7X56
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![BU of 7x56 by Molmil](/molmil-images/mine/7x56) | A CBg-ParM filament with ADP | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ParM/StbA family protein | 著者 | Koh, A, Ali, S, Robinson, R, Narita, A. | 登録日 | 2022-03-04 | 公開日 | 2023-03-08 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | A new actin-like filament from Clostridium botulinum exhibits a new system of filament turn over To Be Published
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1S3N
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![BU of 1s3n by Molmil](/molmil-images/mine/1s3n) | Structural and Functional Characterization of a Novel Archaeal Phosphodiesterase | 分子名称: | Hypothetical protein MJ0936, MANGANESE (II) ION | 著者 | Chen, S, Busso, D, Yakunin, A.F, Kuznetsova, E, Proudfoot, M, Jancrick, J, Kim, R, Kim, S.-H, Berkeley Structural Genomics Center (BSGC) | 登録日 | 2004-01-13 | 公開日 | 2004-08-10 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural and functional characterization of a novel phosphodiesterase from Methanococcus jannaschii J.Biol.Chem., 279, 2004
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7X55
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5JXJ
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![BU of 5jxj by Molmil](/molmil-images/mine/5jxj) | Structure of the proprotein convertase furin complexed to meta-guanidinomethyl-Phac-RVR-Amba in presence of EDTA | 分子名称: | 2UC-ARG-VAL-ARG-00S, CALCIUM ION, CHLORIDE ION, ... | 著者 | Dahms, S.O, Arciniega, M, Steinmetzer, T, Huber, R, Than, M.E. | 登録日 | 2016-05-13 | 公開日 | 2016-10-05 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of the unliganded form of the proprotein convertase furin suggests activation by a substrate-induced mechanism. Proc.Natl.Acad.Sci.USA, 113, 2016
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5JYI
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![BU of 5jyi by Molmil](/molmil-images/mine/5jyi) | Trypsin bound with succinic acid at 1.9A | 分子名称: | CALCIUM ION, Cationic trypsin, SODIUM ION, ... | 著者 | Manohar, R, Kutumbarao, N.H.V, KarthiK, L, Malathy, P, Velmurugan, D, Gunasekaran, K. | 登録日 | 2016-05-14 | 公開日 | 2016-07-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.914 Å) | 主引用文献 | Trypsin bound with succinic acid at 1.9A To Be Published
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5JYB
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![BU of 5jyb by Molmil](/molmil-images/mine/5jyb) | Crystal structure of 3 mutant of Ba3275 (S116A, E243A, H313A), the member of S66 family of serine peptidases | 分子名称: | 1,2-ETHANEDIOL, 2-BUTANOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... | 著者 | Nocek, B, Jedrzejczak, R, Joachimiak, A, CSGID, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2016-05-13 | 公開日 | 2016-06-15 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.647 Å) | 主引用文献 | Crystal structure of 3 mutant of Ba3275 (S116A, E243A, H313A), the member of S66 family of serine peptidases To Be Published
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7X54
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![BU of 7x54 by Molmil](/molmil-images/mine/7x54) | A CBg-ParM filament with ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ParM/StbA family protein | 著者 | Koh, A, Ali, S, Robinson, R, Narita, A. | 登録日 | 2022-03-04 | 公開日 | 2023-03-08 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | A new actin-like filament from Clostridium botulinum exhibits a new system of filament turn over To Be Published
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1SHG
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![BU of 1shg by Molmil](/molmil-images/mine/1shg) | CRYSTAL STRUCTURE OF A SRC-HOMOLOGY 3 (SH3) DOMAIN | 分子名称: | ALPHA-SPECTRIN SH3 DOMAIN | 著者 | Noble, M, Pauptit, R, Musacchio, A, Saraste, M, Wierenga, R.K. | 登録日 | 1993-05-19 | 公開日 | 1993-10-31 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of a Src-homology 3 (SH3) domain. Nature, 359, 1992
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5JZB
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![BU of 5jzb by Molmil](/molmil-images/mine/5jzb) | Crystal structure of HsaD bound to 3,5-dichlorobenzene sulphonamide | 分子名称: | 3,5-dichlorobenzene-1-sulfonamide, 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase, PHOSPHATE ION | 著者 | Ryan, A, Polycarpou, E, Lack, N.A, Evangelopoulos, D, Sieg, C, Halman, A, Bhakta, S, Sinclair, A, Eleftheriadou, O, McHugh, T.D, Keany, S, Lowe, E, Ballet, R, Abihammad, A, Ciulli, A, Sim, E. | 登録日 | 2016-05-16 | 公開日 | 2017-04-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.102 Å) | 主引用文献 | Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. Br. J. Pharmacol., 174, 2017
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6W9C
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![BU of 6w9c by Molmil](/molmil-images/mine/6w9c) | The crystal structure of papain-like protease of SARS CoV-2 | 分子名称: | CHLORIDE ION, Non-structural protein 3, ZINC ION | 著者 | Osipiuk, J, Jedrzejczak, R, Tesar, C, Endres, M, Stols, L, Babnigg, G, Kim, Y, Michalska, K, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2020-03-22 | 公開日 | 2020-04-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | The crystal structure of papain-like protease of SARS CoV-2 to be published
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3MEP
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![BU of 3mep by Molmil](/molmil-images/mine/3mep) | Crystal Structure of ECA2234 protein from Erwinia carotovora, Northeast Structural Genomics Consortium Target EwR44 | 分子名称: | uncharacterized protein ECA2234 | 著者 | Seetharaman, J, Abashidze, M, Forouhar, F, Mao, M, Xiao, R, Ciccosanti, C, Wang, D, Everett, J.K, Nair, R, Acton, T.B, Rost, B, Montelione, G.T, Tong, L, Hunt, J.F, Northeast Structural Genomics Consortium (NESG) | 登録日 | 2010-03-31 | 公開日 | 2010-04-14 | 最終更新日 | 2019-07-17 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Northeast Structural Genomics Consortium Target EwR44 To be Published
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7WWV
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![BU of 7wwv by Molmil](/molmil-images/mine/7wwv) | DNA bound-ICP1 Csy complex | 分子名称: | Csy1, Csy2, Csy3, ... | 著者 | Zhang, M, Peng, R. | 登録日 | 2022-02-14 | 公開日 | 2023-04-26 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Mechanistic insights into DNA binding and cleavage by a compact type I-F CRISPR-Cas system in bacteriophage. Proc.Natl.Acad.Sci.USA, 120, 2023
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7WWU
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![BU of 7wwu by Molmil](/molmil-images/mine/7wwu) | ICP1 Csy complex | 分子名称: | Csy1, Csy2, Csy3, ... | 著者 | Zhang, M, Peng, R. | 登録日 | 2022-02-14 | 公開日 | 2023-04-26 | 最終更新日 | 2024-06-26 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Mechanistic insights into DNA binding and cleavage by a compact type I-F CRISPR-Cas system in bacteriophage. Proc.Natl.Acad.Sci.USA, 120, 2023
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6WAX
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![BU of 6wax by Molmil](/molmil-images/mine/6wax) | C-terminal SH2 domain of p120RasGAP | 分子名称: | 1,2-ETHANEDIOL, Ras GTPase-activating protein 1, SULFATE ION | 著者 | Jaber Chehayeb, R, Wang, J, Stiegler, A.L, Boggon, T.J. | 登録日 | 2020-03-26 | 公開日 | 2020-06-17 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The GTPase-activating protein p120RasGAP has an evolutionarily conserved "FLVR-unique" SH2 domain. J.Biol.Chem., 295, 2020
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1C4V
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![BU of 1c4v by Molmil](/molmil-images/mine/1c4v) | SELECTIVE NON ELECTROPHILIC THROMBIN INHIBITORS WITH CYCLOHEXYL MOIETIES. | 分子名称: | 2-(2,2-DIPHENYL-ETHYL)-7-METHYL-1,3-DIOXO-2,3,5,8-TETRAHYDRO-1H-[1,2,4]TRIAZOLO [1,2-A]PYRIDAZINE-5-CARBOXYLIC ACID(4-CARBAMIMIDOYL-CYCLOHEXYLMETHYL)-AMIDE, HIRUGEN, SODIUM ION, ... | 著者 | Krishnan, R, Mochalkin, I, Arni, R.K, Tulinsky, A. | 登録日 | 1999-09-25 | 公開日 | 2000-09-27 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure of thrombin complexed with selective non-electrophilic inhibitors having cyclohexyl moieties at P1. Acta Crystallogr.,Sect.D, 56, 2000
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1C4U
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![BU of 1c4u by Molmil](/molmil-images/mine/1c4u) | SELECTIVE NON ELECTROPHILIC THROMBIN INHIBITORS WITH CYCLOHEXYL MOIETIES. | 分子名称: | 2-[2-(4-BROMO-BENZENESULFONYL)-ETHYL]-1-3-DIOXO-2,3,5,8-TETRAHYDRO-1H-[1,2,4]TRIAZOLO[1,2-A]PYRIDAZINE-5-CARBOXYLIC ACID(4-CARBAMIMIDOYL-CYCLOHEXYLMETHYL)-AMIDE, PROTEIN (HIRUGEN), SODIUM ION, ... | 著者 | Krishnan, R, Mochalkin, I, Arni, R.K, Tulinsky, A. | 登録日 | 1999-09-25 | 公開日 | 2000-09-27 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure of thrombin complexed with selective non-electrophilic inhibitors having cyclohexyl moieties at P1. Acta Crystallogr.,Sect.D, 56, 2000
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1C4Y
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![BU of 1c4y by Molmil](/molmil-images/mine/1c4y) | SELECTIVE NON-ELECTROPHILIC THROMBIN INHIBITORS | 分子名称: | 2-(2,2-DIPHENYL-ETHYL)-7-METHYL-1,3-DIOXO-2,3,5,8-TETRAHYDRO-1H-[1,2,4] TRIAZOLO[1,2-A]PYRIDAZINE-5-CARBOXYLIC ACID [4-(2-AMINO-3H-IMIDAZOL-4-YL)-CYCLOHEXYL]-AMIDE, HIRUGEN, THROMBIN:LONG CHAIN, ... | 著者 | Krishnan, R, Mochalkin, I, Arni, R.K, Tulinsky, A. | 登録日 | 1999-10-05 | 公開日 | 2000-10-09 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Structure of thrombin complexed with selective non-electrophilic inhibitors having cyclohexyl moieties at P1. Acta Crystallogr.,Sect.D, 56, 2000
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5K8Q
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![BU of 5k8q by Molmil](/molmil-images/mine/5k8q) | Crystal Structure of Calcium-loaded Calmodulin in complex with STRA6 CaMBP2-site peptide. | 分子名称: | CALCIUM ION, Calmodulin, IMIDAZOLE, ... | 著者 | Stowe, S.D, Clarke, O.B, Cavalier, M.C, Godoy-Ruiz, R, Mancia, F, Weber, D.J. | 登録日 | 2016-05-30 | 公開日 | 2016-08-24 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.739 Å) | 主引用文献 | Structure of the STRA6 receptor for retinol uptake. Science, 353, 2016
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5KBG
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![BU of 5kbg by Molmil](/molmil-images/mine/5kbg) | CRYSTAL STRUCTURE OF THE AROMATIC SENSOR DOMAIN OF MOPR IN COMPLEX WITH OCRESOL | 分子名称: | MopR, ZINC ION, o-cresol | 著者 | Ray, S, Anand, R, Panjikar, S. | 登録日 | 2016-06-03 | 公開日 | 2016-07-13 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural Basis of Selective Aromatic Pollutant Sensing by the Effector Binding Domain of MopR, an NtrC Family Transcriptional Regulator. Acs Chem.Biol., 11, 2016
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5KA4
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5KAB
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![BU of 5kab by Molmil](/molmil-images/mine/5kab) | Protein Tyrosine Phosphatase 1B Delta helix 7, P185G mutant in complex with TCS401, open state | 分子名称: | 2-(OXALYL-AMINO)-4,5,6,7-TETRAHYDRO-THIENO[2,3-C]PYRIDINE-3-CARBOXYLIC ACID, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ... | 著者 | Choy, M.S, Machado, L.E.S.F, Peti, W, Page, R. | 登録日 | 2016-06-01 | 公開日 | 2017-03-08 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.968 Å) | 主引用文献 | Conformational Rigidity and Protein Dynamics at Distinct Timescales Regulate PTP1B Activity and Allostery. Mol. Cell, 65, 2017
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5KE3
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![BU of 5ke3 by Molmil](/molmil-images/mine/5ke3) | Crystal structure of SETDB1 Tudor domain in complex with fragment MRT0181a | 分子名称: | (S)-N-(furan-2-ylmethyl)-1-(1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidine-4-carboxamide, BETA-MERCAPTOETHANOL, Histone-lysine N-methyltransferase SETDB1, ... | 著者 | Dong, A, Iqbal, A, Mader, P, Dobrovetsky, E, Ferreira de Freitas, R, Walker, J.R, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Schapira, M, Brown, P.J, Structural Genomics Consortium (SGC) | 登録日 | 2016-06-09 | 公開日 | 2016-08-03 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of SETDB1 Tudor domain in complex with fragment MRT0181a to be published
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3NMA
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![BU of 3nma by Molmil](/molmil-images/mine/3nma) | Mutant P169S of Foot-and-mouth disease Virus RNA dependent RNA-polymerase | 分子名称: | 5'-R(*GP*GP*C)-3', 5'-R(P*CP*C)-3', Genome polyprotein, ... | 著者 | Agudo, R, Ferrer-Orta, C, Arias, A, Perez-Luque, R, Verdaguer, N, Domingo, E. | 登録日 | 2010-06-22 | 公開日 | 2011-05-25 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | A multi-step process of viral adaptation to a mutagenic nucleoside analogue by modulation of transition types leads to extinction-escape. Plos Pathog., 6, 2010
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3RJ9
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![BU of 3rj9 by Molmil](/molmil-images/mine/3rj9) | Structure of alcohol dehydrogenase from Drosophila lebanonesis T114V mutant complexed with NAD+ | 分子名称: | Alcohol dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Morgunova, E, Wuxiuer, Y, Cols, N, Popov, A, Sylte, I, Karshikoff, A, Gonzales-Duarte, R, Ladenstein, R, Winberg, J.O. | 登録日 | 2011-04-15 | 公開日 | 2012-05-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | An intact eight-membered water chain in drosophilid alcohol dehydrogenases is essential for optimal enzyme activity. Febs J., 279, 2012
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5JT2
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![BU of 5jt2 by Molmil](/molmil-images/mine/5jt2) | BRAFV600E Kinase Domain In Complex with Chemically Linked Vemurafenib Inhibitor VEM-BISAMIDE | 分子名称: | 2,2'-oxybis(N-{[4-(3-{2,6-difluoro-3-[(propane-1-sulfonyl)amino]benzoyl}-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl]methyl}acetamide), BENZAMIDINE, Serine/threonine-protein kinase B-raf | 著者 | Grasso, M.J, Marmorstein, R. | 登録日 | 2016-05-09 | 公開日 | 2016-09-14 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.702 Å) | 主引用文献 | Chemically Linked Vemurafenib Inhibitors Promote an Inactive BRAF(V600E) Conformation. Acs Chem.Biol., 11, 2016
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