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Human Nuclear Receptor-Ligand Complex 1
Descriptor:	Peroxisome proliferator activated receptor delta, VACCENIC ACID, heptyl beta-D-glucopyranoside
Authors:	Fyffe, S.A, Alphey, M.S, Buetow, L, Smith, T.K, Ferguson, M.A.J, Sorensen, M.D, Bjorkling, F, Hunter, W.N.
Deposit date:	2005-10-15
Release date:	2006-01-24
Last modified:	2024-03-13
Method:	X-RAY DIFFRACTION (2.3 Å)
Cite:	Reevaluation of the PPAR-beta/delta Ligand Binding Domain Model Reveals Why It Exhibits the Activated Form Mol.Cell, 21, 2006

Crystal structure of the complex between PPARgamma and the partial agonist LT127 (ureidofibrate derivative). This structure has been obtained from crystals soaked for 6 hours.
Descriptor:	(2S)-2-(4-{2-[1,3-BENZOXAZOL-2-YL(HEPTYL)AMINO]ETHYL}PHENOXY)-2-METHYLBUTANOIC ACID, Peroxisome proliferator-activated receptor gamma
Authors:	Pochetti, G, Mazza, F.
Deposit date:	2006-08-23
Release date:	2007-04-17
Last modified:	2023-08-30
Method:	X-RAY DIFFRACTION (2.25 Å)
Cite:	Insights into the mechanism of partial agonism: crystal structures of the peroxisome proliferator-activated receptor gamma ligand-binding domain in the complex with two enantiomeric ligands J.Biol.Chem., 282, 2007

Crystal structure of the complex between PPARgamma and the partial agonist LT127 (ureidofibrate derivative). Structure obtained from crystals of the apo-form soaked for 30 days.
Descriptor:	(2S)-2-(4-{2-[1,3-BENZOXAZOL-2-YL(HEPTYL)AMINO]ETHYL}PHENOXY)-2-METHYLBUTANOIC ACID, Peroxisome proliferator-activated receptor gamma
Authors:	Pochetti, G, Mazza, F.
Deposit date:	2006-08-22
Release date:	2007-04-17
Last modified:	2024-02-21
Method:	X-RAY DIFFRACTION (2.1 Å)
Cite:	Insights into the mechanism of partial agonism: crystal structures of the peroxisome proliferator-activated receptor gamma ligand-binding domain in the complex with two enantiomeric ligands. J.Biol.Chem., 282, 2007

Crystal structure of the complex between PPARgamma and the agonist LT160 (ureidofibrate derivative)
Descriptor:	(2R)-2-(4-{2-[1,3-BENZOXAZOL-2-YL(HEPTYL)AMINO]ETHYL}PHENOXY)-2-METHYLBUTANOIC ACID, Peroxisome proliferator-activated receptor gamma
Authors:	Pochetti, G, Mazza, F.
Deposit date:	2006-08-22
Release date:	2007-04-17
Last modified:	2024-02-21
Method:	X-RAY DIFFRACTION (2.1 Å)
Cite:	Insights into the mechanism of partial agonism: crystal structures of the peroxisome proliferator-activated receptor gamma ligand-binding domain in the complex with two enantiomeric ligands J.Biol.Chem., 282, 2007