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5E80
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BU of 5e80 by Molmil
The crystal structure of PDEd in complex with inhibitor-2a
Descriptor: N-(3-chloro-2-methylphenyl)-4-(3,4-dimethyl-7-oxo-2-phenyl-2,7-dihydro-6H-pyrazolo[3,4-d]pyridazin-6-yl)butanamide, Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta
Authors:Ismail, S, Fansa, E.K, Murarka, S, Wittinghofer, A.
Deposit date:2015-10-13
Release date:2016-05-04
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Identification of pyrazolopyridazinones as PDE delta inhibitors.
Nat Commun, 7, 2016

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