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1NVV
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BU of 1nvv by Molmil
Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
分子名称: MAGNESIUM ION, PHOSPHATE ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ...
著者Margarit, S.M, Sondermann, H, Hall, B.E, Nagar, B, Hoelz, A, Pirruccello, M, Bar-Sagi, D, Kuriyan, J.
登録日2003-02-04
公開日2003-04-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
Cell(Cambridge,Mass.), 112, 2003
1NVX
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BU of 1nvx by Molmil
Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Margarit, S.M, Sondermann, H, Hall, B.E, Nagar, B, Hoelz, A, Pirruccello, M, Bar-Sagi, D, Kuriyan, J.
登録日2003-02-04
公開日2003-04-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
Cell(Cambridge,Mass.), 112, 2003
1NVW
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BU of 1nvw by Molmil
Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
分子名称: MAGNESIUM ION, PHOSPHATE ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ...
著者Margarit, S.M, Sondermann, H, Hall, B.E, Nagar, B, Hoelz, A, Pirruccello, M, Bar-Sagi, D, Kuriyan, J.
登録日2003-02-04
公開日2003-04-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
Cell(Cambridge,Mass.), 112, 2003
1NVU
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BU of 1nvu by Molmil
Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Margarit, S.M, Sondermann, H, Hall, B.E, Nagar, B, Hoelz, A, Pirruccello, M, Bar-Sagi, D, Kuriyan, J.
登録日2003-02-04
公開日2003-04-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural evidence for feedback activation by RasGTP of the Ras-specific nucleotide exchange factor SOS
Cell(Cambridge,Mass.), 112, 2003
2GWK
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BU of 2gwk by Molmil
SpvB ADP-ribosylated actin: orthorhombic crystal form
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Actin, alpha skeletal muscle, ...
著者Stebbins, C.E, Margarit, S.M.
登録日2006-05-04
公開日2006-08-29
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A steric antagonism of actin polymerization by a salmonella virulence protein.
Structure, 14, 2006
2GWJ
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BU of 2gwj by Molmil
SpvB ADP-ribosylated actin: hexagonal crystal form
分子名称: ADENOSINE-5'-TRIPHOSPHATE, Actin, alpha skeletal muscle, ...
著者Stebbins, C.E, Margarit, S.M.
登録日2006-05-04
公開日2006-08-29
最終更新日2017-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A steric antagonism of actin polymerization by a salmonella virulence protein.
Structure, 14, 2006
2GWL
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BU of 2gwl by Molmil
Crystal structure of the Salmonella SpvB ATR Domain in complex with NADH
分子名称: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 65 kDa virulence protein
著者Stebbins, C.E, Margarit, S.M.
登録日2006-05-04
公開日2006-08-29
最終更新日2017-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A steric antagonism of actin polymerization by a salmonella virulence protein.
Structure, 14, 2006
2GWM
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BU of 2gwm by Molmil
Crystal structure of the Salmonella SpvB ATR Domain
分子名称: 65 kDa virulence protein, SULFATE ION
著者Stebbins, C.E, Margarit, S.M.
登録日2006-05-04
公開日2006-08-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献A steric antagonism of actin polymerization by a salmonella virulence protein.
Structure, 14, 2006
1BKD
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BU of 1bkd by Molmil
COMPLEX OF HUMAN H-RAS WITH HUMAN SOS-1
分子名称: H-RAS, SON OF SEVENLESS-1
著者Boriack-Sjodin, P.A, Margarit, S.M, Sagi, D.B, Kuriyan, J.
登録日1998-07-06
公開日1999-01-13
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The structural basis of the activation of Ras by Sos.
Nature, 394, 1998
3I7I
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BU of 3i7i by Molmil
MMP-13 in complex with a non zinc-chelating inhibitor
分子名称: CALCIUM ION, Collagenase 3, N-[4-(5-{[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]carbamoyl}furan-2-yl)phenyl]-1-benzofuran-2-carboxamide, ...
著者Farrow, N.A, Margarit, S.M.
登録日2009-07-08
公開日2009-09-01
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.208 Å)
主引用文献Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors.
Bioorg.Med.Chem.Lett., 19, 2009
5BPA
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BU of 5bpa by Molmil
X-RAY Co-structure of MMP-13 with 4-[({5-[2-(ethoxycarbonyl)-1H-indol-5-yl]-1-methyl-1H-pyrazol-3-yl}formamido)methyl]benzoate
分子名称: 4-{[({5-[2-(ethoxycarbonyl)-1H-indol-5-yl]-1-methyl-1H-pyrazol-3-yl}carbonyl)amino]methyl}benzoic acid, CALCIUM ION, Collagenase 3, ...
著者Farrow, N.A, Margarit, S.M.
登録日2015-05-27
公開日2015-06-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Fragment-based discovery of indole inhibitors of matrix metalloproteinase-13.
J. Med. Chem., 54, 2011

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件を2024-04-24に公開中

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