3W74
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![BU of 3w74 by Molmil](/molmil-images/mine/3w74) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-4-139 | 分子名称: | 2,6-dioxo-5-{2-[4-(trifluoromethoxy)phenyl]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-02-27 | 公開日 | 2014-03-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-4-139 To be Published
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3W7E
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![BU of 3w7e by Molmil](/molmil-images/mine/3w7e) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-5-179 | 分子名称: | 5-[2-(7-methoxynaphthalen-1-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-02-28 | 公開日 | 2014-03-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-5-179 To be Published
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6Q3O
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![BU of 6q3o by Molmil](/molmil-images/mine/6q3o) | PROTEIN-AROMATIC FOLDAMER COMPLEX CRYSTAL STRUCTURE | 分子名称: | 8-azanyl-4-(2-hydroxy-2-oxoethyloxy)quinoline-2-carboxylic acid, 8-azanyl-4-(3-azanylpropoxy)quinoline-2-carboxylic acid, Carbonic anhydrase 2, ... | 著者 | Zeberko, C, Langlois d'Estaintot, B, Fischer, L, Granier, T, Kauffmann, B, Huc, I. | 登録日 | 2018-12-04 | 公開日 | 2019-12-25 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.23 Å) | 主引用文献 | PROTEIN-AROMATIC FOLDAMER COMPLEX CRYSTAL STRUCTURE To Be Published
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3W7Q
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![BU of 3w7q by Molmil](/molmil-images/mine/3w7q) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with TT2-5-127 | 分子名称: | 5-{2-[1-(tert-butoxycarbonyl)-2,3-dihydro-1H-indol-5-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-03-02 | 公開日 | 2014-03-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with TT2-5-127 To be Published
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3W85
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![BU of 3w85 by Molmil](/molmil-images/mine/3w85) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with TT2-3-139 | 分子名称: | 5-{2-[3-(methoxycarbonyl)phenyl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-03-12 | 公開日 | 2014-03-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with TT2-3-139 To be Published
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3W72
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![BU of 3w72 by Molmil](/molmil-images/mine/3w72) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-4-107 | 分子名称: | 5-[2-(naphthalen-1-yl)ethyl]-2,6-dioxo-1,2,3,6- tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-02-27 | 公開日 | 2014-03-05 | 最終更新日 | 2017-11-22 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-4-107 To be Published
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3W7D
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![BU of 3w7d by Molmil](/molmil-images/mine/3w7d) | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-5-170 | 分子名称: | 5-[2-(8-methoxynaphthalen-2-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, COBALT HEXAMMINE(III), Dihydroorotate dehydrogenase (fumarate), ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-02-28 | 公開日 | 2014-03-05 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Structure of Trypanosoma cruzi dihydroorotate dehydrogenase in complex with MII-5-170 To be Published
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3W7R
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![BU of 3w7r by Molmil](/molmil-images/mine/3w7r) | Structure of Human dihydroorotate dehydrogenase in complex with mii-4-097 | 分子名称: | 2,6-dioxo-5-[2-(4-phenylphenyl)ethyl]-1,2,3,6- tetrahydropyrimidine-4-carboxylic acid, ACETATE ION, CHLORIDE ION, ... | 著者 | Inaoka, D.K, Iida, M, Tabuchi, T, Lee, N, Hashimoto, S, Matsuoka, S, Kuranaga, T, Shiba, T, Sakamoto, K, Suzuki, S, Balogun, E.O, Nara, T, Aoki, T, Inoue, M, Honma, T, Tanaka, A, Harada, S, Kita, K. | 登録日 | 2013-03-06 | 公開日 | 2014-03-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Structure of Human dihydroorotate dehydrogenase in complex with mii-4-097 To be Published
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3CKU
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![BU of 3cku by Molmil](/molmil-images/mine/3cku) | |
2H0L
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![BU of 2h0l by Molmil](/molmil-images/mine/2h0l) | Crystal Structure of a Mutant of Rat Annexin A5 | 分子名称: | Annexin A5, CALCIUM ION | 著者 | Langlois D'Estaintot, B, Gallois, B, Granier, T, Tessier, B, Brisson, A. | 登録日 | 2006-05-15 | 公開日 | 2007-06-19 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Identification of the Residues Involved in the Formation of Annexin V Trimers within 2D and 3D Crystals To be Published
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2GLQ
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![BU of 2glq by Molmil](/molmil-images/mine/2glq) | X-ray structure of human alkaline phosphatase in complex with strontium | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Alkaline phosphatase, placental type, ... | 著者 | Llinas, P, Masella, M, Stigbrand, T, Menez, A, Stura, E.A, Le Du, M.H. | 登録日 | 2006-04-05 | 公開日 | 2006-04-25 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural studies of human alkaline phosphatase in complex with strontium: Implication for its secondary effect in bones. Protein Sci., 15, 2006
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7EST
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![BU of 7est by Molmil](/molmil-images/mine/7est) | |
2H0M
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![BU of 2h0m by Molmil](/molmil-images/mine/2h0m) | |
1DAT
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![BU of 1dat by Molmil](/molmil-images/mine/1dat) | CUBIC CRYSTAL STRUCTURE RECOMBINANT HORSE L APOFERRITIN | 分子名称: | CADMIUM ION, L FERRITIN | 著者 | Gallois, B, Granier, T, Langlois D'Estaintot, B, Crichton, R.R, Roland, F. | 登録日 | 1996-11-14 | 公開日 | 1997-03-12 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | X-ray structure of recombinant horse L-chain apoferritin at 2.0 angstrom resolution: Implications for stability and function. J.Biol.Inorg.Chem., 2, 1997
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3PKL
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![BU of 3pkl by Molmil](/molmil-images/mine/3pkl) | Urate oxidase under 0.8 MPa / 8 bars pressure of xenon | 分子名称: | 8-AZAXANTHINE, SODIUM ION, Uricase, ... | 著者 | Marassio, G, Colloc'h, N, Prange, T, Abraini, J.H. | 登録日 | 2010-11-11 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.749 Å) | 主引用文献 | Pressure-response analysis of anesthetic gases xenon and nitrous oxide on urate oxidase: a crystallographic study. Faseb J., 25, 2011
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3PLE
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![BU of 3ple by Molmil](/molmil-images/mine/3ple) | urate oxidase under 0.5 MPa / 5 bars pressure of equimolar mixture xenon : nitrous oxide | 分子名称: | 8-AZAXANTHINE, NITROUS OXIDE, SODIUM ION, ... | 著者 | Marassio, G, Colloc'h, N, Prange, T, Abraini, J.H. | 登録日 | 2010-11-15 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Pressure-response analysis of anesthetic gases xenon and nitrous oxide on urate oxidase: a crystallographic study. Faseb J., 25, 2011
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3PLJ
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![BU of 3plj by Molmil](/molmil-images/mine/3plj) | Urate oxidase under 3.0 MPa / 30 bars pressure of equimolar mixture xenon : nitrous oxide | 分子名称: | 8-AZAXANTHINE, NITROUS OXIDE, SODIUM ION, ... | 著者 | Marassio, G, Colloc'h, N, Prange, T, Abraini, J.H. | 登録日 | 2010-11-15 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.732 Å) | 主引用文献 | Pressure-response analysis of anesthetic gases xenon and nitrous oxide on urate oxidase: a crystallographic study. Faseb J., 25, 2011
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2R5T
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![BU of 2r5t by Molmil](/molmil-images/mine/2r5t) | Crystal Structure of Inactive Serum and Glucocorticoid- Regulated Kinase 1 in Complex with AMP-PNP | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, SULFATE ION, ... | 著者 | Zhao, B, Lehr, R, Smallwood, A.M, Ho, T.F, Maley, K, Randall, T, Head, M.S, Koretke, K.K, Schnackenberg, C.G. | 登録日 | 2007-09-04 | 公開日 | 2008-09-09 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of the kinase domain of serum and glucocorticoid-regulated kinase 1 in complex with AMP PNP. Protein Sci., 16, 2007
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1ICG
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![BU of 1icg by Molmil](/molmil-images/mine/1icg) | STRUCTURE OF THE HYBRID RNA/DNA R-GCUUCGGC-D[F]U IN PRESENCE OF IR(NH3)6+++ | 分子名称: | 5'-R(*GP*CP*UP*UP*CP*GP*GP*C)-D(P*(UFP))-3', CHLORIDE ION, IRIDIUM HEXAMMINE ION | 著者 | Cruse, W, Saludjian, P, Neuman, A, Prange, T. | 登録日 | 2001-03-31 | 公開日 | 2001-04-09 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Destabilizing effect of a fluorouracil extra base in a hybrid RNA duplex compared with bromo and chloro analogues. Acta Crystallogr.,Sect.D, 57, 2001
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1IDW
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![BU of 1idw by Molmil](/molmil-images/mine/1idw) | STRUCTURE OF THE HYBRID RNA/DNA R-GCUUCGGC-D[CL]U IN PRESENCE OF RH(NH3)6+++ | 分子名称: | 5'-R(*GP*CP*UP*UP*CP*GP*GP*C)-D(P*(UCL))-3', CHLORIDE ION, RHODIUM HEXAMINE ION | 著者 | Cruse, W, Saludjian, P, Neuman, A, Prange, T. | 登録日 | 2001-04-05 | 公開日 | 2001-04-12 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Destabilizing effect of a fluorouracil extra base in a hybrid RNA duplex compared with bromo and chloro analogues Acta Crystallogr.,Sect.D, 57, 2001
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1IHA
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![BU of 1iha by Molmil](/molmil-images/mine/1iha) | Structure of the Hybrid RNA/DNA R-GCUUCGGC-D[BR]U in Presence of RH(NH3)6+++ | 分子名称: | 5'-R(*GP*CP*UP*UP*CP*GP*GP*C)-D(P*(BRU))-3', CHLORIDE ION, RHODIUM HEXAMINE ION | 著者 | Cruse, W.B, Saludjian, P, Neuman, A, Prange, T. | 登録日 | 2001-04-19 | 公開日 | 2001-05-07 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Destabilizing effect of a fluorouracil extra base in a hybrid RNA duplex compared with bromo and chloro analogues. Acta Crystallogr.,Sect.D, 57, 2001
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1ISG
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![BU of 1isg by Molmil](/molmil-images/mine/1isg) | Crystal Structure Analysis of BST-1/CD157 with ATPgammaS | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER, bone marrow stromal cell antigen 1 | 著者 | Yamamoto-Katayama, S, Ariyoshi, M, Ishihara, K, Hirano, T, Jingami, H, Morikawa, K. | 登録日 | 2001-12-05 | 公開日 | 2002-03-13 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Crystallographic studies on human BST-1/CD157 with ADP-ribosyl cyclase and NAD glycohydrolase activities. J.Mol.Biol., 316, 2002
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1ISM
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![BU of 1ism by Molmil](/molmil-images/mine/1ism) | Crystal Structure Analysis of BST-1/CD157 complexed with nicotinamide | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, NICOTINAMIDE, bone marrow stromal cell antigen 1 | 著者 | Yamamoto-Katayama, S, Ariyoshi, M, Ishihara, K, Hirano, T, Jingami, H, Morikawa, K. | 登録日 | 2001-12-05 | 公開日 | 2002-03-13 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystallographic studies on human BST-1/CD157 with ADP-ribosyl cyclase and NAD glycohydrolase activities. J.Mol.Biol., 316, 2002
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2ZDK
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![BU of 2zdk by Molmil](/molmil-images/mine/2zdk) | Exploring Trypsin S3 Pocket | 分子名称: | (S)-N-(4-carbamimidoylbenzyl)-1-(3-cyclohexylpropanoyl)pyrrolidine-2-carboxamide, CALCIUM ION, Cationic trypsin, ... | 著者 | Baum, B, Brandt, T, Heine, A, Klebe, G. | 登録日 | 2007-11-26 | 公開日 | 2008-10-14 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Congeneric but still distinct: how closely related trypsin ligands exhibit different thermodynamic and structural properties J.Mol.Biol., 405, 2011
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4BFR
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![BU of 4bfr by Molmil](/molmil-images/mine/4bfr) | Discovery and Optimization of Pyrimidone Indoline Amide PI3Kbeta Inhibitors for the Treatment of Phosphatase and TENsin homologue (PTEN)-Deficient Cancers | 分子名称: | 2-[2-(2-METHYL-2,3-DIHYDRO-INDOL-1-YL)-2-OXO-ETHYL]-6-MORPHOLIN-4-YL-3H-PYRIMIDIN-4-ONE, PHOSPHATIDYLINOSITOL 4,5-BISPHOSPHATE 3-KINASE CATALYTIC S SUBUNIT BETA ISOFORM | 著者 | Certal, V, Carry, J.C, Halley, F, Virone-Oddos, A, Thompson, F, Filoche-Romme, B, El-Ahmad, Y, Karlsson, A, Charrier, V, Delorme, C, Rak, A, Abecassis, P.Y, Amara, C, Vincent, L, Bonnevaux, H, Nicolas, J.P, Mathieu, M, Bertrand, T, Marquette, J.P, Michot, N, Benard, T, Perrin, M.A, Perron, S, Monget, S, Gruss-Leleu, F, Doerflinger, G, Guizani, H, Brollo, M, Delbarre, L, Bertin, L, Richepin, P, Loyau, V, Garcia-Echeverria, C, Lengauer, C, Schio, L. | 登録日 | 2013-03-22 | 公開日 | 2014-01-15 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Discovery and Optimization of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors for the Treatment of Phosphatase and Tensin Homologue (Pten)-Deficient Cancers. J.Med.Chem., 57, 2014
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