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2A9X
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BU of 2a9x by Molmil
TAR RNA recognition by a cyclic peptidomimetic of Tat protein
Descriptor: BIV TAR RNA, BIV-2 cyclic peptide
Authors:Leeper, T.C, Athanassiou, Z, Dias, R.L, Robinson, J.A, Varani, G.
Deposit date:2005-07-12
Release date:2005-11-01
Last modified:2022-03-09
Method:SOLUTION NMR
Cite:TAR RNA recognition by a cyclic peptidomimetic of Tat protein.
Biochemistry, 44, 2005
2AXI
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BU of 2axi by Molmil
HDM2 in complex with a beta-hairpin
Descriptor: 3[N-MORPHOLINO]PROPANE SULFONIC ACID, SULFATE ION, Ubiquitin-protein ligase E3 Mdm2, ...
Authors:Mittl, P.R.E, Fasan, R, Robinson, J, Gruetter, M.G.
Deposit date:2005-09-05
Release date:2006-03-21
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Structure-Activity Studies in a Family of beta-Hairpin Protein Epitope Mimetic Inhibitors of the p53-HDM2 Protein-Protein Interaction.
Chembiochem, 7, 2006
1K3T
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BU of 1k3t by Molmil
Structure of Glycosomal Glyceraldehyde-3-Phosphate Dehydrogenase from Trypanosoma cruzi Complexed with Chalepin, a Coumarin Derivative Inhibitor
Descriptor: 6-(1,1-DIMETHYLALLYL)-2-(1-HYDROXY-1-METHYLETHYL)-2,3-DIHYDRO-7H-FURO[3,2-G]CHROMEN-7-ONE, Glyceraldehyde-3-phosphate dehydrogenase
Authors:Pavao, F.
Deposit date:2001-10-04
Release date:2002-06-19
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Structure of Trypanosoma cruzi glycosomal glyceraldehyde-3-phosphate dehydrogenase complexed with chalepin, a natural product inhibitor, at 1.95 A resolution.
FEBS Lett., 520, 2002
2NS4
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BU of 2ns4 by Molmil
Solution structure of a Beta-Hairpin Peptidomimetic Inhibitor of the BIV Tat-Tar Interaction
Descriptor: L-22 CYCLIC PEPTIDE
Authors:Moehle, K, Patora, K, Robinson, J.A.
Deposit date:2006-11-03
Release date:2007-01-30
Last modified:2023-12-27
Method:SOLUTION NMR
Cite:Structure-Guided Peptidomimetic Design Leads to Nanomolar beta-Hairpin Inhibitors of the Tat-TAR Interaction of Bovine Immunodeficiency Virus
Biochemistry, 46, 2007

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数据于2024-07-24公开中

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