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PDB: 13 件

1SEG
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Crystal structure of a toxin chimera between Lqh-alpha-IT from the scorpion Leiurus quinquestriatus hebraeus and AAH2 from Androctonus australis hector
分子名称: AAH2: LQH-ALPHA-IT (FACE) CHIMERIC TOXIN, NITRATE ION, PROPANOIC ACID, ...
著者Karbat, I, Frolow, F, Froy, O, Gilles, N, Cohen, L, Turkov, M, Gordon, D, Gurevitz, M.
登録日2004-02-17
公開日2004-08-31
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Molecular basis of the high insecticidal potency of scorpion alpha-toxins.
J.Biol.Chem., 279, 2004
2I61
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Depressant anti-insect neurotoxin, LqhIT2 from Leiurus quinquestriatus hebraeus
分子名称: 1,2-ETHANEDIOL, ACETIC ACID, CARBON DIOXIDE, ...
著者Frolow, F, Gurevitz, M, Karbat, I, Turkov, M, Gordon, D.
登録日2006-08-27
公開日2006-12-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献X-ray Structure and Mutagenesis of the Scorpion Depressant Toxin LqhIT2 Reveals Key Determinants Crucial for Activity and Anti-Insect Selectivity.
J.Mol.Biol., 366, 2007
1LQH
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INSECTICIDAL ALPHA SCORPION TOXIN ISOLATED FROM THE VENOM OF SCORPION LEIURUS QUINQUESTRIATUS HEBRAEUS, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: INSECT TOXIN ALPHA
著者Tugarinov, V, Kustanovich, I, Zilberberg, N, Gurevitz, M, Anglister, J.
登録日1996-06-17
公開日1997-03-12
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structures of a highly insecticidal recombinant scorpion alpha-toxin and a mutant with increased activity.
Biochemistry, 36, 1997
1LQI
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INSECTICIDAL ALPHA SCORPION TOXIN ISOLATED FROM THE VENOM OF SCORPION LEIURUS QUINQUESTRIATUS HEBRAEUS, NMR, 29 STRUCTURES
分子名称: INSECT TOXIN ALPHA
著者Tugarinov, V, Kustanovich, I, Zilberberg, N, Gurevitz, M, Anglister, J.
登録日1996-06-17
公開日1997-03-12
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structures of a highly insecticidal recombinant scorpion alpha-toxin and a mutant with increased activity.
Biochemistry, 36, 1997
6ZOI
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A lid blocking mechanism of a cone snail toxin revealed at the atomic level
分子名称: Conknunitzin-C3 mutante
著者Saikia, C, Altman-Gueta, H, Dym, O, Frolow, F, Gurevitz, M, Gordon, D, Reuveny, E, Karbat, I.
登録日2020-07-07
公開日2021-07-14
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.798 Å)
主引用文献A lid blocking mechanism of a cone snail toxin revealed at the atomic level
To Be Published
1BCG
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SCORPION TOXIN BJXTR-IT
分子名称: TOXIN BJXTR-IT
著者Oren, D, Froy, O, Amit, E, Kleinberger-Doron, N, Gurevitz, M, Shaanan, B.
登録日1998-04-29
公開日1998-11-18
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献An excitatory scorpion toxin with a distinctive feature: an additional alpha helix at the C terminus and its implications for interaction with insect sodium channels.
Structure, 6, 1998
2YEO
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A39L mutation of scorpion toxin lqh-alpha-it
分子名称: 1,2-ETHANEDIOL, ALPHA-INSECT TOXIN LQHAIT, CHLORIDE ION, ...
著者Frolow, F, Kahn, R, Gurevitz, M.
登録日2011-03-28
公開日2011-04-13
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.08 Å)
主引用文献Crystal Structures of Scorpion Alpha-Toxinsmutants Reveal Conformational Constraints that Dictate Preference for Mammalian Brain Voltage-Gated Na- Channels
To be Published
6Q61
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Pore-modulating toxins exploit inherent slow inactivation to block K+ channels
分子名称: Kunitz-type conkunitzin-S1, SULFATE ION
著者Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E.
登録日2018-12-10
公開日2019-08-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Pore-modulating toxins exploit inherent slow inactivation to block K+channels.
Proc.Natl.Acad.Sci.USA, 116, 2019
6Q6C
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Pore-modulating toxins exploit inherent slow inactivation to block K+ channels
分子名称: 1,2-ETHANEDIOL, Kunitz-type conkunitzin-S1, NITRATE ION, ...
著者Karbat, I, Gueta, H, Fine, S, Szanto, T, Hamer-Rogotner, S, Dym, O, Frolow, F, Gordon, D, Panyi, G, Gurevitz, M, Reuveny, E.
登録日2018-12-10
公開日2019-08-21
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Pore-modulating toxins exploit inherent slow inactivation to block K+channels.
Proc.Natl.Acad.Sci.USA, 116, 2019
2ATB
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Triple mutant 8D9D10V of scorpion toxin LQH-alpha-IT
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, NITRATE ION, ...
著者Kahn, R, Karbat, I, Gurevitz, M, Frolow, F.
登録日2005-08-24
公開日2006-09-05
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献X-ray structures of Lqh-alpha-IT and Lqh-alpha-IT8D9D10V mutant
To be Published
2ASC
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Scorpion toxin LQH-alpha-IT
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, ETHANOL, ...
著者Kahn, R, Karbat, I, Gurevitz, M, Frolow, F.
登録日2005-08-23
公開日2006-09-05
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献X-ray structures of Lqh-alpha-IT and Lqh-alpha-IT8D9D10V mutant
To be Published
6YHT
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A lid blocking mechanism of a cone snail toxin revealed at the atomic level
分子名称: CITRIC ACID, Conk-C1, SULFATE ION
著者Saikia, C, Altman-Gueta, H, Dym, O, Frolow, F, Gurevitz, M, Gordon, D, Reuveny, E, Karbat, I.
登録日2020-03-31
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献A Molecular Lid Mechanism of K + Channel Blocker Action Revealed by a Cone Peptide.
J.Mol.Biol., 433, 2021
6YHY
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A lid blocking mechanism of a cone snail toxin revealed at the atomic level
分子名称: Conk-S1
著者Saikia, C, Altman-Gueta, H, Dym, O, Frolow, F, Gurevitz, M, Gordon, D, Reuveny, E, Karbat, I.
登録日2020-03-31
公開日2021-04-14
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献A Molecular Lid Mechanism of K + Channel Blocker Action Revealed by a Cone Peptide.
J.Mol.Biol., 433, 2021

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件を2024-07-31に公開中

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