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6HTF
Crystal structure of human Btk SH2 domain bound to rF10 repebody
Descriptor:
Tyrosine-protein kinase BTK, rF10 repebody
Authors:
Duarte, D.P
,
Pojer, F
,
Hantschel, O.
Deposit date:
2018-10-04
Release date:
2020-05-20
Last modified:
2024-01-24
Method:
X-RAY DIFFRACTION (2.102 Å)
Cite:
Btk SH2-kinase interface is critical for allosteric kinase activation and its targeting inhibits B-cell neoplasms.
Nat Commun, 11, 2020
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PDB entries from 2024-06-12