1VA5
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![BU of 1va5 by Molmil](/molmil-images/mine/1va5) | Antigen 85C with octylthioglucoside in active site | 分子名称: | Antigen 85-C, octyl 1-thio-beta-D-glucopyranoside | 著者 | Ronning, D.R, Vissa, V, Besra, G.S, Belisle, J.T, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2004-02-11 | 公開日 | 2004-07-06 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.02 Å) | 主引用文献 | Mycobacterium tuberculosis Antigen 85A and 85C Structures Confirm Binding Orientation and Conserved Substrate Specificity J.Biol.Chem., 279, 2004
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4U3C
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![BU of 4u3c by Molmil](/molmil-images/mine/4u3c) | Docking Site of Maltohexaose in the Mtb GlgE | 分子名称: | Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Ronning, D.R, Lindenberger, J.J. | 登録日 | 2014-07-19 | 公開日 | 2015-07-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.98 Å) | 主引用文献 | Crystal structures of Mycobacterium tuberculosis GlgE and complexes with non-covalent inhibitors. Sci Rep, 5, 2015
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4U33
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![BU of 4u33 by Molmil](/molmil-images/mine/4u33) | Structure of Mtb GlgE bound to maltose | 分子名称: | Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Ronning, D.R, Lindenberger, J.J. | 登録日 | 2014-07-18 | 公開日 | 2015-07-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.293 Å) | 主引用文献 | Crystal structures of Mycobacterium tuberculosis GlgE and complexes with non-covalent inhibitors. Sci Rep, 5, 2015
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4U31
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![BU of 4u31 by Molmil](/molmil-images/mine/4u31) | Sco GlgEI-V279S in Complex with maltose-C-phosphonate | 分子名称: | 1,2-ETHANEDIOL, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, CITRIC ACID, ... | 著者 | Ronning, D.R, Lindenberger, J.J. | 登録日 | 2014-07-18 | 公開日 | 2015-07-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.849 Å) | 主引用文献 | Crystal structures of Mycobacterium tuberculosis GlgE and complexes with non-covalent inhibitors. Sci Rep, 5, 2015
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4U2Z
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![BU of 4u2z by Molmil](/molmil-images/mine/4u2z) | X-ray crystal structure of an Sco GlgEI-V279S/1,2,2-trifluromaltose complex | 分子名称: | Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1, alpha-D-glucopyranose-(1-4)-2-deoxy-2,2-difluoro-alpha-D-arabino-hexopyranosyl fluoride | 著者 | Ronning, D.R, Lindenberger, J.J. | 登録日 | 2014-07-18 | 公開日 | 2015-07-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.26 Å) | 主引用文献 | Synthesis of 2-deoxy-2,2-difluoro-alpha-maltosyl fluoride and its X-ray structure in complex with Streptomyces coelicolor GlgEI-V279S. Org.Biomol.Chem., 13, 2015
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4U2Y
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![BU of 4u2y by Molmil](/molmil-images/mine/4u2y) | Sco GlgEI-V279S in Complex with Reaction Intermediate Azasugar | 分子名称: | (2R,3R,4R,5R)-4-hydroxy-2,5-bis(hydroxymethyl)pyrrolidin-3-yl alpha-D-glucopyranoside, Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase 1 | 著者 | Ronning, D.R, Lindenberger, J.J. | 登録日 | 2014-07-18 | 公開日 | 2015-08-12 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.483 Å) | 主引用文献 | Crystal structures of Mycobacterium tuberculosis GlgE and complexes with non-covalent inhibitors. Sci Rep, 5, 2015
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2A6O
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![BU of 2a6o by Molmil](/molmil-images/mine/2a6o) | Crystal Structure of the ISHp608 Transposase in Complex with Stem-loop DNA | 分子名称: | 5'-D(*CP*CP*CP*CP*TP*AP*GP*CP*TP*TP*TP*AP*GP*CP*TP*AP*TP*GP*GP*GP*GP*A)-3', ISHp608 Transposase | 著者 | Ronning, D.R, Guynet, C, Ton-Hoang, B, Perez, Z.N, Ghirlando, R, Chandler, M, Dyda, F. | 登録日 | 2005-07-03 | 公開日 | 2005-10-25 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Active site sharing and subterminal hairpin recognition in a new class of DNA transposases. Mol.Cell, 20, 2005
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1T0F
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![BU of 1t0f by Molmil](/molmil-images/mine/1t0f) | Crystal Structure of the TnsA/TnsC(504-555) complex | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, MAGNESIUM ION, MALONIC ACID, ... | 著者 | Ronning, D.R, Li, Y, Perez, Z.N, Ross, P.D, Hickman, A.B, Craig, N.L, Dyda, F. | 登録日 | 2004-04-08 | 公開日 | 2004-11-09 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | The carboxy-terminal portion of TnsC activates the Tn7 transposase through a specific interaction with TnsA. Embo J., 23, 2004
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1DQY
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![BU of 1dqy by Molmil](/molmil-images/mine/1dqy) | CRYSTAL STRUCTURE OF ANTIGEN 85C FROM MYCOBACTERIUM TUBERCULOSIS WITH DIETHYL PHOSPHATE INHIBITOR | 分子名称: | (4R)-2-METHYLPENTANE-2,4-DIOL, DIETHYL PHOSPHONATE, PROTEIN (ANTIGEN 85-C) | 著者 | Ronning, D.R, Klabunde, T, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2000-01-05 | 公開日 | 2000-07-12 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Crystal structure of the secreted form of antigen 85C reveals potential targets for mycobacterial drugs and vaccines. Nat.Struct.Biol., 7, 2000
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1DQZ
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![BU of 1dqz by Molmil](/molmil-images/mine/1dqz) | |
1SFR
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![BU of 1sfr by Molmil](/molmil-images/mine/1sfr) | Crystal Structure of the Mycobacterium tuberculosis Antigen 85A Protein | 分子名称: | Antigen 85-A | 著者 | Ronning, D.R, Vissa, V, Besra, G.S, Belisle, J.T, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2004-02-20 | 公開日 | 2004-07-06 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Mycobacterium tuberculosis Antigen 85A and 85C Structures Confirm Binding Orientation and Conserved Substrate Specificity J.Biol.Chem., 279, 2004
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2A6M
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![BU of 2a6m by Molmil](/molmil-images/mine/2a6m) | Crystal Structure of the ISHp608 Transposase | 分子名称: | ISHp608 transposase | 著者 | Ronning, D.R, Guynet, C, Ton-Hoang, B, Perez, Z.N, Ghirlando, R, Chandler, M, Dyda, F. | 登録日 | 2005-07-03 | 公開日 | 2005-10-25 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Active site sharing and subterminal hairpin recognition in a new class of DNA transposases. Mol.Cell, 20, 2005
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3NM5
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![BU of 3nm5 by Molmil](/molmil-images/mine/3nm5) | Helicobacter pylori MTAN complexed with Formycin A | 分子名称: | (1S)-1-(7-amino-1H-pyrazolo[4,3-d]pyrimidin-3-yl)-1,4-anhydro-D-ribitol, MTA/SAH nucleosidase | 著者 | Ronning, D.R, Iacopelli, N.M. | 登録日 | 2010-06-21 | 公開日 | 2010-11-24 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Enzyme-ligand interactions that drive active site rearrangements in the Helicobacter pylori 5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase. Protein Sci., 19, 2010
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3NM4
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![BU of 3nm4 by Molmil](/molmil-images/mine/3nm4) | Helicobacter pylori MTAN | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, MTA/SAH nucleosidase | 著者 | Ronning, D.R, Iacopelli, N.M. | 登録日 | 2010-06-21 | 公開日 | 2010-11-24 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Enzyme-ligand interactions that drive active site rearrangements in the Helicobacter pylori 5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase. Protein Sci., 19, 2010
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3NM6
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![BU of 3nm6 by Molmil](/molmil-images/mine/3nm6) | Helicobacter pylori MTAN complexed with adenine and tris | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ADENINE, ... | 著者 | Ronning, D.R, Iacopelli, N.M. | 登録日 | 2010-06-21 | 公開日 | 2010-11-24 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.602 Å) | 主引用文献 | Enzyme-ligand interactions that drive active site rearrangements in the Helicobacter pylori 5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase. Protein Sci., 19, 2010
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4P54
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![BU of 4p54 by Molmil](/molmil-images/mine/4p54) | |
4V0X
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![BU of 4v0x by Molmil](/molmil-images/mine/4v0x) | The crystal structure of mouse PP1G in complex with truncated human PPP1R15B (631-684) | 分子名称: | MANGANESE (II) ION, PROTEIN PHOSPHATASE 1 REGULATORY SUBUNIT 15B, PROTEIN PHOSPHATASE PP1-GAMMA CATALYTIC SUBUNIT | 著者 | Chen, R, Yan, Y, Casado, A.C, Ron, D, Read, R.J. | 登録日 | 2014-09-18 | 公開日 | 2015-03-25 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | G-actin provides substrate-specificity to eukaryotic initiation factor 2 alpha holophosphatases. Elife, 4, 2015
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1M55
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![BU of 1m55 by Molmil](/molmil-images/mine/1m55) | Catalytic domain of the Adeno Associated Virus type 5 Rep protein | 分子名称: | CHLORIDE ION, Rep protein, ZINC ION | 著者 | Hickman, A.B, Ronning, D.R, Kotin, R.M, Dyda, F. | 登録日 | 2002-07-08 | 公開日 | 2002-08-28 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Structural unity among viral origin binding proteins: crystal structure of the nuclease domain of adeno-associated virus Rep. Mol.Cell, 10, 2002
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1UUT
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![BU of 1uut by Molmil](/molmil-images/mine/1uut) | The Nuclease Domain of Adeno-Associated Virus Rep Complexed with the RBE' Stemloop of the Viral Inverted Terminal Repeat | 分子名称: | 5'-D(*CP*AP*GP*CP*TP*CP*TP*TP*TP*GP *AP*GP*CP*TP*G)-3', CHLORIDE ION, MAGNESIUM ION, ... | 著者 | Dyda, F, Hickman, A.B, Ronning, D.R, Perez, Z.N, Kotin, R.M. | 登録日 | 2004-01-10 | 公開日 | 2004-02-19 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The Nuclease Domain of Adeno-Associated Virus Rep Coordinates Replication Initiation Using Two Distinct DNA Recognition Interfaces Mol.Cell, 13, 2004
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7SEX
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![BU of 7sex by Molmil](/molmil-images/mine/7sex) | M. tb EgtD in complex with TGX221 | 分子名称: | 7-methyl-2-morpholin-4-yl-9-[(1~{R})-1-phenylazanylethyl]-3~{H}-pyrido[1,2-a]pyrimidin-4-one, GLYCEROL, Histidine N-alpha-methyltransferase | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-10-02 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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7SF5
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![BU of 7sf5 by Molmil](/molmil-images/mine/7sf5) | M. tb EgtD in complex with HD3 | 分子名称: | Histidine N-alpha-methyltransferase, N-(benzylcarbamothioyl)-L-histidine | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-10-03 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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7SF4
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![BU of 7sf4 by Molmil](/molmil-images/mine/7sf4) | M. tb EgtD in complex with imatinib | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-4-PYRIDYL-PYRIMIDINE, GLYCEROL, ... | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-10-03 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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7SCF
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![BU of 7scf by Molmil](/molmil-images/mine/7scf) | M. tb EgtD in complex with HD2 | 分子名称: | (2S)-3-(1H-imidazol-5-yl)-2-(1H-pyrrol-1-yl)propanoic acid, DI(HYDROXYETHYL)ETHER, GLYCEROL, ... | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-09-28 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.67 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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7SEW
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![BU of 7sew by Molmil](/molmil-images/mine/7sew) | M. tb EgtD in complex with HD6 | 分子名称: | 1,3-PROPANDIOL, GLYCEROL, Histidine N-alpha-methyltransferase, ... | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-10-02 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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7SEY
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![BU of 7sey by Molmil](/molmil-images/mine/7sey) | M. tb EgtD in complex with SGH | 分子名称: | 2-amino-1-[(3S)-3-methyl-4-(4-methylisoquinoline-5-sulfonyl)-1,4-diazepan-1-yl]ethan-1-one, Histidine N-alpha-methyltransferase | 著者 | Sudasinghe, T.D, Ronning, D.R. | 登録日 | 2021-10-02 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Inhibitors of Mycobacterium tuberculosis EgtD target both substrate binding sites to limit hercynine production. Sci Rep, 11, 2021
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