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1B45
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ALPHA-CNIA CONOTOXIN FROM CONUS CONSORS, NMR, 43 STRUCTURES
分子名称: ALPHA-CNIA
著者Favreau, P, Krimm, I, Le Gall, F, Bobenrieth, M.J, Lamthanh, H, Bouet, F, Servent, D, Molgo, J, Menez, A, Letourneux, Y, Lancelin, J.M.
登録日1999-01-05
公開日1999-07-09
最終更新日2022-02-16
実験手法SOLUTION NMR
主引用文献Biochemical characterization and nuclear magnetic resonance structure of novel alpha-conotoxins isolated from the venom of Conus consors.
Biochemistry, 38, 1999
2YEN
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Solution structure of the skeletal muscle and neuronal voltage gated sodium channel antagonist mu-conotoxin CnIIIC
分子名称: Mu-conotoxin CnIIIC
著者Favreau, P, Benoit, E, Hocking, H.G, Carlier, L, D'hoedt, D, Leipold, E, Markgraf, R, Schlumberger, S, Cordova, M.A, Gaertner, H, Paolini-Bertrand, M, Hartley, O, Tytgat, J, Heinemann, S.H, Bertrand, D, Boelens, R, Stocklin, R, Molgo, J.
登録日2011-03-28
公開日2012-02-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献A Novel Mu-Conopeptide, Cniiic, Exerts Potent and Preferential Inhibition of Na(V) 1.2/1.4 Channels and Blocks Neuronal Nicotinic Acetylcholine Receptors.
Br.J.Pharmacol., 166, 2012
2X00
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CRYSTAL STRUCTURE OF A-ACHBP IN COMPLEX WITH GYMNODIMINE A
分子名称: GYMNODIMINE A, SOLUBLE ACETYLCHOLINE RECEPTOR
著者Bourne, Y, Radic, Z, Araoz, R, Talley, T.T, Benoit, E, Servent, D, Taylor, P, Molgo, J, Marchot, P.
登録日2009-12-04
公開日2010-03-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Determinants in Phycotoxins and Achbp Conferring High Affinity Binding and Nicotinic Achr Antagonism.
Proc.Natl.Acad.Sci.USA, 107, 2010
2WZY
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Crystal structure of A-AChBP in complex with 13-desmethyl spirolide C
分子名称: 13-DESMETHYL SPIROLIDE C, SOLUBLE ACETYLCHOLINE RECEPTOR
著者Bourne, Y, Radic, Z, Araoz, R, Talley, T.T, Benoit, E, Servent, D, Taylor, P, Molgo, J, Marchot, P.
登録日2009-12-03
公開日2010-03-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Structural Determinants in Phycotoxins and Achbp Conferring High Affinity Binding and Nicotinic Achr Antagonism.
Proc.Natl.Acad.Sci.USA, 107, 2010
1G1P
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NMR Solution Structures of delta-Conotoxin EVIA from Conus ermineus that Selectively Acts on Vertebrate Neuronal Na+ Channels
分子名称: CONOTOXIN EVIA
著者Volpon, L, Lamthanh, H, Barbier, J, Gilles, N, Molgo, J, Menez, A, Lancelin, J.M.
登録日2000-10-13
公開日2000-11-01
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR Solution Structures of delta-Conotoxin EVIA from Conus ermineus That Selectively Acts on Vertebrate Neuronal Na+ Channels.
J.Biol.Chem., 279, 2004
8QTL
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Aplysia californica acetylcholine-binding protein in complex with Spiroimine (-)-4 S
分子名称: CHLORIDE ION, ISOPROPYL ALCOHOL, Soluble acetylcholine receptor, ...
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-10-12
公開日2024-04-03
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism
Mar Drugs, 22, 2024
4XK9
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Crystal structure of A-AChBP in complex with pinnatoxin G
分子名称: CHLORIDE ION, Pinnatoxin G, Soluble acetylcholine receptor
著者Bourne, Y, Sulzenbacher, G, Marchot, P.
登録日2015-01-10
公開日2015-06-03
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
4XHE
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Crystal Structure of A-AChBP in complex with pinnatoxin A
分子名称: CALCIUM ION, CHLORIDE ION, Pinnatoxin A, ...
著者Bourne, Y, Sulzenbacher, G, Marchot, P.
登録日2015-01-05
公開日2015-06-03
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Marine Macrocyclic Imines, Pinnatoxins A and G: Structural Determinants and Functional Properties to Distinguish Neuronal alpha 7 from Muscle alpha 12 beta gamma delta nAChRs.
Structure, 23, 2015
8Q1M
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Aplysia californica acetylcholine-binding protein in complex with Spiroimine (+)-4 R
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Soluble acetylcholine receptor, ...
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-07-31
公開日2024-04-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism
Mar Drugs, 22, 2024
8QX2
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Aplysia californica acetylcholine-binding protein in complex with with racemic spiroimine (+)/(-)-4
分子名称: ISOPROPYL ALCOHOL, Soluble acetylcholine receptor, Spiroimine (+)-4 R
著者Sulzenbacher, G, Bourne, Y, Marchot, P.
登録日2023-10-20
公開日2024-04-03
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Cyclic Imine Core Common to the Marine Macrocyclic Toxins Is Sufficient to Dictate Nicotinic Acetylcholine Receptor Antagonism
Mar Drugs, 22, 2024
1G1Z
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NMR Solution Structures of delta-Conotoxin EVIA from Conus ermineus that Selectively Acts on Vertebrate Neuronal Na+ Channels, LEU12-PRO13 Cis isomer
分子名称: CONOTOXIN EVIA
著者Volpon, L, Lamthanh, H, Le Gall, F, Menez, A, Lancelin, J.M.
登録日2000-10-16
公開日2000-11-01
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献NMR Solution Structures of delta-Conotoxin EVIA from Conus ermineus That Selectively Acts on Vertebrate Neuronal Na+ Channels.
J.Biol.Chem., 279, 2004

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件を2024-04-24に公開中

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