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PDB: 1 results

6WIW
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BU of 6wiw by Molmil
c-Src Bound to ATP-Competitive Inhibitor I14
Descriptor: N-(3-{[4-amino-7-(2-methoxyethyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]ethynyl}-4-methylphenyl)acetamide, Proto-oncogene tyrosine-protein kinase Src
Authors:Vilas-Boas, J, Thakur, M.K, Fang, L, Maly, D, Seeliger, M.A.
Deposit date:2020-04-10
Release date:2020-06-17
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:How ATP-Competitive Inhibitors Allosterically Modulate Tyrosine Kinases That Contain a Src-like Regulatory Architecture.
Acs Chem.Biol., 15, 2020

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