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PDB: 1 results

3TN8
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BU of 3tn8 by Molmil
CDK9/cyclin T in complex with CAN508
Descriptor: 4-[(E)-(3,5-DIAMINO-1H-PYRAZOL-4-YL)DIAZENYL]PHENOL, Cyclin-T1, Cyclin-dependent kinase 9, ...
Authors:Baumli, S, Hole, A.J, Endicott, J.E.
Deposit date:2011-09-01
Release date:2012-02-15
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.95 Å)
Cite:The CDK9 C-helix Exhibits Conformational Plasticity That May Explain the Selectivity of CAN508.
Acs Chem.Biol., 7, 2012

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