1V97
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![BU of 1v97 by Molmil](/molmil-images/mine/1v97) | Crystal Structure of Bovine Milk Xanthine Dehydrogenase FYX-051 bound form | 分子名称: | 4-(5-PYRIDIN-4-YL-1H-1,2,4-TRIAZOL-3-YL)PYRIDINE-2-CARBONITRILE, ACETIC ACID, CALCIUM ION, ... | 著者 | Okamoto, K, Matsumoto, K, Hille, R, Eger, B.T, Pai, E.F, Nishino, T. | 登録日 | 2004-01-21 | 公開日 | 2004-06-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | The crystal structure of xanthine oxidoreductase during catalysis: Implications for reaction mechanism and enzyme inhibition. Proc.Natl.Acad.Sci.USA, 101, 2004
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4YYL
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![BU of 4yyl by Molmil](/molmil-images/mine/4yyl) | Phenolic acid derivative bound to influenza strain H1N1 polymerase subunit PA endonuclease | 分子名称: | 2-(4-fluorophenoxy)-1-(2,3,4-trihydroxyphenyl)ethanone, MANGANESE (II) ION, Polymerase acidic protein, ... | 著者 | Fudo, S, Yamamoto, N, Nukaga, M, Odagiri, T, Tashiro, M, Neya, S, Hoshino, T. | 登録日 | 2015-03-24 | 公開日 | 2015-04-29 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.905 Å) | 主引用文献 | Structural and computational study on inhibitory compounds for endonuclease activity of influenza virus polymerase Bioorg.Med.Chem., 23, 2015
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4ZQQ
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![BU of 4zqq by Molmil](/molmil-images/mine/4zqq) | Apo form of influenza strain H1N1 polymerase acidic subunit N-terminal region | 分子名称: | MANGANESE (II) ION, Polymerase acidic protein,Polymerase acidic protein, SULFATE ION | 著者 | Fudo, S, Yamamoto, N, Nukaga, M, Odagiri, T, Tashiro, M, Neya, S, Hoshino, T. | 登録日 | 2015-05-11 | 公開日 | 2015-06-03 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Two Distinctive Binding Modes of Endonuclease Inhibitors to the N-Terminal Region of Influenza Virus Polymerase Acidic Subunit. Biochemistry, 55, 2016
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4ZI0
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![BU of 4zi0 by Molmil](/molmil-images/mine/4zi0) | Endonuclease inhibitor bound to influenza strain H1N1 polymerase acidic subunit N-terminal region without a chelation to the metal ions in the active site | 分子名称: | 4-{(E)-[2-(4-chlorophenyl)hydrazinylidene]methyl}benzene-1,2,3-triol, MANGANESE (II) ION, Polymerase acidic protein, ... | 著者 | Fudo, S, Yamamoto, N, Nukaga, M, Odagiri, T, Tashiro, M, Neya, S, Hoshino, T. | 登録日 | 2015-04-27 | 公開日 | 2015-05-13 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.802 Å) | 主引用文献 | Two Distinctive Binding Modes of Endonuclease Inhibitors to the N-Terminal Region of Influenza Virus Polymerase Acidic Subunit Biochemistry, 55, 2016
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1VDV
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![BU of 1vdv by Molmil](/molmil-images/mine/1vdv) | Bovine Milk Xanthine Dehydrogenase Y-700 Bound Form | 分子名称: | 1-[3-CYANO-4-(NEOPENTYLOXY)PHENYL]-1H-PYRAZOLE-4-CARBOXYLIC ACID, ACETIC ACID, CALCIUM ION, ... | 著者 | Fukunari, A, Okamoto, K, Nishino, T, Eger, B.T, Pai, E.F, Kamezawa, M, Yamada, I, Kato, N. | 登録日 | 2004-03-25 | 公開日 | 2004-12-21 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Y-700 [1-[3-Cyano-4-(2,2-dimethylpropoxy)phenyl]-1H-pyrazole-4-carboxylic acid]: a potent xanthine oxidoreductase inhibitor with hepatic excretion J.Pharmacol.Exp.Ther., 311, 2004
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6LPG
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![BU of 6lpg by Molmil](/molmil-images/mine/6lpg) | human VASH1-SVBP complex | 分子名称: | SULFATE ION, Small vasohibin-binding protein, Tubulinyl-Tyr carboxypeptidase 1 | 著者 | Ikeda, A, Nishino, T. | 登録日 | 2020-01-10 | 公開日 | 2020-10-21 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The crystal structure of the tetrameric human vasohibin-1-SVBP complex reveals a variable arm region within the structural core. Acta Crystallogr D Struct Biol, 76, 2020
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7D5J
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3AX7
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![BU of 3ax7 by Molmil](/molmil-images/mine/3ax7) | Bovine Xanthine Oxidase, protease cleaved form | 分子名称: | 2-HYDROXYBENZOIC ACID, BICARBONATE ION, CALCIUM ION, ... | 著者 | Ishikita, H, Eger, B.T, Pai, E.F, Okamoto, K, Nishino, T. | 登録日 | 2011-03-30 | 公開日 | 2012-02-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Protein conformational gating of enzymatic activity in xanthine oxidoreductase J.Am.Chem.Soc., 134, 2012
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3AX9
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![BU of 3ax9 by Molmil](/molmil-images/mine/3ax9) | Bovine xanthine oxidase, protease cleaved form | 分子名称: | 2-HYDROXYBENZOIC ACID, BICARBONATE ION, CALCIUM ION, ... | 著者 | Ishikita, H, Eger, B.T, Pai, E.F, Okamoto, K, Nishino, T. | 登録日 | 2011-03-31 | 公開日 | 2012-02-22 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Protein conformational gating of enzymatic activity in xanthine oxidoreductase J.Am.Chem.Soc., 134, 2012
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1QQ2
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![BU of 1qq2 by Molmil](/molmil-images/mine/1qq2) | CRYSTAL STRUCTURE OF A MAMMALIAN 2-CYS PEROXIREDOXIN, HBP23. | 分子名称: | CHLORIDE ION, THIOREDOXIN PEROXIDASE 2 | 著者 | Hirotsu, S, Abe, Y, Okada, K, Nagahara, N, Hori, H, Nishino, T, Hakoshima, T. | 登録日 | 1999-06-10 | 公開日 | 1999-10-29 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystal structure of a multifunctional 2-Cys peroxiredoxin heme-binding protein 23 kDa/proliferation-associated gene product. Proc.Natl.Acad.Sci.USA, 96, 1999
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8JYH
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![BU of 8jyh by Molmil](/molmil-images/mine/8jyh) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with laccaic acid C | 分子名称: | 7-[5-[(2~{S})-2-azanyl-3-oxidanyl-3-oxidanylidene-propyl]-2-oxidanyl-phenyl]-3,5,6,8-tetrakis(oxidanyl)-9,10-bis(oxidanylidene)anthracene-1,2-dicarboxylic acid, MANGANESE (II) ION, Pol protein,Pol protein,HIV-1 Reverse Transcriptase RNase H active domain, ... | 著者 | Ito, Y, Lu, H, Kitajima, M, Ishikawa, H, Nakata, Y, Iwatani, Y, Hoshino, T. | 登録日 | 2023-07-03 | 公開日 | 2023-08-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Sticklac-Derived Natural Compounds Inhibiting RNase H Activity of HIV-1 Reverse Transcriptase. J.Nat.Prod., 86, 2023
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8JYJ
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![BU of 8jyj by Molmil](/molmil-images/mine/8jyj) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with laccaic acid A | 分子名称: | 7-[5-(2-acetamidoethyl)-2-oxidanyl-phenyl]-3,5,6,8-tetrakis(oxidanyl)-9,10-bis(oxidanylidene)anthracene-1,2-dicarboxylic acid, MANGANESE (II) ION, Pol protein,Pol protein,HIV-1 Reverse Transcriptase RNase H active domain, ... | 著者 | Ito, Y, Lu, H, Kitajima, M, Ishikawa, H, Nakata, Y, Iwatani, Y, Hoshino, T. | 登録日 | 2023-07-03 | 公開日 | 2023-08-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Sticklac-Derived Natural Compounds Inhibiting RNase H Activity of HIV-1 Reverse Transcriptase. J.Nat.Prod., 86, 2023
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8JYI
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![BU of 8jyi by Molmil](/molmil-images/mine/8jyi) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with laccaic acid E | 分子名称: | 7-[5-(2-azanylethyl)-2-oxidanyl-phenyl]-3,5,6,8-tetrakis(oxidanyl)-9,10-bis(oxidanylidene)anthracene-1,2-dicarboxylic acid, MANGANESE (II) ION, Pol protein,Pol protein,Ribonuclease H, ... | 著者 | Ito, Y, Lu, H, Kitajima, M, Ishikawa, H, Nakata, Y, Iwatani, Y, Hoshino, T. | 登録日 | 2023-07-03 | 公開日 | 2023-08-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Sticklac-Derived Natural Compounds Inhibiting RNase H Activity of HIV-1 Reverse Transcriptase. J.Nat.Prod., 86, 2023
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2RQH
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![BU of 2rqh by Molmil](/molmil-images/mine/2rqh) | Structure of GSPT1/ERF3A-PABC | 分子名称: | G1 to S phase transition 1, Polyadenylate-binding protein 1 | 著者 | Osawa, M, Nakanishi, T, Hosoda, N, Uchida, S, Hoshino, T, Katada, I, Shimada, I. | 登録日 | 2009-05-08 | 公開日 | 2010-05-26 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Eukaryotic Translation Termination Factor Gspt/Erf3 Recognizes Pabp with Chemical Exchange Using Two Overlapping Motifs To be Published
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3AM9
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![BU of 3am9 by Molmil](/molmil-images/mine/3am9) | Complex of bovine xanthine dehydrogenase and trihydroxy FYX-051 | 分子名称: | 4-[5-(2,6-dioxo-1,2,3,6-tetrahydropyridin-4-yl)-1H-1,2,4-triazol-3-yl]-6-oxo-1,6-dihydropyridine-2-carbonitrile, BICARBONATE ION, CALCIUM ION, ... | 著者 | Matsumoto, K, Okamoto, K, Ashizawa, N, Matsumura, T, Kusano, T, Nishino, T. | 登録日 | 2010-08-18 | 公開日 | 2010-11-03 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.17 Å) | 主引用文献 | FYX-051: A Novel and Potent Hybrid-Type Inhibitor of Xanthine Oxidoreductase J.Pharmacol.Exp.Ther., 336, 2011
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2RQG
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![BU of 2rqg by Molmil](/molmil-images/mine/2rqg) | Structure of GSPT1/ERF3A-PABC | 分子名称: | G1 to S phase transition 1, Polyadenylate-binding protein 1 | 著者 | Osawa, M, Nakanishi, T, Hosoda, N, Uchida, S, Hoshino, T, Katada, I, Shimada, I. | 登録日 | 2009-05-08 | 公開日 | 2010-05-26 | 最終更新日 | 2024-05-15 | 実験手法 | SOLUTION NMR | 主引用文献 | Eukaryotic Translation Termination Factor Gspt/Erf3 Recognizes Pabp with Chemical Exchange Using Two Overlapping Motifs To be Published
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3AN1
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![BU of 3an1 by Molmil](/molmil-images/mine/3an1) | Crystal structure of rat D428A mutant, urate bound form | 分子名称: | BICARBONATE ION, CALCIUM ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Okamoto, K, Kawaguchi, Y, Eger, B.T, Pai, E.F, Nishino, T. | 登録日 | 2010-08-27 | 公開日 | 2010-12-01 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Crystal Structures of Urate Bound Form of Xanthine Oxidoreductase: Substrate Orientation and Structure of the Key Reaction Intermediate J.Am.Chem.Soc., 132, 2010
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3AMZ
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![BU of 3amz by Molmil](/molmil-images/mine/3amz) | Bovine Xanthine Oxidoreductase urate bound form | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, BICARBONATE ION, CALCIUM ION, ... | 著者 | Okamoto, K, Eger, B.T, Pai, E.F, Nishino, T. | 登録日 | 2010-08-27 | 公開日 | 2010-12-01 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal Structures of Urate Bound Form of Xanthine Oxidoreductase: Substrate Orientation and Structure of the Key Reaction Intermediate J.Am.Chem.Soc., 132, 2010
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1SIO
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![BU of 1sio by Molmil](/molmil-images/mine/1sio) | Structure of Kumamolisin-As complexed with a covalently-bound inhibitor, AcIPF | 分子名称: | Ace-ILE-PRO-PHL peptide inhibitor, CALCIUM ION, SULFATE ION, ... | 著者 | Li, M, Wlodawer, A, Gustchina, A, Tsuruoka, N, Ashida, M, Minakata, H, Oyama, H, Oda, K, Nishino, T, Nakayama, T. | 登録日 | 2004-03-01 | 公開日 | 2004-03-30 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystallographic and biochemical investigations of kumamolisin-As, a serine-carboxyl peptidase with collagenase activity J.Biol.Chem., 279, 2004
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1SIU
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![BU of 1siu by Molmil](/molmil-images/mine/1siu) | KUMAMOLISIN-AS E78H MUTANT | 分子名称: | CALCIUM ION, SULFATE ION, kumamolisin-As | 著者 | Li, M, Wlodawer, A, Gustchina, A, Tsuruoka, N, Ashida, M, Minakata, H, Oyama, H, Oda, K, Nishino, T, Nakayama, T. | 登録日 | 2004-03-01 | 公開日 | 2004-03-30 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Crystallographic and biochemical investigations of kumamolisin-As, a serine-carboxyl peptidase with collagenase activity J.Biol.Chem., 279, 2004
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7XGC
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![BU of 7xgc by Molmil](/molmil-images/mine/7xgc) | |
7XGQ
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![BU of 7xgq by Molmil](/molmil-images/mine/7xgq) | |
7XIU
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![BU of 7xiu by Molmil](/molmil-images/mine/7xiu) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with nitrofuran methoxy(methoxycarbonyl)phenyl ester | 分子名称: | MANGANESE (II) ION, Reverse Transcriptase RNase H domain, ZINC ION, ... | 著者 | Lu, H, Komukai, Y, Usami, K, Guo, Y, Qiao, X, Nukaga, M, Hoshino, T. | 登録日 | 2022-04-14 | 公開日 | 2022-04-27 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Computational and Crystallographic Analysis of Binding Structures of Inhibitory Compounds for HIV-1 RNase H Activity. J.Chem.Inf.Model., 62, 2022
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7XIT
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![BU of 7xit by Molmil](/molmil-images/mine/7xit) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with nitrofuran methoxy(methoxycarbonyl)phenyl ester | 分子名称: | MANGANESE (II) ION, Reverse Transcriptase RNase H domain, ZINC ION, ... | 著者 | Lu, H, Komukai, Y, Usami, K, Guo, Y, Qiao, X, Nukaga, M, Hoshino, T. | 登録日 | 2022-04-14 | 公開日 | 2022-04-27 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Computational and Crystallographic Analysis of Binding Structures of Inhibitory Compounds for HIV-1 RNase H Activity. J.Chem.Inf.Model., 62, 2022
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7XJ5
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![BU of 7xj5 by Molmil](/molmil-images/mine/7xj5) | Crystal structure of engineered HIV-1 Reverse Transcriptase RNase H domain complexed with nitrofuran methoxy(methoxycarbonyl)phenyl ester | 分子名称: | MANGANESE (II) ION, Reverse Transcriptase RNase H domain, ZINC ION, ... | 著者 | Lu, H, Komukai, Y, Usami, K, Guo, Y, Qiao, X, Nukaga, M, Hoshino, T. | 登録日 | 2022-04-15 | 公開日 | 2022-04-27 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Computational and Crystallographic Analysis of Binding Structures of Inhibitory Compounds for HIV-1 RNase H Activity. J.Chem.Inf.Model., 62, 2022
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