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PDB: 3 results

4YUR
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BU of 4yur by Molmil
Crystal Structure of Plk4 Kinase Domain Bound to Centrinone
Descriptor: 2-({2-fluoro-4-[(2-fluoro-3-nitrobenzyl)sulfonyl]phenyl}sulfanyl)-5-methoxy-N-(3-methyl-1H-pyrazol-5-yl)-6-(morpholin-4-yl)pyrimidin-4-amine, Serine/threonine-protein kinase PLK4
Authors:Shiau, A.K, Motamedi, A.
Deposit date:2015-03-19
Release date:2015-06-17
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.65 Å)
Cite:Cell biology. Reversible centriole depletion with an inhibitor of Polo-like kinase 4.
Science, 348, 2015
5I4N
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BU of 5i4n by Molmil
Crystal Structure of the E596A V617F Mutant JAK2 Pseudokinase Domain Bound to Mg-ATP
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GLYCEROL, MAGNESIUM ION, ...
Authors:Shiau, A.K, Motamedi, A.
Deposit date:2016-02-12
Release date:2016-04-13
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.54 Å)
Cite:Uncoupling JAK2 V617F activation from cytokine-induced signalling by modulation of JH2 alpha C helix.
Biochem.J., 473, 2016
5EW9
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BU of 5ew9 by Molmil
Crystal Structure of Aurora A Kinase Domain Bound to MK-5108
Descriptor: 4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid, Aurora kinase A
Authors:Shiau, A.K, Motamedi, A.
Deposit date:2015-11-20
Release date:2016-01-20
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.181 Å)
Cite:A Cell Biologist's Field Guide to Aurora Kinase Inhibitors.
Front Oncol, 5, 2015

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