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PDB: 85 件

7ER9
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Crystal structure of human Biliverdin IX-beta reductase B with Febuxostat (TEI)
分子名称: 2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE-CARBOXYLIC ACID, Flavin reductase (NADPH), NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Griesinger, C, Lee, D, Ryu, K.S, Kim, M, Ha, J.H.
登録日2021-05-06
公開日2022-01-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Repositioning Food and Drug Administration-Approved Drugs for Inhibiting Biliverdin IX beta Reductase B as a Novel Thrombocytopenia Therapeutic Target.
J.Med.Chem., 65, 2022
7ERA
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Crystal structure of human Biliverdin IX-beta reductase B with Olsalazine Sodium (OSS)
分子名称: 5-[(E)-(3-carboxy-4-oxidanyl-phenyl)diazenyl]-2-oxidanyl-benzoic acid, Flavin reductase (NADPH), NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Griesinger, C, Lee, D, Ryu, K.S, Kim, M, Ha, J.H.
登録日2021-05-06
公開日2022-01-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献Repositioning Food and Drug Administration-Approved Drugs for Inhibiting Biliverdin IX beta Reductase B as a Novel Thrombocytopenia Therapeutic Target.
J.Med.Chem., 65, 2022
7ER6
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Crystal structure of human Biliverdin IX-beta reductase B
分子名称: Flavin reductase (NADPH), NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, SULFATE ION
著者Griesinger, C, Lee, D, Ryu, K.S, Kim, M, Ha, J.H.
登録日2021-05-06
公開日2022-01-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Repositioning Food and Drug Administration-Approved Drugs for Inhibiting Biliverdin IX beta Reductase B as a Novel Thrombocytopenia Therapeutic Target.
J.Med.Chem., 65, 2022
7ERE
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Crystal structure of human Biliverdin IX-beta reductase B with Pyrantel Pamoate (PPA)
分子名称: 4-[(3-carboxy-2-oxidanyl-naphthalen-1-yl)methyl]-3-oxidanyl-naphthalene-2-carboxylic acid, Flavin reductase (NADPH), NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Griesinger, C, Lee, D, Ryu, K.S, Kim, M, Ha, J.H.
登録日2021-05-06
公開日2022-01-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Repositioning Food and Drug Administration-Approved Drugs for Inhibiting Biliverdin IX beta Reductase B as a Novel Thrombocytopenia Therapeutic Target.
J.Med.Chem., 65, 2022
7ERD
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Crystal structure of human Biliverdin IX-beta reductase B with Flunixin Meglumin (FMG)
分子名称: 2-[[2-methyl-3-(trifluoromethyl)phenyl]amino]pyridine-3-carboxylic acid, Flavin reductase (NADPH), NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Griesinger, C, Lee, D, Ryu, K.S, Kim, M, Ha, J.H.
登録日2021-05-06
公開日2022-01-19
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Repositioning Food and Drug Administration-Approved Drugs for Inhibiting Biliverdin IX beta Reductase B as a Novel Thrombocytopenia Therapeutic Target.
J.Med.Chem., 65, 2022
1IU7
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HOLO FORM OF COPPER-CONTAINING AMINE OXIDASE FROM ARTHROBACTER GLOBIFORMIS
分子名称: AMINE OXIDASE, COPPER (II) ION
著者Kishishita, S, Okajima, T, Kim, M, Yamaguchi, H, Hirota, S, Suzuki, S, Kuroda, S, Tanizawa, K, Mure, M.
登録日2002-02-28
公開日2003-02-04
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Role of Copper Ion in Bacterial Copper Amine Oxidase: Spectroscopic and Crystallographic Studies of Metal-Substituted Enzymes
J.AM.CHEM.SOC., 125, 2003
1QA9
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BU of 1qa9 by Molmil
Structure of a Heterophilic Adhesion Complex Between the Human CD2 and CD58(LFA-3) Counter-Receptors
分子名称: HUMAN CD2 PROTEIN, HUMAN CD58 PROTEIN
著者Wang, J.-H, Smolyar, A, Tan, K, Liu, J.-H, Kim, M, Sun, Z.J, Wagner, G, Reinherz, E.L.
登録日1999-04-13
公開日1999-04-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structure of a heterophilic adhesion complex between the human CD2 and CD58 (LFA-3) counterreceptors.
Cell(Cambridge,Mass.), 97, 1999
1IQX
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CRYSTAL STRUCTURE OF COBALT-SUBSTITUTED AMINE OXIDASE FROM ARTHROBACTER GLOBIFORMIS
分子名称: CO(II)-SUBSTITUTED AMINE OXIDASE, COBALT (II) ION
著者Kishishita, S, Okajima, T, Mure, M, Kim, M, Yamaguchi, H, Hirota, S, Suzuki, S, Kuroda, S, Tanizawa, K.
登録日2001-08-27
公開日2003-02-04
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Role of Copper Ion in Bacterial Copper Amine Oxidase: Spectroscopic and Crystallographic Studies of Metal-Substituted Enzymes
J.AM.CHEM.SOC., 125, 2003
1IQY
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BU of 1iqy by Molmil
CRYSTAL STRUCTURE OF NICKEL-SUBSTITUTED AMINE OXIDASE FROM ARTHROBACTER GLOBIFORMIS
分子名称: AMINE OXIDASE, NICKEL (II) ION
著者Kishishita, S, Okajima, T, Mure, M, Kim, M, Yamaguchi, H, Hirota, S, Kuroda, S, Tanizawa, K.
登録日2001-08-28
公開日2003-02-04
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Role of Copper Ion in Bacterial Copper Amine Oxidase: Spectroscopic and Crystallographic Studies of Metal-Substituted Enzymes
J.AM.CHEM.SOC., 125, 2003
6K6I
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BU of 6k6i by Molmil
The crystal structure of light-driven cyanobacterial chloride importer from Mastigocladopsis repens
分子名称: CHLORIDE ION, Cyanobacterial chloride importer, OLEIC ACID, ...
著者Yun, J.H, Park, J.H, Jin, Z, Ohki, M, Wang, Y, Lupala, C.S, Kim, M, Liu, H, Park, S.Y, Lee, W.
登録日2019-06-03
公開日2020-06-03
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献The crystal structure of light-driven cyanobacterial chloride importer from Mastigocladopsis repens
To Be Published
6K6K
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The crystal structure of light-driven cyanobacterial chloride importer (N63A/P118A) Mastigocladopsis repens
分子名称: CHLORIDE ION, Cyanobacterial chloride importer, OLEIC ACID, ...
著者Yun, J.H, Park, J.H, Jin, Z, Ohki, M, Wang, Y, Lupala, C.S, Kim, M, Liu, H, Park, S.Y, Lee, W.
登録日2019-06-03
公開日2020-06-03
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.197 Å)
主引用文献The crystal structure of light-driven cyanobacterial chloride importer (N63A/P118A) Mastigocladopsis repens
To Be Published
7VYT
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BU of 7vyt by Molmil
Crystal structure of human TIGIT(23-129) in complex with the scFv fragment of anti-TIGIT antibody MG1131
分子名称: CITRATE ANION, MG1131 heavy chain variable region, MG1131 light chain variable region, ...
著者Jeong, B.-S, Nam, H, Kim, M, Oh, B.-H.
登録日2021-11-15
公開日2022-03-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Structural and functional characterization of a monoclonal antibody blocking TIGIT.
Mabs, 14, 2022
6K6J
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BU of 6k6j by Molmil
The crystal structure of light-driven cyanobacterial chloride importer from Mastigocladopsis repens with Bromide ion
分子名称: BROMIDE ION, Cyanobacterial chloride importer, OLEIC ACID, ...
著者Yun, J.H, Park, J.H, Jin, Z, Ohki, M, Wang, Y, Lupala, C.S, Kim, M, Liu, H, Park, S.Y, Lee, W.
登録日2019-06-03
公開日2020-06-03
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The crystal structure of light-driven cyanobacterial chloride importer from Mastigocladopsis repens with Bromide ion
To Be Published
4H8A
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BU of 4h8a by Molmil
Crystal structure of ureidoglycolate dehydrogenase in binary complex with NADH
分子名称: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, Ureidoglycolate dehydrogenase
著者Rhee, S, Shin, I, Kim, M.
登録日2012-09-22
公開日2013-01-16
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.64 Å)
主引用文献Structural and functional insights into (s)-ureidoglycolate dehydrogenase, a metabolic branch point enzyme in nitrogen utilization.
Plos One, 7, 2012
5CKR
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BU of 5ckr by Molmil
Crystal Structure of MraY in complex with Muraymycin D2
分子名称: Muraymycin D2, Phospho-N-acetylmuramoyl-pentapeptide-transferase
著者Lee, S.Y, Chung, B.C, Mashalidis, E.H, Tanino, T, Kim, M, Hong, J, Ichikawa, S.
登録日2015-07-15
公開日2016-03-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Structural insights into inhibition of lipid I production in bacterial cell wall synthesis.
Nature, 533, 2016
6BSH
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BU of 6bsh by Molmil
Structure of HIV-1 RT complexed with RNA/DNA hybrid in the RNA hydrolysis mode
分子名称: (-)-6-CHLORO-4-CYCLOPROPYLETHYNYL-4-TRIFLUOROMETHYL-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONE, CALCIUM ION, DNA (5'-D(*GP*TP*AP*TP*GP*CP*CP*AP*CP*TP*AP*GP*TP*TP*AP*TP*TP*GP*TP*GP*GP*CP*C)-3'), ...
著者Tian, L, Kim, M, Yang, W.
登録日2017-12-03
公開日2018-01-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.649 Å)
主引用文献Structure of HIV-1 reverse transcriptase cleaving RNA in an RNA/DNA hybrid.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
6BSI
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BU of 6bsi by Molmil
Structure of HIV-1 RT complexed with an RNA/DNA hybrid containing the polypurine-tract sequence
分子名称: (-)-6-CHLORO-4-CYCLOPROPYLETHYNYL-4-TRIFLUOROMETHYL-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONE, CALCIUM ION, DNA (5'-D(*GP*TP*TP*TP*TP*TP*CP*TP*TP*TP*TP*GP*TP*TP*AP*TP*TP*GP*TP*GP*GP*CP*C)-3'), ...
著者Tian, L, Kim, M, Yang, W.
登録日2017-12-03
公開日2018-01-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (3.25 Å)
主引用文献Structure of HIV-1 reverse transcriptase cleaving RNA in an RNA/DNA hybrid.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
6BSJ
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BU of 6bsj by Molmil
Structure of HIV-1 RT complexed with an RNA/DNA hybrid sequence non-preferred for RNA hydrolysis
分子名称: (-)-6-CHLORO-4-CYCLOPROPYLETHYNYL-4-TRIFLUOROMETHYL-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONE, CALCIUM ION, DNA (5'-D(*GP*TP*AP*TP*GP*CP*CP*TP*AP*TP*AP*GP*TP*TP*AP*TP*TP*GP*TP*GP*GP*CP*C)-3'), ...
著者Tian, L, Kim, M, Yang, W.
登録日2017-12-03
公開日2018-01-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Structure of HIV-1 reverse transcriptase cleaving RNA in an RNA/DNA hybrid.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
6BSG
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BU of 6bsg by Molmil
Structure of HIV-1 RT complexed with RNA/DNA hybrid in an RNA hydrolysis-off mode
分子名称: (-)-6-CHLORO-4-CYCLOPROPYLETHYNYL-4-TRIFLUOROMETHYL-1,4-DIHYDRO-2H-3,1-BENZOXAZIN-2-ONE, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
著者Tian, L, Kim, M, Yang, W.
登録日2017-12-03
公開日2018-01-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Structure of HIV-1 reverse transcriptase cleaving RNA in an RNA/DNA hybrid.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
3CLJ
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BU of 3clj by Molmil
Structure of the RNA polymerase II CTD-interacting domain of Nrd1
分子名称: GLYCEROL, Protein NRD1, SULFATE ION
著者Vasiljeva, L, Kim, M, Mutschler, H, Buratowski, S, Meinhart, A.
登録日2008-03-19
公開日2008-07-29
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Nrd1-Nab3-Sen1 termination complex interacts with the Ser5-phosphorylated RNA polymerase II C-terminal domain.
Nat.Struct.Mol.Biol., 15, 2008
3W30
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BU of 3w30 by Molmil
Structual basis for the recognition of Ubc13 by the Shigella flexneri effector OspI
分子名称: ORF169b
著者Nishide, A, Kim, M, Takagi, K, Sasakawa, C, Mizushima, T.
登録日2012-12-07
公開日2013-03-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.99 Å)
主引用文献Structural Basis for the Recognition of Ubc13 by the Shigella flexneri Effector OspI.
J.Mol.Biol., 425, 2013
3W31
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Structual basis for the recognition of Ubc13 by the Shigella flexneri effector OspI
分子名称: IODIDE ION, ORF169b, Ubiquitin-conjugating enzyme E2 N
著者Nishide, A, Kim, M, Takagi, K, Sasakawa, C, Mizushima, T.
登録日2012-12-07
公開日2013-03-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.96 Å)
主引用文献Structural basis for the recognition of Ubc13 by the Shigella flexneri effector OspI.
J.Mol.Biol., 425, 2013
2KM4
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BU of 2km4 by Molmil
Solution structure of Rtt103 CTD interacting domain
分子名称: Regulator of Ty1 transposition protein 103
著者Lunde, B.M, Reichow, S, Kim, M, Leeper, T.C, Becker, R, Buratowski, S, Meinhart, A, Varani, G.
登録日2009-07-20
公開日2010-09-08
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Cooperative interaction of transcription termination factors with the RNA polymerase II C-terminal domain.
Nat.Struct.Mol.Biol., 17, 2010
7YA8
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BU of 7ya8 by Molmil
The crystal structure of IpaH2.5 LRR domain
分子名称: RING-type E3 ubiquitin transferase
著者Hiragi, K, Nishide, A, Takagi, K, Iwai, K, Kim, M, Mizushima, T.
登録日2022-06-27
公開日2023-02-08
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Structural insight into the recognition of the linear ubiquitin assembly complex by Shigella E3 ligase IpaH1.4/2.5.
J.Biochem., 173, 2023
7YA7
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BU of 7ya7 by Molmil
The crystal structure of IpaH1.4 LRR domain
分子名称: RING-type E3 ubiquitin transferase
著者Hiragi, K, Nishide, A, Takagi, K, Iwai, K, Kim, M, Mizushima, T.
登録日2022-06-27
公開日2023-02-08
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structural insight into the recognition of the linear ubiquitin assembly complex by Shigella E3 ligase IpaH1.4/2.5.
J.Biochem., 173, 2023

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