5IFU
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![BU of 5ifu by Molmil](/molmil-images/mine/5ifu) | Crystal Structure of Prolyl-tRNA synthetase (ProRS, Proline--tRNA ligase) from Plasmodium falciparum in complex with Glyburide | Descriptor: | 1,2-ETHANEDIOL, 5-chloro-N-(2-{4-[(cyclohexylcarbamoyl)sulfamoyl]phenyl}ethyl)-2-methoxybenzamide, CHLORIDE ION, ... | Authors: | Dranow, D.M, Hewitt, S.N, Abendroth, J, Structural Genomics Consortium (SGC) | Deposit date: | 2016-02-26 | Release date: | 2016-11-16 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.45 Å) | Cite: | Biochemical and Structural Characterization of Selective Allosteric Inhibitors of the Plasmodium falciparum Drug Target, Prolyl-tRNA-synthetase. ACS Infect Dis, 3, 2017
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5IRD
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6BFA
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![BU of 6bfa by Molmil](/molmil-images/mine/6bfa) | Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with inhibitor UW1553 | Descriptor: | 1-{4-amino-3-[6-(cyclopropyloxy)naphthalen-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-1-yl}-2-methylpropan-2-ol, Calmodulin-domain protein kinase 1 | Authors: | Merritt, E.A. | Deposit date: | 2017-10-26 | Release date: | 2017-12-06 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Development of an Orally Available and Central Nervous System (CNS) Penetrant Toxoplasma gondii Calcium-Dependent Protein Kinase 1 (TgCDPK1) Inhibitor with Minimal Human Ether-a-go-go-Related Gene (hERG) Activity for the Treatment of Toxoplasmosis. J. Med. Chem., 59, 2016
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5K0T
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5K0S
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4JBV
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![BU of 4jbv by Molmil](/molmil-images/mine/4jbv) | |
4M84
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![BU of 4m84 by Molmil](/molmil-images/mine/4m84) | |
4WI1
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![BU of 4wi1 by Molmil](/molmil-images/mine/4wi1) | |
8TZM
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8SOY
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![BU of 8soy by Molmil](/molmil-images/mine/8soy) | |
5UJ5
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![BU of 5uj5 by Molmil](/molmil-images/mine/5uj5) | |
5VMT
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![BU of 5vmt by Molmil](/molmil-images/mine/5vmt) | |
3TL3
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3TMQ
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3TX2
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3TRR
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![BU of 3trr by Molmil](/molmil-images/mine/3trr) | |
3U7J
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![BU of 3u7j by Molmil](/molmil-images/mine/3u7j) | |
3TZQ
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![BU of 3tzq by Molmil](/molmil-images/mine/3tzq) | |
3UE9
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![BU of 3ue9 by Molmil](/molmil-images/mine/3ue9) | |
3UK1
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![BU of 3uk1 by Molmil](/molmil-images/mine/3uk1) | |
3BJE
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![BU of 3bje by Molmil](/molmil-images/mine/3bje) | |
6VYE
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![BU of 6vye by Molmil](/molmil-images/mine/6vye) | |
6UHW
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![BU of 6uhw by Molmil](/molmil-images/mine/6uhw) | |
4EWG
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![BU of 4ewg by Molmil](/molmil-images/mine/4ewg) | |
4F32
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![BU of 4f32 by Molmil](/molmil-images/mine/4f32) | Crystal structure of 3-oxoacyl-[acyl-carrier-protein] synthase II from Burkholderia vietnamiensis in complex with platencin | Descriptor: | 1,2-ETHANEDIOL, 2,4-dihydroxy-3-({3-[(2S,4aS,8S,8aR)-8-methyl-3-methylidene-7-oxo-1,3,4,7,8,8a-hexahydro-2H-2,4a-ethanonaphthalen-8-yl]propanoyl}amino)benzoic acid, 3-oxoacyl-[acyl-carrier-protein] synthase 2, ... | Authors: | Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2012-05-08 | Release date: | 2012-05-23 | Last modified: | 2014-02-12 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Combining functional and structural genomics to sample the essential Burkholderia structome. Plos One, 8, 2013
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