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PDB: 11 件

4TW9
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BU of 4tw9 by Molmil
Difluoro-dioxolo-benzoimidazol-benzamides as potent inhibitors of CK1delta and epsilon with nanomolar inhibitory activity on cancer cell proliferation
分子名称: CHLORIDE ION, Casein kinase I isoform delta, N-(2,2-difluoro-5H-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide, ...
著者Richter, J, Bischof, J, Zaja, M, Kohlhof, H, Othersen, O, Vitt, D, Alscher, V, Pospiech, I, Garcia-Reyes, B, Berg, S, Leban, J, Knippschild, U.
登録日2014-06-30
公開日2014-07-30
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Difluoro-dioxolo-benzoimidazol-benzamides As Potent Inhibitors of CK1 delta and epsilon with Nanomolar Inhibitory Activity on Cancer Cell Proliferation.
J.Med.Chem., 57, 2014
5CK7
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BU of 5ck7 by Molmil
Mouse ADP-dependent Glucokinase; AMP bound
分子名称: ADENOSINE MONOPHOSPHATE, ADP-dependent glucokinase
著者Richter, J.P, Ronimus, R.S, Sutherland-Smith, A.J.
登録日2015-07-15
公開日2015-11-18
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献The Structural and Functional Characterization of Mammalian ADP-dependent Glucokinase.
J.Biol.Chem., 291, 2016
5CCF
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Structure of Mouse ADP-Dependent Glucokinase
分子名称: ADP-dependent glucokinase
著者Richter, J.P, Ronimus, R.S, Sutherland-Smith, A.J.
登録日2015-07-02
公開日2015-11-18
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Structural and Functional Characterization of Mammalian ADP-dependent Glucokinase.
J.Biol.Chem., 291, 2016
2XGC
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BU of 2xgc by Molmil
Crystal structure of a designed heterodimeric variant T-A(I)B of the tetracycline repressor
分子名称: TETRACYCLINE REPRESSOR PROTEIN CLASS B FROM TRANSPOSON TN10, TETRACYCLINE REPRESSOR PROTEIN CLASS D
著者Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A.
登録日2010-06-03
公開日2010-09-22
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer.
J.Mol.Biol., 403, 2010
2XGD
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BU of 2xgd by Molmil
Crystal structure of a designed homodimeric variant T-A(L)A(L) of the tetracycline repressor
分子名称: CHLORIDE ION, TETRACYCLINE REPRESSOR PROTEIN CLASS B FROM TRANSPOSON TN10, TETRACYCLINE REPRESSOR PROTEIN CLASS D
著者Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A.
登録日2010-06-03
公開日2010-09-22
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer.
J.Mol.Biol., 403, 2010
2XGE
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BU of 2xge by Molmil
Crystal structure of a designed heterodimeric variant T-A(A)B of the tetracycline repressor
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, SODIUM ION, ...
著者Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A.
登録日2010-06-03
公開日2010-09-22
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer.
J.Mol.Biol., 403, 2010
1YRF
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BU of 1yrf by Molmil
Chicken villin subdomain HP-35, N68H, pH6.7
分子名称: ACETATE ION, SULFATE ION, Villin
著者Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R.
登録日2005-02-03
公開日2005-05-03
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.07 Å)
主引用文献High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein.
Proc.Natl.Acad.Sci.Usa, 102, 2005
2F4K
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BU of 2f4k by Molmil
Chicken villin subdomain HP-35, K65(NLE), N68H, K70(NLE), PH9
分子名称: Villin-1
著者Chiu, T.K, Davies, D.R, Kubelka, J, Hofrichter, J, Eaton, W.A.
登録日2005-11-23
公開日2006-04-11
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.05 Å)
主引用文献Sub-microsecond Protein Folding.
J.Mol.Biol., 359, 2006
1YRI
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BU of 1yri by Molmil
Chicken villin subdomain HP-35, N68H, pH6.4
分子名称: ACETATE ION, IODIDE ION, Villin
著者Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R.
登録日2005-02-03
公開日2005-05-03
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein.
Proc.Natl.Acad.Sci.Usa, 102, 2005
1WY4
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BU of 1wy4 by Molmil
Chicken villin subdomain HP-35, K65(NLE), N68H, pH5.1
分子名称: IODIDE ION, SODIUM ION, Villin
著者Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R.
登録日2005-02-04
公開日2005-05-03
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein.
Proc.Natl.Acad.Sci.Usa, 102, 2005
1WY3
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BU of 1wy3 by Molmil
Chicken villin subdomain HP-35, K65(NLE), N68H, pH7.0
分子名称: Villin
著者Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R.
登録日2005-02-04
公開日2005-05-03
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (0.95 Å)
主引用文献High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein.
Proc.Natl.Acad.Sci.Usa, 102, 2005

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