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PDB: 2 results

6C45
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BU of 6c45 by Molmil
Crystal structure of human inorganic pyrophosphatase in the P212121 space group
Descriptor: Inorganic pyrophosphatase
Authors:Niu, H, Zhu, J, Huang, X, Du, Z.
Deposit date:2018-01-11
Release date:2019-01-16
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.388 Å)
Cite:Expression, purification and crystallization of the human protein PPA1
To be Published
7XSV
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BU of 7xsv by Molmil
Crystal Structures of PIM1 in Complex with Macrocyclic Compound H3
Descriptor: 8-Methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene, Serine/threonine-protein kinase pim-1
Authors:Shen, C, Xie, Y, Ren, X, Zhou, Y, Niu, H.
Deposit date:2022-05-15
Release date:2022-07-13
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.66 Å)
Cite:Design, synthesis, and bioactivity evaluation of macrocyclic benzo[b]pyrido[4,3-e][1,4]oxazine derivatives as novel Pim-1 kinase inhibitors.
Bioorg.Med.Chem.Lett., 72, 2022

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