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PDB: 1 results

7ZH8
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BU of 7zh8 by Molmil
DYRK1a in Complex with a Bromo-Triazolo-Pyridine
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 6-bromanyl-3H-[1,2,3]triazolo[4,5-b]pyridine, CHLORIDE ION, ...
Authors:Dammann, M, Stahlecker, J, Stehle, T, Boeckler, F.M.
Deposit date:2022-04-05
Release date:2022-11-09
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Screening of a Halogen-Enriched Fragment Library Leads to Unconventional Binding Modes.
J.Med.Chem., 65, 2022

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