5H8U
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![BU of 5h8u by Molmil](/molmil-images/mine/5h8u) | Crystal structure of mycobacterium tuberculosis wild-type malate synthase in complex with product malate | Descriptor: | (2S)-2-hydroxybutanedioic acid, GLYOXYLIC ACID, MAGNESIUM ION, ... | Authors: | Krieger, I.V, Huang, H.-L, Sacchettini, J.C. | Deposit date: | 2015-12-23 | Release date: | 2016-10-26 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.85 Å) | Cite: | Mycobacterium tuberculosis Malate Synthase Structures with Fragments Reveal a Portal for Substrate/Product Exchange. J. Biol. Chem., 291, 2016
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3SAD
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![BU of 3sad by Molmil](/molmil-images/mine/3sad) | Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 4-(2-mehtylphenyl)-2,4-dioxobutanoic acid inhibitor | Descriptor: | 4-(2-methylphenyl)-2,4-dioxobutanoic acid, MAGNESIUM ION, Malate synthase G | Authors: | Krieger, I.V, Sun, Q, Sacchettini, J.C, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB) | Deposit date: | 2011-06-02 | Release date: | 2012-11-07 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.82 Å) | Cite: | Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase. Chem.Biol., 19, 2012
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3SB0
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![BU of 3sb0 by Molmil](/molmil-images/mine/3sb0) | Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 4-(2-chloro-6-fluoro-3-methylphenyl)-2,4-dioxobutanoic acid inhibitor | Descriptor: | 4-(2-chloro-6-fluoro-3-methylphenyl)-2,4-dioxobutanoic acid, MAGNESIUM ION, Malate synthase G | Authors: | Krieger, I.V, Sun, Q, Sacchettini, J.C, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB) | Deposit date: | 2011-06-03 | Release date: | 2012-11-07 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.199 Å) | Cite: | Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase. Chem.Biol., 19, 2012
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5H8P
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![BU of 5h8p by Molmil](/molmil-images/mine/5h8p) | |
3SAZ
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![BU of 3saz by Molmil](/molmil-images/mine/3saz) | Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 4-(3-bromophenyl)-2,4-dioxobutanoic acid inhibitor | Descriptor: | 4-(3-bromophenyl)-2,4-dioxobutanoic acid, MAGNESIUM ION, Malate synthase G | Authors: | Krieger, I.V, Sun, Q, Sacchettini, J.C, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB) | Deposit date: | 2011-06-03 | Release date: | 2012-11-07 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (2.04 Å) | Cite: | Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase. Chem.Biol., 19, 2012
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3S9I
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![BU of 3s9i by Molmil](/molmil-images/mine/3s9i) | Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 2-4-dioxo-4-phenylbutanoic acid inhibitor | Descriptor: | 2-4-DIOXO-4-PHENYLBUTANOIC ACID, MAGNESIUM ION, Malate synthase G | Authors: | Krieger, I.V, Sun, Q, Sacchettini, J.C, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB) | Deposit date: | 2011-06-01 | Release date: | 2012-11-07 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase. Chem.Biol., 19, 2012
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3S9Z
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![BU of 3s9z by Molmil](/molmil-images/mine/3s9z) | Crystal structure of Mycobacterium tuberculosis malate synthase in complex with 4-(2-bromophenyl)-2,4-dioxobutanoic acid inhibitor | Descriptor: | 4-(2-bromophenyl)-2,4-dioxobutanoic acid, MAGNESIUM ION, Malate synthase G | Authors: | Krieger, I.V, Sun, Q, Sacchettini, J.C, Mycobacterium Tuberculosis Structural Proteomics Project (XMTB) | Deposit date: | 2011-06-02 | Release date: | 2012-11-07 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.793 Å) | Cite: | Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase. Chem.Biol., 19, 2012
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6APZ
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![BU of 6apz by Molmil](/molmil-images/mine/6apz) | |
6ASU
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![BU of 6asu by Molmil](/molmil-images/mine/6asu) | |
5CAH
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![BU of 5cah by Molmil](/molmil-images/mine/5cah) | |
6AS6
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![BU of 6as6 by Molmil](/molmil-images/mine/6as6) | |
5CC5
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![BU of 5cc5 by Molmil](/molmil-images/mine/5cc5) | |
5C7V
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![BU of 5c7v by Molmil](/molmil-images/mine/5c7v) | |
6BA7
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![BU of 6ba7 by Molmil](/molmil-images/mine/6ba7) | |
5C9X
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![BU of 5c9x by Molmil](/molmil-images/mine/5c9x) | |
6AXB
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![BU of 6axb by Molmil](/molmil-images/mine/6axb) | |
5CBI
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![BU of 5cbi by Molmil](/molmil-images/mine/5cbi) | |
5CC6
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![BU of 5cc6 by Molmil](/molmil-images/mine/5cc6) | |
5CJM
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![BU of 5cjm by Molmil](/molmil-images/mine/5cjm) | |
5CC3
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![BU of 5cc3 by Molmil](/molmil-images/mine/5cc3) | |
6C2X
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![BU of 6c2x by Molmil](/molmil-images/mine/6c2x) | |
6C6O
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![BU of 6c6o by Molmil](/molmil-images/mine/6c6o) | |
6C7B
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![BU of 6c7b by Molmil](/molmil-images/mine/6c7b) | |
6C8P
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![BU of 6c8p by Molmil](/molmil-images/mine/6c8p) | |
5C9W
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![BU of 5c9w by Molmil](/molmil-images/mine/5c9w) | |