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PDB: 2 results

4HV6
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BU of 4hv6 by Molmil
Structure of MNTR H77A mutant in apo- and mn-bound forms
Descriptor: MAGNESIUM ION, MANGANESE (II) ION, Transcriptional regulator MntR
Authors:Glasfeld, A, Grauer-Gray, K, McGuire, A.
Deposit date:2012-11-05
Release date:2012-11-21
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Roles of the A and C sites in the manganese-specific activation of MntR.
Biochemistry, 52, 2013
3VAP
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BU of 3vap by Molmil
Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity
Descriptor: 3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1H-pyrazol-4-yl)-6-methyl-8-[(3-{[(1R,3R)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-ium, Aurora kinase A
Authors:Voss, M.E, Rainka, M.P, Fleming, M, Peterson, L.H, Belanger, D.B, Siddiqui, M.A, Hruza, A, Voigt, J, Basso, A.D, Gray, K.
Deposit date:2011-12-29
Release date:2012-05-02
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (2.66 Å)
Cite:Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity.
Bioorg.Med.Chem.Lett., 22, 2012

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