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5J5T
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BU of 5j5t by Molmil
GLK co-crystal structure with aminopyrrolopyrimidine inhibitor
Descriptor: 5-[2-(piperidin-4-yl)-1,3-thiazol-5-yl]-3-[(pyridin-4-yl)methoxy]pyridin-2-amine, Mitogen-activated protein kinase kinase kinase kinase 3
Authors:Silvian, L.F, Marcotte, D.
Deposit date:2016-04-03
Release date:2016-10-26
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (2.85 Å)
Cite:Germinal-center kinase-like kinase co-crystal structure reveals a swapped activation loop and C-terminal extension.
Protein Sci., 26, 2017
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