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Crystal structure of Maternal Embryonic Leucine Zipper Kinase (MELK) in complex with dorsomorphin (Compound C)
Descriptor:	1,2-ETHANEDIOL, 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine, Maternal embryonic leucine zipper kinase
Authors:	Golik, P, Rembacz, K.P, Zrubek, K, Romanowska, M, Bugusz, J, Wladyka, B, Dubin, G.
Deposit date:	2018-06-21
Release date:	2019-05-29
Last modified:	2024-01-17
Method:	X-RAY DIFFRACTION (2.24 Å)
Cite:	Crystal structure of Maternal Embryonic Leucine Zipper Kinase (MELK) in complex with dorsomorphin (Compound C). Arch.Biochem.Biophys., 671, 2019

Crystal structure of PIM1 kinase in complex with small-molecule inhibitor
Descriptor:	(5E)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-one, IMIDAZOLE, Serine/threonine-protein kinase pim-1
Authors:	Dubin, G, Bogusz, J.
Deposit date:	2017-05-17
Release date:	2017-11-01
Last modified:	2024-10-16
Method:	X-RAY DIFFRACTION (2.4 Å)
Cite:	Structural analysis of PIM1 kinase complexes with ATP-competitive inhibitors. Sci Rep, 7, 2017

Crystal structure of PIM1 kinase in complex with small-molecule inhibitor
Descriptor:	5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid, CHLORIDE ION, GLYCEROL, ...
Authors:	Bogusz, J, Dubin, G.
Deposit date:	2017-05-17
Release date:	2017-11-01
Last modified:	2024-01-17
Method:	X-RAY DIFFRACTION (2.4 Å)
Cite:	Structural analysis of PIM1 kinase complexes with ATP-competitive inhibitors. Sci Rep, 7, 2017

Crystal structure of PIM1 kinase in complex with small-molecule inhibitor
Descriptor:	(3~{E})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{H}-indol-2-one, CHLORIDE ION, IMIDAZOLE, ...
Authors:	Dubin, G, Bogusz, J.
Deposit date:	2017-05-17
Release date:	2017-11-01
Last modified:	2024-01-17
Method:	X-RAY DIFFRACTION (2.44 Å)
Cite:	Structural analysis of PIM1 kinase complexes with ATP-competitive inhibitors. Sci Rep, 7, 2017