PDB Search results for query - Protein Data Bank Japan

PDB: 1 results

Crystal structure of SMYD3 conjugate with piperidine-based covalent inhibitor EM127
Descriptor:	ACETATE ION, Histone-lysine N-methyltransferase SMYD3, N-[1-(2-Chloroacetyl)piperidin-4-yl]-5-cyclopropyl-1,2-oxazole-3-carboxamide, ...
Authors:	Talibov, V.O, Eriksson, D.
Deposit date:	2020-07-13
Release date:	2022-07-27
Last modified:	2024-01-31
Method:	X-RAY DIFFRACTION (1.55 Å)
Cite:	Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3 Eur.J.Med.Chem., 2022