PDB クエリの検索結果 - 日本蛋白質構造データバンク

PDB: 3 件

Selective pharmacological inhibition of the CREB binding protein bromodomain regulates inflammatory cytokines in macrophages and RGS4 in neurons
分子名称:	5-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[2-(4-methoxyphenyl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-1H-benzimidazole, CREB-binding protein
著者	Chekler, E.L, Jones, L.H.
登録日	2015-07-09
公開日	2016-04-20
最終更新日	2023-09-27
実験手法	X-RAY DIFFRACTION (1.96 Å)
主引用文献	Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. Chem.Biol., 22, 2015

Selective pharmacological inhibition of the CREB binding protein bromodomain regulates inflammatory cytokines in macrophages and RGS4 in neurons
分子名称:	5-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[2-(4-methoxyphenyl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-1H-benzimidazole, Bromodomain-containing protein 4
著者	Chekler, E.L, Jones, L.H.
登録日	2015-07-08
公開日	2016-04-20
最終更新日	2023-09-27
実験手法	X-RAY DIFFRACTION (1.15 Å)
主引用文献	Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. Chem.Biol., 22, 2015

Direct photocapture of bromodomains using tropolone chemical probes
分子名称:	1,2-ETHANEDIOL, 2-methoxy-4-{1-[2-(morpholin-4-yl)ethyl]-2-(2-phenylethyl)-1H-benzimidazol-5-yl}cyclohepta-2,4,6-trien-1-one, Bromodomain-containing protein 4
著者	Hett, E.C, Piatnitski Chekler, E.L, Basak, A, Bonin, P.D, Denny, R.A, Flick, A.C, Geoghegan, K.F, Liu, S, Pletcher, M.T, Robinson, R.P, Sahasrabudhe, P, Salter, S, Stock, I.A, Jones, L.H.
登録日	2014-09-23
公開日	2015-10-28
最終更新日	2023-12-27
実験手法	X-RAY DIFFRACTION (1.345 Å)
主引用文献	Direct photocapture of bromodomains using tropolone chemical probes To Be Published