6OP0
| Asymmetric hTNF-alpha | Descriptor: | (R)-{1-[(2,5-dimethylphenyl)methyl]-6-(1-methyl-1H-pyrazol-4-yl)-1H-benzimidazol-2-yl}(pyridin-4-yl)methanol, Tumor necrosis factor | Authors: | Arakaki, T.L, Edwards, T.E, Fairman, J.W, Davies, D.R, Foley, A, Ceska, T. | Deposit date: | 2019-04-23 | Release date: | 2019-12-25 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.55 Å) | Cite: | Small molecules that inhibit TNF signalling by stabilising an asymmetric form of the trimer. Nat Commun, 10, 2019
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3QK8
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3QIV
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3Q8N
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3QHA
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3QUA
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3QUV
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3QRE
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3RV2
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3R2N
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3RFQ
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3R9T
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3RRV
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3R1I
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3R9R
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3R1J
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3R6H
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3RD5
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3RIH
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3QYR
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3R4T
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3R9P
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3TDE
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3R9S
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3R0O
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