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PDB: 9 件

1F7Z
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RAT TRYPSINOGEN K15A COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR
分子名称: CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ...
著者Pasternak, A, White, A, Jeffery, C.J, Medina, N, Cahoon, M, Ringe, D, Hedstrom, L.
登録日2000-06-28
公開日2001-07-04
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity.
Protein Sci., 10, 2001
1FY8
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CRYSTAL STRUCTURE OF THE DELTAILE16VAL17 RAT ANIONIC TRYPSINOGEN-BPTI COMPLEX
分子名称: CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ...
著者Pasternak, A, White, A, Jeffery, C.J, Ringe, D, Hedstrom, L.
登録日2000-09-28
公開日2000-11-08
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity.
Protein Sci., 10, 2001
1F5R
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RAT TRYPSINOGEN MUTANT COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR
分子名称: CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, TRYPSIN II, ...
著者Pasternak, A, White, A, Cahoon, M, Ringe, D, Hedstrom, L.
登録日2000-06-15
公開日2001-07-04
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity.
Protein Sci., 10, 2001
3TGK
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TRYPSINOGEN MUTANT D194N AND DELETION OF ILE 16-VAL 17 COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI)
分子名称: CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ...
著者Pasternak, A, White, A, Jeffery, C.J, Medina, N, Cahoon, M, Ringe, D, Hedstrom, L.
登録日1998-07-19
公開日2001-07-04
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity.
Protein Sci., 10, 2001
3TGI
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BU of 3tgi by Molmil
WILD-TYPE RAT ANIONIC TRYPSIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI)
分子名称: BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ...
著者Pasternak, A, Ringe, D, Hedstrom, L.
登録日1998-07-15
公開日1998-12-23
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Comparison of Anionic and Cationic Trypsinogens: The Anionic Activation Domain is More Flexible in Solution and Differs in its Mode of Bpti Binding in the Crystal Structure
Protein Sci., 8, 1999
3TGJ
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S195A TRYPSINOGEN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR (BPTI)
分子名称: BOVINE PANCREATIC TRYPSIN INHIBITOR, CALCIUM ION, SULFATE ION, ...
著者Pasternak, A, Ringe, D, Hedstrom, L.
登録日1998-07-16
公開日1998-12-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Comparison of Anionic and Cationic Trypsinogens: The Anionic Activation Domain is More Flexible in Solution and Differs in its Mode of Bpti Binding in the Crystal Structure
Protein Sci., 8, 1999
1LSI
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LSIII (NMR, 23 STRUCTURES)
分子名称: LSIII
著者Connolly, P.J, Stern, A.S, Hoch, J.C.
登録日1995-11-26
公開日1996-03-15
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structure of LSIII, a long neurotoxin from the venom of Laticauda semifasciata.
Biochemistry, 35, 1996
3T2N
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Human hepsin protease in complex with the Fab fragment of an inhibitory antibody
分子名称: Antibody, Fab fragment, Heavy Chain, ...
著者Koschubs, T, Dengl, S, Duerr, H, Kaluza, K, Georges, G, Hartl, C, Jennewein, S, Lanzendoerfer, M, Auer, J, Stern, A, Huang, K.-S, Kostrewa, D, Ries, S, Hansen, S, Kohnert, U, Cramer, P, Mundigl, O.
登録日2011-07-22
公開日2011-12-28
最終更新日2012-07-25
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Allosteric antibody inhibition of human hepsin protease.
Biochem.J., 442, 2012
1NPA
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crystal structure of HIV-1 protease-hup
分子名称: (3S)-TETRAHYDROFURAN-3-YL (1R,2S)-3-[4-((1R)-2-{[(S)-AMINO(HYDROXY)METHYL]OXY}-2,3-DIHYDRO-1H-INDEN-1-YL)-2-BENZYL-3-OXOPYRROLIDIN-2-YL]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, POL polyprotein
著者Smith III, A.B, Hirschmann, R, Pasternak, A, Yao, W, Sprengeler, P.A, Holloway, M.K, Kuo, L.C, Chen, Z, Darke, P.L, Schleif, W.A.
登録日2003-01-17
公開日2004-01-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An orally bioavailable pyrrolinone inhibitor of HIV-1 protease: computational analysis and X-ray crystal structure of the enzyme complex.
J.MED.CHEM., 40, 1997

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