ION
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-12-22
公開日2007-06-26
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the RNA binding domain in the human muscleblind-like protein 2
Protein Sci., 18, 2009
2E72
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BU of 2e72 by Molmil
Solution structure of the zinc finger domain of human KIAA0461
分子名称: Pogo transposable element with ZNF domain, ZINC ION
著者Tanabe, W, Suzuki, S, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2007-01-05
公開日2007-07-10
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the zinc finger domain of human KIAA0461
To be Published
7GG6
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BU of 7gg6 by Molmil
Group deposition SARS-CoV-2 main protease in complex with inhibitors from the COVID Moonshot -- Crystal Structure of SARS-CoV-2 main protease in complex with ALP-POS-477dc5b7-2 (Mpro-x12171)
分子名称: (4R)-6-chloro-N-(isoquinolin-4-yl)-1,2,3,4-tetrahydroquinoline-4-carboxamide, 3C-like proteinase, DIMETHYL SULFOXIDE
著者Fearon, D, Aimon, A, Aschenbrenner, J.C, Balcomb, B.H, Bertram, F.K.R, Brandao-Neto, J, Dias, A, Douangamath, A, Dunnett, L, Godoy, A.S, Gorrie-Stone, T.J, Koekemoer, L, Krojer, T, Lithgo, R.M, Lukacik, P, Marples, P.G, Mikolajek, H, Nelson, E, Owen, C.D, Powell, A.J, Rangel, V.L, Skyner, R, Strain-Damerell, C.M, Thompson, W, Tomlinson, C.W.E, Wild, C, Walsh, M.A, von Delft, F.
登録日2023-08-11
公開日2023-11-08
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.599 Å)
主引用文献Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Science, 382, 2023
3TUH
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BU of 3tuh by Molmil
Crystal Structure of the N-terminal domain of an HSP90 in the presence of an the inhibitor ganetespib
分子名称: 5-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-4-(1-methyl-1H-indol-5-yl)-2,4-dihydro-3H-1,2,4-triazol-3-one, Heat shock protein HSP 90-alpha
著者Ying, W.
登録日2011-09-16
公開日2012-09-19
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of the N-terminal domain of an HSP90 in the presence of an the inhibitor ganetespib
TO BE PUBLISHED
7GG7
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Group deposition SARS-CoV-2 main protease in complex with inhibitors from the COVID Moonshot -- Crystal Structure of SARS-CoV-2 main protease in complex with CHO-MSK-00c5269a-2 (Mpro-x12177)
分子名称: 2-(1H-benzotriazol-1-yl)-N-[(3-chlorophenyl)methyl]-N-(4-methoxyphenyl)acetamide, 3C-like proteinase, DIMETHYL SULFOXIDE
著者Fearon, D, Aimon, A, Aschenbrenner, J.C, Balcomb, B.H, Bertram, F.K.R, Brandao-Neto, J, Dias, A, Douangamath, A, Dunnett, L, Godoy, A.S, Gorrie-Stone, T.J, Koekemoer, L, Krojer, T, Lithgo, R.M, Lukacik, P, Marples, P.G, Mikolajek, H, Nelson, E, Owen, C.D, Powell, A.J, Rangel, V.L, Skyner, R, Strain-Damerell, C.M, Thompson, W, Tomlinson, C.W.E, Wild, C, Walsh, M.A, von Delft, F.
登録日2023-08-11
公開日2023-11-08
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Science, 382, 2023
7GGM
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BU of 7ggm by Molmil
Group deposition SARS-CoV-2 main protease in complex with inhibitors from the COVID Moonshot -- Crystal Structure of SARS-CoV-2 main protease in complex with MAT-POS-afd4d4fd-2 (Mpro-x12677)
分子名称: 2-(6-chloropyridin-2-yl)-N-(isoquinolin-4-yl)acetamide, 3C-like proteinase, DIMETHYL SULFOXIDE
著者Fearon, D, Aimon, A, Aschenbrenner, J.C, Balcomb, B.H, Bertram, F.K.R, Brandao-Neto, J, Dias, A, Douangamath, A, Dunnett, L, Godoy, A.S, Gorrie-Stone, T.J, Koekemoer, L, Krojer, T, Lithgo, R.M, Lukacik, P, Marples, P.G, Mikolajek, H, Nelson, E, Owen, C.D, Powell, A.J, Rangel, V.L, Skyner, R, Strain-Damerell, C.M, Thompson, W, Tomlinson, C.W.E, Wild, C, Walsh, M.A, von Delft, F.
登録日2023-08-11
公開日2023-11-08
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.839 Å)
主引用文献Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Science, 382, 2023
7GGO
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BU of 7ggo by Molmil
Group deposition SARS-CoV-2 main protease in complex with inhibitors from the COVID Moonshot -- Crystal Structure of SARS-CoV-2 main protease in complex with ALP-POS-8b8a49e1-4 (Mpro-x12682)
分子名称: (4R)-6-chloro-N-[(4R)-2-oxopiperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-4-carboxamide, 3C-like proteinase, DIMETHYL SULFOXIDE
著者Fearon, D, Aimon, A, Aschenbrenner, J.C, Balcomb, B.H, Bertram, F.K.R, Brandao-Neto, J, Dias, A, Douangamath, A, Dunnett, L, Godoy, A.S, Gorrie-Stone, T.J, Koekemoer, L, Krojer, T, Lithgo, R.M, Lukacik, P, Marples, P.G, Mikolajek, H, Nelson, E, Owen, C.D, Powell, A.J, Rangel, V.L, Skyner, R, Strain-Damerell, C.M, Thompson, W, Tomlinson, C.W.E, Wild, C, Walsh, M.A, von Delft, F.
登録日2023-08-11
公開日2023-11-08
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.687 Å)
主引用文献Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Science, 382, 2023
7GGP
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Group deposition SARS-CoV-2 main protease in complex with inhibitors from the COVID Moonshot -- Crystal Structure of SARS-CoV-2 main protease in complex with VLA-UCB-29506327-1 (Mpro-x12686)
分子名称: (1'M,4S)-6-chloro-1'-(isoquinolin-4-yl)-2,3-dihydrospiro[[1]benzopyran-4,4'-imidazolidine]-2',5'-dione, 3C-like proteinase, DIMETHYL SULFOXIDE
著者Fearon, D, Aimon, A, Aschenbrenner, J.C, Balcomb, B.H, Bertram, F.K.R, Brandao-Neto, J, Dias, A, Douangamath, A, Dunnett, L, Godoy, A.S, Gorrie-Stone, T.J, Koekemoer, L, Krojer, T, Lithgo, R.M, Lukacik, P, Marples, P.G, Mikolajek, H, Nelson, E, Owen, C.D, Powell, A.J, Rangel, V.L, Skyner, R, Strain-Damerell, C.M, Thompson, W, Tomlinson, C.W.E, Wild, C, Walsh, M.A, von Delft, F.
登録日2023-08-11
公開日2023-11-08
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.902 Å)
主引用文献Open science discovery of potent noncovalent SARS-CoV-2 main protease inhibitors.
Science, 382, 2023

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件を2024-07-31に公開中

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