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PDB: 9 件

4HHE
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Quinolinate synthase from Pyrococcus furiosus
分子名称: CHLORIDE ION, Quinolinate synthase A
著者Soriano, E.V, Zhang, Y, Settembre, E.C, Colabroy, K, Sanders, J.M, Dorrestein, P.C, Begley, T.P, Ealick, S.E.
登録日2012-10-09
公開日2013-08-28
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.797 Å)
主引用文献Active-site models for complexes of quinolinate synthase with substrates and intermediates.
Acta Crystallogr.,Sect.D, 69, 2013
5LI1
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BU of 5li1 by Molmil
Structure of a Par3-inhibitory peptide bound to PKCiota core kinase domain
分子名称: GLYCEROL, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ...
著者Soriano, E.V, Purkiss, A.G, McDonald, N.Q.
登録日2016-07-13
公開日2016-09-14
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献aPKC Inhibition by Par3 CR3 Flanking Regions Controls Substrate Access and Underpins Apical-Junctional Polarization.
Dev.Cell, 38, 2016
5LIH
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Structure of a peptide-substrate bound to PKCiota core kinase domain
分子名称: ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MANGANESE (II) ION, ...
著者Soriano, E.V, Purkiss, A.G, McDonald, N.Q.
登録日2016-07-14
公開日2016-09-14
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献aPKC Inhibition by Par3 CR3 Flanking Regions Controls Substrate Access and Underpins Apical-Junctional Polarization.
Dev.Cell, 38, 2016
3ZH8
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A novel small molecule aPKC inhibitor
分子名称: (2S)-3-phenyl-N~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine, 1,2-ETHANEDIOL, CHLORIDE ION, ...
著者Kjaer, S, Purkiss, A.G, Kostelecky, B, Knowles, P.P, Soriano, E, Murray-Rust, J, McDonald, N.Q.
登録日2012-12-20
公開日2013-02-27
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.739 Å)
主引用文献Adenosine-Binding Motif Mimicry and Cellular Effects of a Thieno[2,3-D]Pyrimidine-Based Chemical Inhibitor of Atypical Protein Kinase C Isozymes.
Biochem.J., 451, 2013
2QQD
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BU of 2qqd by Molmil
N47A mutant of Pyruvoyl-dependent Arginine Decarboxylase from Methanococcus jannashii
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, AGMATINE, PYRUVIC ACID, ...
著者Ealick, S.E, Soriano, E.S.
登録日2007-07-26
公開日2008-03-18
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of the N47A and E109Q mutant proteins of pyruvoyl-dependent arginine decarboxylase from Methanococcus jannaschii.
Acta Crystallogr.,Sect.D, 64, 2008
2QQC
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E109Q mutant of Pyruvoyl-dependent Arginine Decarboxylase from Methanococcus jannashii
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, AGMATINE, Pyruvoyl-dependent arginine decarboxylase subunit alpha, ...
著者Ealick, S.E, Soriano, E.S.
登録日2007-07-26
公開日2008-03-18
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structures of the N47A and E109Q mutant proteins of pyruvoyl-dependent arginine decarboxylase from Methanococcus jannaschii.
Acta Crystallogr.,Sect.D, 64, 2008
2QRO
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Human Deoxycytidine kinase dAMP, UDP, Mg ion product complex
分子名称: 2'-DEOXYADENOSINE-5'-MONOPHOSPHATE, Deoxycytidine kinase, MAGNESIUM ION, ...
著者Ealick, S.E, Soriano, E.V.
登録日2007-07-28
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Structures of human deoxycytidine kinase product complexes.
Acta Crystallogr.,Sect.D, 63, 2007
2QRN
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Human Deoxycytidine kinase dCMP, UDP, Mg ion product complex
分子名称: 2'-DEOXYCYTIDINE-5'-MONOPHOSPHATE, Deoxycytidine kinase, MAGNESIUM ION, ...
著者Ealick, S.E, Soriano, E.V.
登録日2007-07-28
公開日2007-12-11
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Structures of human deoxycytidine kinase product complexes.
Acta Crystallogr.,Sect.D, 63, 2007
2QRY
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Periplasmic thiamin binding protein
分子名称: THIAMIN PHOSPHATE, Thiamine-binding periplasmic protein
著者Ealick, S.E, Soriano, E.V.
登録日2007-07-30
公開日2008-02-05
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structural Similarities between Thiamin-Binding Protein and Thiaminase-I Suggest a Common Ancestor
Biochemistry, 47, 2008

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件を2024-07-24に公開中

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