5UMH
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![BU of 5umh by Molmil](/molmil-images/mine/5umh) | |
5V0W
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4WEC
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![BU of 4wec by Molmil](/molmil-images/mine/4wec) | |
6CFP
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![BU of 6cfp by Molmil](/molmil-images/mine/6cfp) | |
6CXM
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![BU of 6cxm by Molmil](/molmil-images/mine/6cxm) | |
5DD7
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5K9F
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5K9Z
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6Q09
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6PTR
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![BU of 6ptr by Molmil](/molmil-images/mine/6ptr) | |
6O49
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6O4A
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6HVF
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![BU of 6hvf by Molmil](/molmil-images/mine/6hvf) | Kinase domain of cSrc in complex with compound 29B | Descriptor: | 1,2-ETHANEDIOL, Proto-oncogene tyrosine-protein kinase Src, ~{N}-[3-[3-ethyl-6-[4-(4-methylpiperazin-1-yl)phenyl]-4-oxidanylidene-7~{H}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]prop-2-enamide | Authors: | Keul, M, Mueller, M.P, Rauh, D. | Deposit date: | 2018-10-10 | Release date: | 2019-10-23 | Last modified: | 2020-01-01 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S. Chem Sci, 10, 2019
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6HVE
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![BU of 6hve by Molmil](/molmil-images/mine/6hve) | Kinase domain of cSrc in complex with compound 9 | Descriptor: | Proto-oncogene tyrosine-protein kinase Src, ~{N}-[3-(4-methoxy-7~{H}-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]prop-2-enamide | Authors: | Keul, M, Mueller, M.P, Rauh, D. | Deposit date: | 2018-10-10 | Release date: | 2019-10-23 | Last modified: | 2020-01-01 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S. Chem Sci, 10, 2019
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3EK2
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3EJ2
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6WCI
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![BU of 6wci by Molmil](/molmil-images/mine/6wci) | |
3EZO
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![BU of 3ezo by Molmil](/molmil-images/mine/3ezo) | |
7SWH
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7SWK
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![BU of 7swk by Molmil](/molmil-images/mine/7swk) | |
7T24
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7T29
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7SZV
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7STZ
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7T93
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![BU of 7t93 by Molmil](/molmil-images/mine/7t93) | |