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PDB: 2 results

4H1Q
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BU of 4h1q by Molmil
Crystal structure of mutant MMP-9 catalytic domain in complex with a twin inhibitor.
Descriptor: CALCIUM ION, Matrix metalloproteinase-9, N-(4-{[(3R)-3-[(biphenyl-4-ylsulfonyl)(propan-2-yloxy)amino]-4-(hydroxyamino)-4-oxobutyl]amino}-4-oxobutyl)-N'-(4-{[(3S)-3-[(biphenyl-4-ylsulfonyl)(propan-2-yloxy)amino]-4-(hydroxyamino)-4-oxobutyl]amino}-4-oxobutyl)benzene-1,3-dicarboxamide, ...
Authors:Stura, E.A, Vera, L, Cassar-Lajeunesse, E, Nuti, E, Catalani, M.P, Dive, V, Rossello, A.
Deposit date:2012-09-11
Release date:2013-04-24
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.59 Å)
Cite:Crystallization of bi-functional ligand protein complexes.
J.Struct.Biol., 182, 2013
4H2E
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BU of 4h2e by Molmil
Crystal structure of an MMP twin inhibitor complexing two MMP-9 catalytic domains
Descriptor: ACETATE ION, BICINE, CALCIUM ION, ...
Authors:Stura, E.A, Vera, L, Cassar-Lajeunesse, E, Nuti, E, Catalani, M.P, Dive, V, Rossello, A.
Deposit date:2012-09-12
Release date:2013-04-24
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.902 Å)
Cite:Crystallization of bi-functional ligand protein complexes.
J.Struct.Biol., 182, 2013

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