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PDB: 1 results

3S3I
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p38 kinase crystal structure in complex with small molecule inhibitor
Descriptor: 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-N-cyclopropyl-4-methylbenzamide, Mitogen-activated protein kinase 14
Authors:Segarra, V, Aiguade, J, Roca, R, Fisher, M, Lamers, M.
Deposit date:2011-05-18
Release date:2012-04-04
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Novel triazolopyridylbenzamides as potent and selective p38 alpha inhibitors.
Bioorg.Med.Chem.Lett., 22, 2012

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