4TW9
| Difluoro-dioxolo-benzoimidazol-benzamides as potent inhibitors of CK1delta and epsilon with nanomolar inhibitory activity on cancer cell proliferation | 分子名称: | CHLORIDE ION, Casein kinase I isoform delta, N-(2,2-difluoro-5H-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide, ... | 著者 | Richter, J, Bischof, J, Zaja, M, Kohlhof, H, Othersen, O, Vitt, D, Alscher, V, Pospiech, I, Garcia-Reyes, B, Berg, S, Leban, J, Knippschild, U. | 登録日 | 2014-06-30 | 公開日 | 2014-07-30 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Difluoro-dioxolo-benzoimidazol-benzamides As Potent Inhibitors of CK1 delta and epsilon with Nanomolar Inhibitory Activity on Cancer Cell Proliferation. J.Med.Chem., 57, 2014
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5CK7
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5CCF
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2XGC
| Crystal structure of a designed heterodimeric variant T-A(I)B of the tetracycline repressor | 分子名称: | TETRACYCLINE REPRESSOR PROTEIN CLASS B FROM TRANSPOSON TN10, TETRACYCLINE REPRESSOR PROTEIN CLASS D | 著者 | Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A. | 登録日 | 2010-06-03 | 公開日 | 2010-09-22 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer. J.Mol.Biol., 403, 2010
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2XGD
| Crystal structure of a designed homodimeric variant T-A(L)A(L) of the tetracycline repressor | 分子名称: | CHLORIDE ION, TETRACYCLINE REPRESSOR PROTEIN CLASS B FROM TRANSPOSON TN10, TETRACYCLINE REPRESSOR PROTEIN CLASS D | 著者 | Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A. | 登録日 | 2010-06-03 | 公開日 | 2010-09-22 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer. J.Mol.Biol., 403, 2010
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2XGE
| Crystal structure of a designed heterodimeric variant T-A(A)B of the tetracycline repressor | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, SODIUM ION, ... | 著者 | Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A. | 登録日 | 2010-06-03 | 公開日 | 2010-09-22 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer. J.Mol.Biol., 403, 2010
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1YRF
| Chicken villin subdomain HP-35, N68H, pH6.7 | 分子名称: | ACETATE ION, SULFATE ION, Villin | 著者 | Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R. | 登録日 | 2005-02-03 | 公開日 | 2005-05-03 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.07 Å) | 主引用文献 | High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein. Proc.Natl.Acad.Sci.Usa, 102, 2005
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2F4K
| Chicken villin subdomain HP-35, K65(NLE), N68H, K70(NLE), PH9 | 分子名称: | Villin-1 | 著者 | Chiu, T.K, Davies, D.R, Kubelka, J, Hofrichter, J, Eaton, W.A. | 登録日 | 2005-11-23 | 公開日 | 2006-04-11 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Sub-microsecond Protein Folding. J.Mol.Biol., 359, 2006
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1YRI
| Chicken villin subdomain HP-35, N68H, pH6.4 | 分子名称: | ACETATE ION, IODIDE ION, Villin | 著者 | Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R. | 登録日 | 2005-02-03 | 公開日 | 2005-05-03 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein. Proc.Natl.Acad.Sci.Usa, 102, 2005
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1WY4
| Chicken villin subdomain HP-35, K65(NLE), N68H, pH5.1 | 分子名称: | IODIDE ION, SODIUM ION, Villin | 著者 | Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R. | 登録日 | 2005-02-04 | 公開日 | 2005-05-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein. Proc.Natl.Acad.Sci.Usa, 102, 2005
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1WY3
| Chicken villin subdomain HP-35, K65(NLE), N68H, pH7.0 | 分子名称: | Villin | 著者 | Chiu, T.K, Kubelka, J, Herbst-Irmer, R, Eaton, W.A, Hofrichter, J, Davies, D.R. | 登録日 | 2005-02-04 | 公開日 | 2005-05-03 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (0.95 Å) | 主引用文献 | High-resolution x-ray crystal structures of the villin headpiece subdomain, an ultrafast folding protein. Proc.Natl.Acad.Sci.Usa, 102, 2005
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