1YGC
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![BU of 1ygc by Molmil](/molmil-images/mine/1ygc) | Short Factor VIIa with a small molecule inhibitor | Descriptor: | (R)-4-[2-(3-AMINO-BENZENESULFONYLAMINO)-1-(3,5-DIETHOXY-2-FLUOROPHENYL)-2-OXO-ETHYLAMINO]-2-HYDROXY-BENZAMIDINE, CALCIUM ION, Coagulation factor VII, ... | Authors: | Olivero, A.G, Eigenbrot, C, Goldsmith, R, Robarge, K, Artis, D.R, Flygare, J, Rawson, T, Refino, C, Bunting, S, Kirchhofer, D. | Deposit date: | 2005-01-04 | Release date: | 2005-01-18 | Last modified: | 2011-07-13 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | A selective, slow binding inhibitor of factor VIIa binds to a nonstandard active site conformation and attenuates thrombus formation in vivo. J.Biol.Chem., 280, 2005
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4HGE
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![BU of 4hge by Molmil](/molmil-images/mine/4hge) | JAK2 kinase (JH1 domain) in complex with compound 8 | Descriptor: | N-[1-(3-chlorophenyl)-3-methyl-1H-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide, Tyrosine-protein kinase JAK2 | Authors: | Eigenbrot, C, Ultsch, M. | Deposit date: | 2012-10-08 | Release date: | 2012-10-24 | Last modified: | 2023-12-06 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Discovery of potent and selective pyrazolopyrimidine janus kinase 2 inhibitors. J.Med.Chem., 55, 2012
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1NOM
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![BU of 1nom by Molmil](/molmil-images/mine/1nom) | |
8ICM
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![BU of 8icm by Molmil](/molmil-images/mine/8icm) | DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DATP (1 MILLIMOLAR), MNCL2 (5 MILLIMOLAR), AND AMMONIUM SULFATE (75 MILLIMOLAR) | Descriptor: | DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*G)-3'), PROTEIN (DNA POLYMERASE BETA (E.C.2.7.7.7)), ... | Authors: | Pelletier, H, Sawaya, M.R. | Deposit date: | 1996-01-04 | Release date: | 1996-11-15 | Last modified: | 2023-08-02 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta. Biochemistry, 35, 1996
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8ICJ
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![BU of 8icj by Molmil](/molmil-images/mine/8icj) | |
8ICH
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![BU of 8ich by Molmil](/molmil-images/mine/8ich) | |
8ICV
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![BU of 8icv by Molmil](/molmil-images/mine/8icv) | |
8ICU
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![BU of 8icu by Molmil](/molmil-images/mine/8icu) | |
8ICY
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![BU of 8icy by Molmil](/molmil-images/mine/8icy) | |
8ICX
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![BU of 8icx by Molmil](/molmil-images/mine/8icx) | |
8ICE
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![BU of 8ice by Molmil](/molmil-images/mine/8ice) | |
8ICR
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![BU of 8icr by Molmil](/molmil-images/mine/8icr) | |
8ICI
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![BU of 8ici by Molmil](/molmil-images/mine/8ici) | |
8ICF
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![BU of 8icf by Molmil](/molmil-images/mine/8icf) | |
8ICW
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![BU of 8icw by Molmil](/molmil-images/mine/8icw) | |
8ICS
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![BU of 8ics by Molmil](/molmil-images/mine/8ics) | |
8ICQ
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![BU of 8icq by Molmil](/molmil-images/mine/8icq) | |
8ICB
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![BU of 8icb by Molmil](/molmil-images/mine/8icb) | |
8ICA
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![BU of 8ica by Molmil](/molmil-images/mine/8ica) | |
8ICP
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![BU of 8icp by Molmil](/molmil-images/mine/8icp) | |
8ICN
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![BU of 8icn by Molmil](/molmil-images/mine/8icn) | |
8ICK
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![BU of 8ick by Molmil](/molmil-images/mine/8ick) | DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DATP (1 MILLIMOLAR), MGCL2 (5 MILLIMOLAR), AND MNCL2 (5 MILLIMOLAR) | Descriptor: | 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*GP*A)-3'), ... | Authors: | Pelletier, H, Sawaya, M.R. | Deposit date: | 1996-04-19 | Release date: | 1996-11-15 | Last modified: | 2023-08-02 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta. Biochemistry, 35, 1996
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8ICL
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![BU of 8icl by Molmil](/molmil-images/mine/8icl) | |
8ICZ
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![BU of 8icz by Molmil](/molmil-images/mine/8icz) | DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF OF DATP (1 MILLIMOLAR), MNCL2 (5 MILLIMOLAR), AND LITHIUM SULFATE (75 MILLIMOLAR) | Descriptor: | DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*G)-3'), PROTEIN (DNA POLYMERASE BETA (E.C.2.7.7.7)), ... | Authors: | Pelletier, H, Sawaya, M.R. | Deposit date: | 1996-01-04 | Release date: | 1996-11-15 | Last modified: | 2023-08-02 | Method: | X-RAY DIFFRACTION (3.1 Å) | Cite: | Characterization of the metal ion binding helix-hairpin-helix motifs in human DNA polymerase beta by X-ray structural analysis. Biochemistry, 35, 1996
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8ICC
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![BU of 8icc by Molmil](/molmil-images/mine/8icc) | |