Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 22 件

5C9N
DownloadVisualize
BU of 5c9n by Molmil
Crystal structure of GEMC1 coiled-coil domain
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, Geminin coiled-coil domain-containing protein 1
著者Caillat, C, Perrakis, A.
登録日2015-06-28
公開日2015-11-11
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The structure of the GemC1 coiled coil and its interaction with the Geminin family of coiled-coil proteins.
Acta Crystallogr.,Sect.D, 71, 2015
6SNC
DownloadVisualize
BU of 6snc by Molmil
crystal structure of LN01 Fab in complex with an HIV-1 gp41 peptide
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp160, LNO1 Heavy Chain, ...
著者Caillat, C, Pinto, D, Corti, D, Fenwick, C, Pantaleo, G, Weissenhorn, W.
登録日2019-08-23
公開日2019-11-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural Basis for Broad HIV-1 Neutralization by the MPER-Specific Human Broadly Neutralizing Antibody LN01.
Cell Host Microbe, 26, 2019
6SNE
DownloadVisualize
BU of 6sne by Molmil
crystal structure of LN01 Fab in complex with an HIV-1 gp41 peptide
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp160, LN01 heavy chain, ...
著者Caillat, C, Pinto, D, Corti, D, Fenwick, C, Pantaleo, G, Weissenhorn, W.
登録日2019-08-23
公開日2019-11-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.9 Å)
主引用文献Structural Basis for Broad HIV-1 Neutralization by the MPER-Specific Human Broadly Neutralizing Antibody LN01.
Cell Host Microbe, 26, 2019
6SND
DownloadVisualize
BU of 6snd by Molmil
crystal structure of LN01 Fab in complex with an HIV-1 gp41 peptide
分子名称: 1,2-DICAPROYL-SN-PHOSPHATIDYL-L-SERINE, 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp160, ...
著者Caillat, C, Pinto, D, Corti, D, Fenwick, C, Pantaleo, G, Weissenhorn, W.
登録日2019-08-23
公開日2019-11-06
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for Broad HIV-1 Neutralization by the MPER-Specific Human Broadly Neutralizing Antibody LN01.
Cell Host Microbe, 26, 2019
7AEJ
DownloadVisualize
BU of 7aej by Molmil
Crystal structure of asymmetric HIV-1 gp41 containing all membrane anchors
分子名称: 2H10, Envelope glycoprotein gp160,Envelope glycoprotein gp160
著者Caillat, C, Guilligay, D, Weissenhorn, W.
登録日2020-09-17
公開日2021-05-26
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Structure of HIV-1 gp41 with its membrane anchors targeted by neutralizing antibodies.
Elife, 10, 2021
4BRY
DownloadVisualize
BU of 4bry by Molmil
The Idas:Geminin heterodimeric parallel coiled-coil
分子名称: GEMININ, MULTICILIN, PHOSPHATE ION, ...
著者Caillat, C, Perrakis, A.
登録日2013-06-06
公開日2013-10-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献The Geminin and Idas Coiled Coils Preferentially Form a Heterodimer that Inhibits Geminin Function in DNA Replication Licensing
J.Biol.Chem., 288, 2013
2XX3
DownloadVisualize
BU of 2xx3 by Molmil
HUMAN THYMIDYLATE KINASE COMPLEXED WITH thymidine butenyl phosphonate monophosphate and ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, N1-[(E)-4-DIHYDROXYPHOSPHONYL-BUT-2-ENYL]-THYMINE, ...
著者Caillat, C, Meyer, P.
登録日2010-11-08
公開日2011-12-07
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Novel Antiviral C5-Substituted Pyrimidine Acyclic Nucleoside Phosphonates Selected as Human Thymidylate Kinase Substrates.
J.Med.Chem., 54, 2011
4D81
DownloadVisualize
BU of 4d81 by Molmil
Metallosphera sedula Vps4 crystal structure
分子名称: AAA ATPase, central domain protein, ADENOSINE-5'-DIPHOSPHATE
著者Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P.
登録日2014-12-02
公開日2015-11-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly.
Nat.Commun., 6, 2015
5O2U
DownloadVisualize
BU of 5o2u by Molmil
Llama VHH in complex with p24
分子名称: Capsid protein p24, VHH 59H10
著者Caillat, C, Verrips, T, Weissenhorn, W.
登録日2017-05-22
公開日2017-06-21
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.76 Å)
主引用文献Unravelling the Molecular Basis of High Affinity Nanobodies against HIV p24: In Vitro Functional, Structural, and in Silico Insights.
ACS Infect Dis, 3, 2017
2V54
DownloadVisualize
BU of 2v54 by Molmil
Crystal structure of vaccinia virus thymidylate kinase bound to TDP
分子名称: MAGNESIUM ION, PYROPHOSPHATE 2-, THYMIDINE-5'-DIPHOSPHATE, ...
著者Caillat, C, Topalis, D, Agrofoglio, L.A, Pochet, S, Balzarini, J, Deville-Bonne, D, Meyer, P.
登録日2008-10-01
公開日2008-10-21
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal Structure of Poxvirus Thymidylate Kinase: An Unexpected Dimerization Has Implications for Antiviral Therapy
Proc.Natl.Acad.Sci.USA, 105, 2008
2W0S
DownloadVisualize
BU of 2w0s by Molmil
Crystal structure of vaccinia virus thymidylate kinase bound to brivudin-5'-monophosphate
分子名称: (E)-5-(2-BROMOVINYL)-2'-DEOXYURIDINE-5'-MONOPHOSPHATE, MAGNESIUM ION, SULFATE ION, ...
著者Caillat, C, Topalis, D, Agrofoglio, L.A, Pochet, S, Balzarini, J, Deville-Bonne, D, Meyer, P.
登録日2008-10-08
公開日2008-10-21
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.918 Å)
主引用文献Crystal Structure of Poxvirus Thymidylate Kinase: An Unexpected Dimerization Has Implications for Antiviral Therapy
Proc.Natl.Acad.Sci.USA, 105, 2008
4D82
DownloadVisualize
BU of 4d82 by Molmil
Metallosphera sedula Vps4 crystal structure
分子名称: AAA ATPase, central domain protein, ADENOSINE-5'-DIPHOSPHATE
著者Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P.
登録日2014-12-02
公開日2015-11-25
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly.
Nat.Commun., 6, 2015
4D80
DownloadVisualize
BU of 4d80 by Molmil
Metallosphera sedula Vps4 crystal structure
分子名称: AAA ATPASE, CENTRAL DOMAIN PROTEIN
著者Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P.
登録日2014-12-02
公開日2015-10-28
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly.
Nat.Commun., 6, 2015
7AJ6
DownloadVisualize
BU of 7aj6 by Molmil
LN02 Fab
分子名称: LN02, LN02 heavy chain
著者Caillat, C, Fenwick, G, Pantaleo, G, Weissenhorn, W.
登録日2020-09-28
公開日2021-10-06
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献LN02 Fab
To Be Published
8WU1
DownloadVisualize
BU of 8wu1 by Molmil
Cryo-EM structure of CB1-beta-arrestin1 complex
分子名称: Beta-arrestin-1, Cannabinoid receptor 1,Vasopressin V2 receptor, Fab30 heavy chain, ...
著者Liao, Y, Zhang, H, Shen, Q, Cai, C.
登録日2023-10-19
公開日2024-03-20
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Cryo-EM structure of CB1-beta-arrestin1 complex
to be published
2AWW
DownloadVisualize
BU of 2aww by Molmil
Synapse associated protein 97 PDZ2 domain variant C378G with C-terminal GluR-A peptide
分子名称: 18-residue C-terminal peptide from glutamate receptor, ionotropic, AMPA1, ...
著者Von Ossowski, I, Oksanen, E, Von Ossowski, L, Cai, C, Sundberg, M, Goldman, A, Keinanen, K.
登録日2005-09-02
公開日2006-08-29
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献Crystal structure of the second PDZ domain of SAP97 in complex with a GluR-A C-terminal peptide
Febs J., 273, 2006
2AWX
DownloadVisualize
BU of 2awx by Molmil
Synapse associated protein 97 PDZ2 domain variant C378S
分子名称: HISTIDINE, Synapse associated protein 97
著者Von Ossowski, I, Oksanen, E, Von Ossowski, L, Cai, C, Sundberg, M, Goldman, A, Keinanen, K.
登録日2005-09-02
公開日2006-08-29
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of the second PDZ domain of SAP97 in complex with a GluR-A C-terminal peptide
Febs J., 273, 2006
2AWU
DownloadVisualize
BU of 2awu by Molmil
Synapse associated protein 97 PDZ2 domain variant C378G
分子名称: AHH, Synapse-associated protein 97
著者Von Ossowski, I, Oksanen, E, Von Ossowski, L, Cai, C, Sundberg, M, Goldman, A, Keinanen, K.
登録日2005-09-02
公開日2006-08-29
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Crystal structure of the second PDZ domain of SAP97 in complex with a GluR-A C-terminal peptide
Febs J., 273, 2006
2FS4
DownloadVisualize
BU of 2fs4 by Molmil
Ketopiperazine-Based Renin Inhibitors: Optimization of the C ring
分子名称: (6R)-6-({[1-(3-HYDROXYPROPYL)-1,7-DIHYDROQUINOLIN-7-YL]OXY}METHYL)-1-(4-{3-[(2-METHOXYBENZYL)OXY]PROPOXY}PHENYL)PIPERAZIN-2-ONE, Renin
著者Holsworth, D.D, Cai, C, Cheng, X.-M, Cody, W.L, Downing, D.M, Erasga, N, Lee, C, Powell, N.A, Edmunds, J.J, Stier, M, Jalaie, M, Zhang, E, McConnell, P, Ryan, M.J, Bryant, J, Li, T, Kasani, A, Hall, E, Subedi, R, Rahim, M, Maiti, S.
登録日2006-01-20
公開日2006-06-13
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Ketopiperazine-Based Renin Inhibitors: Optimization of the "C" Ring
BIOORG.MED.CHEM.LETT., 16, 2006
2G2L
DownloadVisualize
BU of 2g2l by Molmil
Crystal Structure of the Second PDZ Domain of SAP97 in Complex with a GluR-A C-terminal Peptide
分子名称: 18-mer peptide from glutamate receptor, ionotropic, AMPA1, ...
著者Von Ossowski, I, Oksanen, E, Von Ossowski, L, Cai, C, Sundberg, M, Goldman, A, Keinanen, K.
登録日2006-02-16
公開日2006-08-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structure of the second PDZ domain of SAP97 in complex with a GluR-A C-terminal peptide
Febs J., 273, 2006
5HM1
DownloadVisualize
BU of 5hm1 by Molmil
Llama VHH 2E7 in complex with gp41
分子名称: gp41, lama VHH antibody 2E7
著者Hock, M, Caillat, C, Haffke, M, Weissenhorn, W.
登録日2016-01-15
公開日2017-01-25
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.962 Å)
主引用文献Structure of HIV neutralizing VHH 2E7 in complex with gp41 peptide
To Be Published
4U01
DownloadVisualize
BU of 4u01 by Molmil
HCV NS3/4A serine protease in complex with 6570
分子名称: (2S,3aS,10Z,11aS,12aR)-2-({8-fluoro-7-methoxy-2-[4-(propan-2-yl)-1,3-thiazol-2-yl]quinolin-4-yl}oxy)-5-methyl-N-[(1-methylcyclopropyl)sulfonyl]-4,14-dioxo-1,2,3,3a,4,5,6,7,8,9,11a,12,13,14-tetradecahydro-12aH-cyclopropa[m]pyrrolo[1,2-c][1,3,6]triazacyclotetradecine-12a-carboxamide, CHLORIDE ION, NS4A protein, ...
著者Parsy, C.C, Alexandre, F.-R, Brandt, G, Caillet, C, Chaves, D, Derock, M, Gloux, D, Griffon, Y, Lallos, L.B, Leroy, F, Liuzzi, M, Loi, A.-G, Mayes, B, Moulat, L, Moussa, A, Chiara, M, Roques, V, Rosinovsky, E, Seifer, M, Stewart, A, Wang, J, Standring, D, Surleraux, D.
登録日2014-07-11
公開日2015-07-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery and structural diversity of the hepatitis C virus NS3/4A serine protease inhibitor series leading to clinical candidate IDX320.
Bioorg.Med.Chem.Lett., 25, 2015

221371

件を2024-06-19に公開中

PDB statisticsPDBj update infoContact PDBjnumon