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3KI3
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BU of 3ki3 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-H
Descriptor: 2-[(dimethylamino)methyl]-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.27 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI6
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BU of 3ki6 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-L
Descriptor: 8-fluoro-2-(3-piperidin-1-ylpropanoyl)-1,3,4,5-tetrahydrobenzo[c][1,6]naphthyridin-6(2H)-one, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.54 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI5
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BU of 3ki5 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-M
Descriptor: Cholix toxin, N-(6-oxo-5,6-dihydrobenzo[c][1,5]naphthyridin-2-yl)-2-(4-pyrrolidin-1-ylpiperidin-1-yl)acetamide
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI1
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BU of 3ki1 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-F
Descriptor: 2-{4-[3-(dimethylamino)propoxy]phenyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.43 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI0
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BU of 3ki0 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-D
Descriptor: 3-(morpholin-4-ylmethyl)-1,5-dihydro-6H-[1,2]diazepino[4,5,6-cd]indol-6-one, CHLORIDE ION, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.29 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI7
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BU of 3ki7 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-I
Descriptor: 2-{2-[4-(pyrrolidin-1-ylmethyl)phenyl]ethyl}-5,6-dihydroimidazo[4,5,1-jk][1,4]benzodiazepin-7(4H)-one, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.32 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI2
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BU of 3ki2 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-G
Descriptor: 2-(4-methylpiperazin-1-yl)benzo[c][1,5]naphthyridin-6(5H)-one, Cholix toxin
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.28 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3KI4
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BU of 3ki4 by Molmil
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-P
Descriptor: (11bR)-3-oxo-1,2,3,11b-tetrahydrochromeno[4,3,2-de]isoquinoline-10-sulfonic acid, Cholix toxin, GLYCEROL
Authors:Jorgensen, R, Edwards, P.R, Merrill, A.R.
Deposit date:2009-10-31
Release date:2010-10-27
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae
To be Published
3NY6
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BU of 3ny6 by Molmil
Catalytic fragment of cholix toxin from vibrio cholerae in complex with inhibitor V30
Descriptor: 2-[(5,6-dimethyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2-hydroxyethyl)acetamide, Cholix toxin, GLYCEROL, ...
Authors:Merrill, A.R, Jorgensen, R.
Deposit date:2010-07-14
Release date:2010-12-29
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (1.68 Å)
Cite:Newly discovered and characterized antivirulence compounds inhibit bacterial mono-ADP-ribosyltransferase toxins.
Antimicrob.Agents Chemother., 55, 2011

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