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PDB: 6 results

3FWQ
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BU of 3fwq by Molmil
Inactive conformation of human protein kinase CK2 catalytic subunit
Descriptor: CHLORIDE ION, Casein kinase II subunit alpha, GLYCEROL, ...
Authors:Niefind, K, Raaf, J, Issinger, O.G.
Deposit date:2009-01-19
Release date:2009-02-17
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:First inactive conformation of CK2 alpha, the catalytic subunit of protein kinase CK2
J.Mol.Biol., 386, 2009
4RLL
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BU of 4rll by Molmil
Crystal structure of human CK2alpha in complex with the ATP-competitive inhibitor 4-[(E)-(fluoren-9-ylidenehydrazinylidene)-methyl] benzoate
Descriptor: 4-[(E)-(9H-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid, Casein kinase II subunit alpha, GLYCEROL
Authors:Guerra, B, Rasmussen, T.D.L, Schnitzler, A, Jensen, H.H, Boldyreff, B.S, Miyata, Y, Marcussen, N, Niefind, K, Issinger, O.G.
Deposit date:2014-10-17
Release date:2014-12-17
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Protein kinase CK2 inhibition is associated with the destabilization of HIF-1 alpha in human cancer cells.
Cancer Lett, 356, 2015
1DAY
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BU of 1day by Molmil
CRYSTAL STRUCTURE OF A BINARY COMPLEX OF PROTEIN KINASE CK2 (ALPHA-SUBUNIT) AND MG-GMPPNP
Descriptor: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, PROTEIN KINASE CK2
Authors:Niefind, K, Puetter, M, Guerra, B, Issinger, O.G, Schomburg, D.
Deposit date:1999-11-01
Release date:2000-05-03
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:GTP plus water mimic ATP in the active site of protein kinase CK2.
Nat.Struct.Biol., 6, 1999
1DAW
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BU of 1daw by Molmil
CRYSTAL STRUCTURE OF A BINARY COMPLEX OF PROTEIN KINASE CK2 (ALPHA-SUBUNIT) AND MG-AMPPNP
Descriptor: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, PROTEIN KINASE CK2
Authors:Niefind, K, Puetter, M, Guerra, B, Issinger, O.G, Schomburg, D.
Deposit date:1999-11-01
Release date:2000-05-03
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:GTP plus water mimic ATP in the active site of protein kinase CK2.
Nat.Struct.Biol., 6, 1999
1JWH
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BU of 1jwh by Molmil
Crystal Structure of Human Protein Kinase CK2 Holoenzyme
Descriptor: Casein kinase II beta chain, Casein kinase II, alpha chain, ...
Authors:Niefind, K, Guerra, B, Ermakowa, I, Issinger, O.G.
Deposit date:2001-09-04
Release date:2002-03-04
Last modified:2023-08-16
Method:X-RAY DIFFRACTION (3.1 Å)
Cite:Crystal structure of human protein kinase CK2: insights into basic properties of the CK2 holoenzyme.
EMBO J., 20, 2001
4RLK
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BU of 4rlk by Molmil
Crystal structure of Z. mays CK2alpha in complex with the ATP-competitive inhibitor 4-[(E)-(fluoren-9-ylidenehydrazinylidene)-methyl] benzoate
Descriptor: 4-[(E)-(9H-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid, ACETATE ION, Casein kinase II subunit alpha, ...
Authors:Guerra, B, Rasmussen, T.D.L, Schnitzler, A, Jensen, H.H, Boldyreff, B.S, Miyata, Y, Marcussen, N, Niefind, K, Issinger, O.G.
Deposit date:2014-10-17
Release date:2014-12-17
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:Protein kinase CK2 inhibition is associated with the destabilization of HIF-1 alpha in human cancer cells.
Cancer Lett, 356, 2015

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