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PDB: 12 件

1Q5K
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crystal structure of Glycogen synthase kinase 3 in complexed with inhibitor
分子名称: Glycogen synthase kinase-3 beta, N-(4-METHOXYBENZYL)-N'-(5-NITRO-1,3-THIAZOL-2-YL)UREA
著者Bhat, R, Xue, Y, Berg, S, Hellberg, S, Ormo, M, Nilsson, Y, Radesater, A.C, Jerning, E, Markgren, P.O, Borgegard, T, Nylof, M, Gimenez-Cassina, A, Hernandez, F, Lucas, J.J, Diaz-Mido, J, Avila, J.
登録日2003-08-08
公開日2004-08-10
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Structural insights and biological effects of glycogen synthase kinase 3-specific inhibitor AR-A014418.
J.Biol.Chem., 278, 2003
1H7C
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human tubulin chaperone cofactor a
分子名称: ACETIC ACID, SULFATE ION, TUBULIN-SPECIFIC CHAPERONE A
著者Guasch, A, Aloria, K, Perez, R, Campo, R, Avila, J, Zabala, J.C, Coll, M.
登録日2001-07-04
公開日2002-06-13
最終更新日2017-08-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Three-Dimensional Structure of Human Tubulin Chaperone Cofactor A
J.Mol.Biol., 318, 2002
1AFP
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SOLUTION STRUCTURE OF THE ANTIFUNGAL PROTEIN FROM ASPERGILLUS GIGANTEUS. EVIDENCE FOR DISULPHIDE CONFIGURATIONAL ISOMERISM
分子名称: ANTIFUNGAL PROTEIN FROM ASPERGILLUS GIGANTEUS
著者Campos-Olivas, R, Bruix, M, Santoro, J, Lacadena, J, Del Pozo, A.M, Gavilanes, J.G, Rico, M.
登録日1994-11-11
公開日1995-02-07
最終更新日2024-04-10
実験手法SOLUTION NMR
主引用文献NMR solution structure of the antifungal protein from Aspergillus giganteus: evidence for cysteine pairing isomerism.
Biochemistry, 34, 1995
1DE3
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BU of 1de3 by Molmil
SOLUTION STRUCTURE OF THE CYTOTOXIC RIBONUCLEASE ALPHA-SARCIN
分子名称: RIBONUCLEASE ALPHA-SARCIN
著者Perez-Canadillas, J.M, Campos-Olivas, R, Santoro, J, Lacadena, J, Martinez del Pozo, A, Gavilanes, J.G, Rico, M, Bruix, M.
登録日1999-11-12
公開日2000-06-21
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献The highly refined solution structure of the cytotoxic ribonuclease alpha-sarcin reveals the structural requirements for substrate recognition and ribonucleolytic activity.
J.Mol.Biol., 299, 2000
1O71
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Crystal structure of the water-soluble state of the pore-forming cytolysin Sticholysin II complexed with glycerol
分子名称: GLYCEROL, STICHOLYSIN II
著者Mancheno, J.M, Martinez-Ripoll, M, Gavilanes, J.G, Hermoso, J.A.
登録日2002-10-23
公開日2003-11-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Crystal and Electron Microscopy Structures of Sticholysin II Actinoporin Reveal Insights Into the Mechanism of Membrane Pore Formation
Structure, 11, 2003
1O72
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Crystal structure of the water-soluble state of the pore-forming cytolysin Sticholysin II complexed with phosphorylcholine
分子名称: PHOSPHOCHOLINE, STICHOLYSIN II
著者Mancheno, J.M, Martinez-Ripoll, M, Gavilanes, J.G, Hermoso, J.A.
登録日2002-10-23
公開日2003-11-13
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献Crystal and Electron Microscopy Structures of Sticholysin II Actinoporin Reveal Insights Into the Mechanism of Membrane Pore Formation
Structure, 11, 2003
1GWY
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BU of 1gwy by Molmil
Crystal structure of the water-soluble state of the pore-forming cytolysin Sticholysin II
分子名称: STICHOLYSIN II, SULFATE ION
著者Mancheno, J.M, Martin-Benito, J, Martinez-Ripoll, M, Gavilanes, J.G, Hermoso, J.A.
登録日2002-03-26
公開日2003-06-12
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Crystal and Electron Microscopy Structures of Sticholysin II Actinoporin Reveal Insights Into the Mechanism of Membrane Pore Formation
Structure, 11, 2003
6XB7
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BU of 6xb7 by Molmil
IRES-targeting Small Molecule Inhibits Enterovirus 71 Replication via Allosteric Stabilization of a Ternary Complex
分子名称: 3-amino-N-(diaminomethylidene)-5-(dimethylamino)-6-(phenylethynyl)pyrazine-2-carboxamide, RNA (41-MER)
著者Tolbert, B.S, Davila, J, Sugarman, A.L, Chiu, L.Y.
登録日2020-06-05
公開日2020-09-02
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献IRES-targeting small molecule inhibits enterovirus 71 replication via allosteric stabilization of a ternary complex.
Nat Commun, 11, 2020
1R4Y
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SOLUTION STRUCTURE OF THE DELETION MUTANT DELTA(7-22) OF THE CYTOTOXIC RIBONUCLEASE ALPHA-SARCIN
分子名称: Ribonuclease alpha-sarcin
著者Garcia-Mayoral, M.F, Garcia-Ortega, L, Lillo, M.P, Santoro, J, Martinez Del Pozo, A, Gavilanes, J.G, Rico, M, Bruix, M.
登録日2003-10-09
公開日2004-04-06
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献NMR structure of the noncytotoxic {alpha}-sarcin mutant {Delta}(7-22): The importance of the native conformation of peripheral loops for activity.
Protein Sci., 13, 2004
2L38
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R29Q Sticholysin II mutant
分子名称: Sticholysin-2
著者Castrillo, I, Alegre-Cebollada, J, Martinez-del-Pozo, A, Gavilanes, J, Bruix, M.
登録日2010-09-10
公開日2010-09-22
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献NMR Structure of StnIIR29Q, a defective lipid binding mutant of the sea anemone actinoporin Sticholysin II
To be Published
1S0Q
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Native Bovine Pancreatic Trypsin
分子名称: CALCIUM ION, Trypsinogen
著者Garcia-Granda, S, Chamorro Gavilanes, J.A.
登録日2004-01-02
公開日2005-01-18
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.02 Å)
主引用文献Pancratic bovine Trypsin native and inhibited with Benzamidine from synchotron data.
To be Published
1S0R
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Bovine Pancreatic Trypsin inhibited with Benzamidine at Atomic resolution
分子名称: BENZAMIDINE, CALCIUM ION, Trypsinogen
著者Chamorro Gavilanes, J.A, Garca-Granda, S.
登録日2004-01-02
公開日2005-01-18
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.02 Å)
主引用文献Pancratic bovine Trypsin native and inhibited with Benzamidine from synchotron data.
To be Published

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件を2024-07-31に公開中

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