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3T8M
Rational Design of PI3K-alpha Inhibitors that Exhibit Selectivity Over the PI3K-beta Isoform
Descriptor:
N~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-N~2~,N~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamide, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Authors:
Murray, J.M
,
Wiesmann, C.
Deposit date:
2011-08-01
Release date:
2011-11-16
Last modified:
2024-02-28
Method:
X-RAY DIFFRACTION (2.5 Å)
Cite:
Rational Design of PI3K-alpha Inhibitors that Exhibit Selectivity Over the PI3K-beta Isoform
To be Published
2KLL
Solution structure of human interleukin-33
Descriptor:
Interleukin-33
Authors:
Lingel, A
,
Fairbrother, W.
Deposit date:
2009-07-06
Release date:
2009-11-17
Last modified:
2023-06-14
Method:
SOLUTION NMR
Cite:
Structure of IL-33 and its interaction with the ST2 and IL-1RAcP receptors--insight into heterotrimeric IL-1 signaling complexes.
Structure, 17, 2009
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PDB entries from 2024-04-24