7GU5
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![BU of 7gu5 by Molmil](/molmil-images/mine/7gu5) | |
7GU4
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![BU of 7gu4 by Molmil](/molmil-images/mine/7gu4) | |
7GU7
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![BU of 7gu7 by Molmil](/molmil-images/mine/7gu7) | |
7GU9
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![BU of 7gu9 by Molmil](/molmil-images/mine/7gu9) | |
7GTX
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![BU of 7gtx by Molmil](/molmil-images/mine/7gtx) | |
7GTW
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![BU of 7gtw by Molmil](/molmil-images/mine/7gtw) | |
7GU0
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![BU of 7gu0 by Molmil](/molmil-images/mine/7gu0) | |
7GTZ
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![BU of 7gtz by Molmil](/molmil-images/mine/7gtz) | |
7GU6
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![BU of 7gu6 by Molmil](/molmil-images/mine/7gu6) | |
7GU1
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![BU of 7gu1 by Molmil](/molmil-images/mine/7gu1) | |
7GTY
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![BU of 7gty by Molmil](/molmil-images/mine/7gty) | |
7GUB
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![BU of 7gub by Molmil](/molmil-images/mine/7gub) | |
7GU8
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![BU of 7gu8 by Molmil](/molmil-images/mine/7gu8) | |
7GUA
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![BU of 7gua by Molmil](/molmil-images/mine/7gua) | |
7GUC
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![BU of 7guc by Molmil](/molmil-images/mine/7guc) | |
7GU2
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![BU of 7gu2 by Molmil](/molmil-images/mine/7gu2) | |
7GU3
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![BU of 7gu3 by Molmil](/molmil-images/mine/7gu3) | |
7FQT
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![BU of 7fqt by Molmil](/molmil-images/mine/7fqt) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with FMOMB000293a | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3,4,6,7-tetrahydroacridine-1,8(2H,5H)-dione, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-19 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.54 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRP
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![BU of 7frp by Molmil](/molmil-images/mine/7frp) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with XST00000245b | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 5-(2-methyl-1,3-thiazol-4-yl)thiophene-2-carboxylic acid, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-24 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.77 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FQM
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![BU of 7fqm by Molmil](/molmil-images/mine/7fqm) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with FMOPL000619a | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-({[(thiophen-2-yl)methyl]amino}methyl)phenol, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-19 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.94 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FQV
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![BU of 7fqv by Molmil](/molmil-images/mine/7fqv) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with XST00000847b | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, N,N-dimethylpyridin-4-amine, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-19 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.04 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRE
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![BU of 7fre by Molmil](/molmil-images/mine/7fre) | PanDDA analysis group deposition -- Crystal structure of PTP1B after initial refinement with no ligand modeled | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-20 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRT
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![BU of 7frt by Molmil](/molmil-images/mine/7frt) | PanDDA analysis group deposition of ground-state model of PTP1B, using pre-clustering, cluster 1 | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-26 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FRU
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![BU of 7fru by Molmil](/molmil-images/mine/7fru) | PanDDA analysis group deposition of ground-state model of PTP1B, using pre-clustering, cluster 2 | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-26 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.98 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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7FQU
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![BU of 7fqu by Molmil](/molmil-images/mine/7fqu) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with FMSOA000470b | Descriptor: | (3-chlorophenoxy)acetic acid, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | Authors: | Mehlman, T, Biel, J, Azeem, S.M, Nelson, E.R, Hossain, S, Dunnett, L.E, Paterson, N.G, Douangamath, A, Talon, R, Axford, D, Orins, H, von Delft, F, Keedy, D.A. | Deposit date: | 2022-10-19 | Release date: | 2022-11-23 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | Room-temperature crystallography reveals altered binding of small-molecule fragments to PTP1B. Elife, 12, 2023
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