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5TYH
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BU of 5tyh by Molmil
PglD from Campylobacter jejuni NCTC 11168 in complex with 5-(2-furanyl)-1H-pyrazole-3-carboxylic acid
分子名称: 3-(furan-2-yl)-1H-pyrazole-5-carboxylic acid, UDP-N-acetylbacillosamine N-acetyltransferase
著者Morrison, J.P, Imperiali, B.
登録日2016-11-20
公開日2017-04-12
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Targeting Bacillosamine Biosynthesis in Bacterial Pathogens: Development of Inhibitors to a Bacterial Amino-Sugar Acetyltransferase from Campylobacter jejuni.
J. Med. Chem., 60, 2017
2X6T
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BU of 2x6t by Molmil
AGME bound to ADP-B-mannose
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADP-L-GLYCERO-D-MANNO-HEPTOSE-6-EPIMERASE, CHLORIDE ION, ...
著者Kowatz, T, Morrison, J.P, Tanner, M.E, Naismith, J.H.
登録日2010-02-21
公開日2010-03-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献The Crystal Structure of the Y140F Mutant of Adp-L-Glycero-D-Manno-Heptose 6-Epimerase Bound to Adp-Beta-D-Mannose Suggests a One Base Mechanism.
Protein Sci., 19, 2010
2X86
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BU of 2x86 by Molmil
AGME bound to ADP-B-mannose
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADP-L-GLYCERO-D-MANNO-HEPTOSE-6-EPIMERASE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Kowatz, T, Morrison, J.P, Tanner, M.E, Naismith, J.H.
登録日2010-03-06
公開日2010-03-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Crystal Structure of the Y140F Mutant of Adp-L-Glycero-D-Manno-Heptose 6-Epimerase Bound to Adp-Beta-D-Mannose Suggests a One Base Mechanism.
Protein Sci., 19, 2010
5T2Y
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BU of 5t2y by Molmil
Crystal Structure of C. jejuni PglD in complex with 5-methyl-4-(methylamino)-2-phenethylthieno[2,3-d]pyrimidine-6-carboxylic acid
分子名称: 5-methyl-4-(methylamino)-2-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxylic acid, DIMETHYL SULFOXIDE, GLYCEROL, ...
著者De Schutter, J.W, Imperiali, B.
登録日2016-08-24
公開日2017-02-22
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Targeting Bacillosamine Biosynthesis in Bacterial Pathogens: Development of Inhibitors to a Bacterial Amino-Sugar Acetyltransferase from Campylobacter jejuni.
J. Med. Chem., 60, 2017

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件を2024-05-15に公開中

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