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8IVD
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BU of 8ivd by Molmil
COMPLEX STRUCTURE OF CD93-IGFBP7
Descriptor: Insulin-like growth factor-binding protein 7,Complement component C1q receptor
Authors:Xu, Y.M, Song, G.J.
Deposit date:2023-03-27
Release date:2024-01-17
Method:X-RAY DIFFRACTION (3.24 Å)
Cite:structural insight into CD93 recognition by IGFBP7
To Be Published
7S3P
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BU of 7s3p by Molmil
BD2 domain of human BRD3 bound to Physachenolide C
Descriptor: Bromodomain-containing protein 3, CHLORIDE ION, Physachenolide C
Authors:Horton, N.C, Chapman, E, Sivinski, J, Zerio, C, Ghadirian, N.
Deposit date:2021-09-07
Release date:2023-01-11
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.89 Å)
Cite:Physachenolide C is a Potent, Selective BET Inhibitor.
J.Med.Chem., 66, 2023
7R8R
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BU of 7r8r by Molmil
Physachenolide C with Bromodomain (BRD3-BD1)
Descriptor: Bromodomain-containing protein 3, Physachenolide C
Authors:Fromme, R, Sivinski, J, Zerio, C, Gunatilaka, A.A.L, Chapman, E.
Deposit date:2021-06-27
Release date:2022-09-21
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Physachenolide C is a Potent, Selective BET Inhibitor.
J.Med.Chem., 66, 2023
6LTK
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BU of 6ltk by Molmil
HSP90 in complex with SNX-2112
Descriptor: 4-[6,6-dimethyl-4-oxidanylidene-3-(trifluoromethyl)-5,7-dihydroindazol-1-yl]-2-[(4-oxidanylcyclohexyl)amino]benzamide, Heat shock protein HSP 90-alpha
Authors:Cao, H.L.
Deposit date:2020-01-22
Release date:2021-01-27
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.141 Å)
Cite:Complex Crystal Structure Determination and in vitro Anti-non-small Cell Lung Cancer Activity of Hsp90 N Inhibitor SNX-2112.
Front Cell Dev Biol, 9, 2021

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數據於2024-07-24公開中

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