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4CE2
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BU of 4ce2 by Molmil
Hsp90 N-terminal domain bound to macrolactam analogues of radicicol.
Descriptor: (9E)-19-CHLORANYL-13-METHYL-16,18-BIS(OXIDANYL)-13-AZABICYCLO[13.4.0]NONADECA-1(15),9,16,18-TETRAENE-3,14-DIONE, ATP-DEPENDENT MOLECULAR CHAPERONE HSP82
Authors:Roe, S.M, Parry-Morris, S, Prodromou, C.
Deposit date:2013-11-08
Release date:2014-01-29
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.38 Å)
Cite:Synthesis of macrolactam analogues of radicicol and their binding to heat shock protein Hsp90.
Org. Biomol. Chem., 12, 2014
4CE3
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BU of 4ce3 by Molmil
Hsp90 N-terminal domain bound to macrolactam analogues of radicicol.
Descriptor: 13-Chloro-14,16-dihydroxy-2-methyl-2,3,4,5,9,10-hexahydrobenz[c][1]azacyclotetradecine-1,11(8H,12H)-dione, ATP-DEPENDENT MOLECULAR CHAPERONE HSP82
Authors:Roe, S.M, Parry-Morris, S, Prodromou, C.
Deposit date:2013-11-08
Release date:2014-01-29
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.31 Å)
Cite:Synthesis of Macrolactam Analogues of Radicicol and Their Binding to Heat Shock Protein Hsp90.
Org.Biomol.Chem., 12, 2014
4CE1
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BU of 4ce1 by Molmil
Hsp90 N-terminal domain bound to macrolactam analogues of radicicol.
Descriptor: 15-Chloro-16,18-dihydroxy-2-methyl-3,4,7,8,9,10,11,12-octahydrobenz[c][1]azacyclohexadecine-1,13(2H,14H)-dione, ATP-DEPENDENT MOLECULAR CHAPERONE HSP82
Authors:Roe, S.M, Parry-Morris, S, Prodromou, C.
Deposit date:2013-11-08
Release date:2014-01-29
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.01 Å)
Cite:Synthesis of Macrolactam Analogues of Radicicol and Their Binding to Heat Shock Protein Hsp90.
Org.Biomol.Chem., 12, 2014
7AKO
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BU of 7ako by Molmil
Crystal structure of CHK1 kinase domain in complex with a CLASPIN phosphopeptide
Descriptor: 1,2-ETHANEDIOL, Claspin, STAUROSPORINE, ...
Authors:Day, M, Oliver, A.W, Pearl, L.H.
Deposit date:2020-10-01
Release date:2021-04-14
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Structural basis for recruitment of the CHK1 DNA damage kinase by the CLASPIN scaffold protein.
Structure, 29, 2021
7AKM
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BU of 7akm by Molmil
Crystal structure of CHK1 kinase domain in complex with ATPyS
Descriptor: 1,2-ETHANEDIOL, CITRIC ACID, MAGNESIUM ION, ...
Authors:Day, M, Oliver, A.W, Pearl, L.H.
Deposit date:2020-10-01
Release date:2021-04-14
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.93 Å)
Cite:Structural basis for recruitment of the CHK1 DNA damage kinase by the CLASPIN scaffold protein.
Structure, 29, 2021
4CGV
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BU of 4cgv by Molmil
First TPR of Spaghetti (RPAP3) bound to HSP90 peptide SRMEEVD
Descriptor: GLYCEROL, HEAT SHOCK PROTEIN HSP 90-ALPHA, RNA POLYMERASE II-ASSOCIATED PROTEIN 3
Authors:Roe, S.M, Pal, M.
Deposit date:2013-11-26
Release date:2014-05-14
Last modified:2014-06-25
Method:X-RAY DIFFRACTION (2.54 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CHH
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BU of 4chh by Molmil
N-terminal domain of yeast PIH1p
Descriptor: 1,2-ETHANEDIOL, PROTEIN INTERACTING WITH HSP90 1
Authors:Roe, S.M, Pal, M.
Deposit date:2013-12-02
Release date:2014-05-14
Last modified:2014-06-25
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CGU
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BU of 4cgu by Molmil
Full length Tah1 bound to yeast PIH1 and HSP90 peptide SRMEEVD
Descriptor: GLYCEROL, HEAT SHOCK PROTEIN HSP 90-ALPHA, PROTEIN INTERACTING WITH HSP90 1, ...
Authors:Roe, S.M, Pal, M.
Deposit date:2013-11-26
Release date:2014-05-14
Last modified:2017-06-28
Method:X-RAY DIFFRACTION (2.11 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CV4
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BU of 4cv4 by Molmil
PIH N-terminal domain
Descriptor: COBALT (II) ION, PIH1 DOMAIN-CONTAINING PROTEIN 1, SULFATE ION
Authors:Morgan, R.M, Roe, S.M.
Deposit date:2014-03-23
Release date:2014-05-14
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.902 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CSE
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BU of 4cse by Molmil
PIH N-terminal domain
Descriptor: PIH1 DOMAIN-CONTAINING PROTEIN 1, TELOMERE LENGTH REGULATION PROTEIN TEL2 HOMOLOG
Authors:Morgan, R.M, Roe, S.M.
Deposit date:2014-03-07
Release date:2014-05-14
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (3.3 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CGW
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BU of 4cgw by Molmil
Second TPR of Spaghetti (RPAP3) bound to HSP90 peptide SRMEEVD
Descriptor: HEAT SHOCK PROTEIN HSP 90-ALPHA, RNA POLYMERASE II-ASSOCIATED PROTEIN 3
Authors:Roe, S.M, Pal, M.
Deposit date:2013-11-26
Release date:2014-05-14
Last modified:2014-06-25
Method:X-RAY DIFFRACTION (3.001 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014
4CKT
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BU of 4ckt by Molmil
PIH1 N-terminal domain
Descriptor: PIH1 DOMAIN-CONTAINING PROTEIN 1, TELOMERE LENGTH REGULATION PROTEIN TEL2 HOMOLOG
Authors:Morgan, R.M, Roe, S.M.
Deposit date:2014-01-08
Release date:2014-05-14
Last modified:2014-06-25
Method:X-RAY DIFFRACTION (3 Å)
Cite:Structural Basis for Phosphorylation-Dependent Recruitment of Tel2 to Hsp90 by Pih1.
Structure, 22, 2014

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