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PDB: 497 件

8H46
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Blasnase-T13A/P55N with L-asn
分子名称: ASPARAGINE, FORMIC ACID, GLYCEROL, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H47
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BU of 8h47 by Molmil
Blasnase-T13A/P55F
分子名称: FORMIC ACID, GLYCEROL, L-asparaginase, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4B
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BU of 8h4b by Molmil
Blasnase-T13A/M57P with L-asn
分子名称: ASPARAGINE, FORMIC ACID, L-asparaginase, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4D
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BU of 8h4d by Molmil
Blasnase-T13A/M57N
分子名称: FORMIC ACID, GLYCEROL, L-asparaginase, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H44
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BU of 8h44 by Molmil
Blasnase-P55N
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H45
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BU of 8h45 by Molmil
Blasnase-T13A/P55N
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H48
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BU of 8h48 by Molmil
Blasnase-T13A/P55F with L-asn
分子名称: ASPARAGINE, FORMIC ACID, L-asparaginase, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H49
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BU of 8h49 by Molmil
Blasnase-M57P
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4A
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BU of 8h4a by Molmil
Blasnase-T13A/M57P
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4C
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BU of 8h4c by Molmil
Blasnase-T13A/M57P
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4G
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BU of 8h4g by Molmil
Blasnase-T13A/M57N
分子名称: FORMIC ACID, L-asparaginase, MAGNESIUM ION
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-10-18
実験手法X-RAY DIFFRACTION (1.81 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
8H4F
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BU of 8h4f by Molmil
Blasnase-T13A/P55F with D-asn
分子名称: D-ASPARAGINE, FORMIC ACID, L-asparaginase, ...
著者Lu, F, Wang, W, Chi, H, Ran, T.
登録日2022-10-10
公開日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme
To Be Published
1EQU
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BU of 1equ by Molmil
TYPE 1 17-BETA HYDROXYSTEROID DEHYDROGENASE EQUILIN COMPLEXED WITH NADP+
分子名称: EQUILIN, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, PROTEIN (ESTRADIOL 17 BETA-DEHYDROGENASE 1)
著者Sawicki, M.W, Erman, M, Puranen, T, Vihko, P, Ghosh, D.
登録日1998-12-02
公開日1999-12-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of the ternary complex of human 17beta-hydroxysteroid dehydrogenase type 1 with 3-hydroxyestra-1,3,5,7-tetraen-17-one (equilin) and NADP+.
Proc.Natl.Acad.Sci.USA, 96, 1999
8IVM
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BU of 8ivm by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-28
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
8IVS
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BU of 8ivs by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-28
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.52 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
7E2P
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BU of 7e2p by Molmil
The Crystal Structure of Mycoplasma bovis enolase
分子名称: Enolase
著者Chen, R, Zhang, S, Gan, R, Wang, W, Ran, T, Shao, G, Xiong, Q, Feng, Z.
登録日2021-02-07
公開日2022-02-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Evidence for the Rapid and Divergent Evolution of Mycoplasmas: Structural and Phylogenetic Analysis of Enolases.
Front Mol Biosci, 8, 2022
8IW6
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BU of 8iw6 by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-29
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
8IW3
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BU of 8iw3 by Molmil
crystal structure of SulE mutant
分子名称: 2-[[[[(4-CHLORO-6-METHOXY-2-PYRIMIDINYL)AMINO]CARBONYL]AMINO]SULFONYL]BENZOIC ACID ETHYL ESTER, Alpha/beta fold hydrolase, GLYCEROL, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-29
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
8IVE
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BU of 8ive by Molmil
crystal structure of SulE mutant
分子名称: 2-[[[[(4-CHLORO-6-METHOXY-2-PYRIMIDINYL)AMINO]CARBONYL]AMINO]SULFONYL]BENZOIC ACID ETHYL ESTER, Alpha/beta fold hydrolase, GLYCEROL
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-27
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
8IVN
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BU of 8ivn by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-28
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
8IVT
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BU of 8ivt by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-28
公開日2023-08-02
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Crystal structures of herbicide-detoxifying esterase reveal a lid loop affecting substrate binding and activity.
Nat Commun, 14, 2023
7E2Q
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BU of 7e2q by Molmil
Crystal structure of Mycoplasma pneumoniae Enolase
分子名称: Enolase, SULFATE ION
著者Chen, R, Zhang, S, Gan, R, Wang, W, Ran, T, Xiong, Q, Shao, G, Feng, Z.
登録日2021-02-07
公開日2022-02-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Evidence for the Rapid and Divergent Evolution of Mycoplasmas: Structural and Phylogenetic Analysis of Enolases.
Front Mol Biosci, 8, 2022
8H0M
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BU of 8h0m by Molmil
Crystal structure of VioD
分子名称: (2S)-2-ethylhexan-1-ol, FLAVIN-ADENINE DINUCLEOTIDE, FORMIC ACID, ...
著者Xu, M, Ran, T, Wang, W.
登録日2022-09-29
公開日2023-04-12
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.702 Å)
主引用文献Structural basis for substrate binding and catalytic mechanism of the key enzyme VioD in the violacein synthesis pathway.
Proteins, 91, 2023
8IVH
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BU of 8ivh by Molmil
crystal structure of SulE mutant
分子名称: Alpha/beta fold hydrolase, GLYCEROL, L(+)-TARTARIC ACID, ...
著者Liu, B, He, J, Ran, T, Wang, W.
登録日2023-03-27
公開日2024-04-10
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献crystal structure of SulE mutant
To Be Published
4UYN
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SAR156497 an exquisitely selective inhibitor of Aurora kinases
分子名称: AURORA KINASE A, ethyl (9S)-9-[5-(1H-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2H-pyrrolo[3,4-b]quinoline-3-carboxylate
著者Carry, J.C, Clerc, F, Minoux, H, Schio, L, Mauger, J, Nair, A, Parmantier, E, Lemoigne, R, Delorme, C, Nicolas, J.P, Krick, A, Abecassis, P.Y, Crocq-Stuerga, V, Pouzieux, S, Delarbre, L, Maignan, S, Bertrand, T, Bjergarde, K, Ma, N, Lachaud, S, Guizani, H, Lebel, R, Doerflinger, G, Monget, S, Perron, S, Gasse, F, Angouillant-Boniface, O, Filoche-Romme, B, Murer, M, Gontier, S, Prevost, C, Monteiro, M.L, Combeau, C.
登録日2014-09-02
公開日2014-11-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Sar156497, an Exquisitely Selective Inhibitor of Aurora Kinases.
J.Med.Chem., 58, 2015

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件を2024-06-26に公開中

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