6BQB
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![BU of 6bqb by Molmil](/molmil-images/mine/6bqb) | MGG4 Fab in complex with peptide | Descriptor: | GLYCEROL, MGG4 Fab heavy chain, MGG4 Fab light chain, ... | Authors: | Oyen, D, Tan, J, Lanzavecchia, A, Wilson, I.A. | Deposit date: | 2017-11-27 | Release date: | 2018-03-07 | Last modified: | 2018-04-25 | Method: | X-RAY DIFFRACTION (1.769 Å) | Cite: | A public antibody lineage that potently inhibits malaria infection through dual binding to the circumsporozoite protein. Nat. Med., 24, 2018
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7POM
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![BU of 7pom by Molmil](/molmil-images/mine/7pom) | |
7PP9
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![BU of 7pp9 by Molmil](/molmil-images/mine/7pp9) | |
6TL6
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![BU of 6tl6 by Molmil](/molmil-images/mine/6tl6) | |
6TL5
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![BU of 6tl5 by Molmil](/molmil-images/mine/6tl5) | |
6FE0
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![BU of 6fe0 by Molmil](/molmil-images/mine/6fe0) | |
6FE2
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![BU of 6fe2 by Molmil](/molmil-images/mine/6fe2) | Three dimensional structure of human carbonic anhydrase IX | Descriptor: | Carbonic anhydrase 9, ZINC ION | Authors: | Leitans, J, Tars, K. | Deposit date: | 2017-12-28 | Release date: | 2018-07-04 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.87 Å) | Cite: | Novel fluorinated carbonic anhydrase IX inhibitors reduce hypoxia-induced acidification and clonogenic survival of cancer cells. Oncotarget, 9, 2018
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6FE1
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![BU of 6fe1 by Molmil](/molmil-images/mine/6fe1) | |
5MJN
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![BU of 5mjn by Molmil](/molmil-images/mine/5mjn) | |
6G98
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![BU of 6g98 by Molmil](/molmil-images/mine/6g98) | |
6G9U
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![BU of 6g9u by Molmil](/molmil-images/mine/6g9u) | |
5AMG
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![BU of 5amg by Molmil](/molmil-images/mine/5amg) | |
5AML
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![BU of 5aml by Molmil](/molmil-images/mine/5aml) | |
5AMD
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![BU of 5amd by Molmil](/molmil-images/mine/5amd) | |
8JFC
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![BU of 8jfc by Molmil](/molmil-images/mine/8jfc) | V1/S quadruple mutant Plasmodium falciparum dihydrofolate reductase-thymidylate synthase (PfDHFR-TS) complexed with compound 6 (B21591), NADPH and dUMP | Descriptor: | 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 4-[3-[[2,4-bis(azanyl)-6-ethyl-pyrimidin-5-yl]methyl]phenyl]benzoic acid, Bifunctional dihydrofolate reductase-thymidylate synthase, ... | Authors: | Vanichtanankul, J, Saeyang, T, Vitsupakorn, D, Saepua, S, Thongpanchang, C, Yuthavong, Y, Kamchonwongpaisan, S, Hoarau, M. | Deposit date: | 2023-05-17 | Release date: | 2023-08-23 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Discovery of rigid biphenyl Plasmodium falciparum DHFR inhibitors using a fragment linking strategy. Rsc Med Chem, 14, 2023
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8JFB
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![BU of 8jfb by Molmil](/molmil-images/mine/8jfb) | V1/S quadruple mutant Plasmodium falciparum dihydrofolate reductase-thymidylate synthase (PfDHFR-TS) complexed with compound 4 (B21588), NADPH and dUMP | Descriptor: | 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 3-[4-[[2,4-bis(azanyl)-6-ethyl-pyrimidin-5-yl]methyl]phenyl]benzoic acid, Bifunctional dihydrofolate reductase-thymidylate synthase, ... | Authors: | Vanichtanankul, J, Saeyang, T, Vitsupakorn, D, Saepua, S, Thongpanchang, C, Yuthavong, Y, Kamchonwongpaisan, S, Hoarau, M. | Deposit date: | 2023-05-17 | Release date: | 2023-08-23 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (2.65 Å) | Cite: | Discovery of rigid biphenyl Plasmodium falciparum DHFR inhibitors using a fragment linking strategy. Rsc Med Chem, 14, 2023
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8JFD
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![BU of 8jfd by Molmil](/molmil-images/mine/8jfd) | V1/S quadruple mutant Plasmodium falciparum dihydrofolate reductase-thymidylate synthase (PfDHFR-TS) complexed with compound 8 (B21594), NADPH and dUMP | Descriptor: | 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 3-[3-[[2,4-bis(azanyl)-6-ethyl-pyrimidin-5-yl]methyl]phenyl]benzoic acid, Bifunctional dihydrofolate reductase-thymidylate synthase, ... | Authors: | Vanichtanankul, J, Saeyang, T, Vitsupakorn, D, Saepua, S, Thongpanchang, C, Yuthavong, Y, Kamchonwongpaisan, S, Hoarau, M. | Deposit date: | 2023-05-17 | Release date: | 2023-08-23 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Discovery of rigid biphenyl Plasmodium falciparum DHFR inhibitors using a fragment linking strategy. Rsc Med Chem, 14, 2023
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2OYW
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![BU of 2oyw by Molmil](/molmil-images/mine/2oyw) | Neurotensin in TFE:H2O (80:20) | Descriptor: | neurotensin | Authors: | Monti, J.P, Coutant, J, Curmi, P.A. | Deposit date: | 2007-02-23 | Release date: | 2007-05-08 | Last modified: | 2019-12-25 | Method: | SOLUTION NMR | Cite: | NMR Solution Structure of Neurotensin in Membrane-Mimetic Environments: Molecular Basis for Neurotensin Receptor Recognition. Biochemistry, 46, 2007
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5GR8
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![BU of 5gr8 by Molmil](/molmil-images/mine/5gr8) | Crystal structure of PEPR1-AtPEP1 | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Elicitor peptide 1, ... | Authors: | Chai, J.J, Tang, J. | Deposit date: | 2016-08-08 | Release date: | 2016-12-14 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.587 Å) | Cite: | Structural basis for recognition of an endogenous peptide by the plant receptor kinase PEPR1 Cell Res., 25, 2015
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2OYV
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![BU of 2oyv by Molmil](/molmil-images/mine/2oyv) | Neurotensin in DPC micelles | Descriptor: | neurotensin | Authors: | Monti, J.P, Coutant, J, Curmi, P.A. | Deposit date: | 2007-02-23 | Release date: | 2007-05-08 | Last modified: | 2019-12-25 | Method: | SOLUTION NMR | Cite: | NMR Solution Structure of Neurotensin in Membrane-Mimetic Environments: Molecular Basis for Neurotensin Receptor Recognition. Biochemistry, 46, 2007
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6KP7
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![BU of 6kp7 by Molmil](/molmil-images/mine/6kp7) | |
6KP2
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![BU of 6kp2 by Molmil](/molmil-images/mine/6kp2) | |
6KOT
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![BU of 6kot by Molmil](/molmil-images/mine/6kot) | |
6LEV
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![BU of 6lev by Molmil](/molmil-images/mine/6lev) | Quadruple mutant (N51I+C59R+S108N+I164L) plasmodium falciparum dihydrofolate reductase-thymidylate synthase (PfDHFR-TS) complexed with compound 46 and NADPH | Descriptor: | 2-[[4,6-bis(azanyl)-2,2-dimethyl-1,3,5-triazin-1-yl]oxy]-N-(4-chlorophenyl)ethanamide, Bifunctional dihydrofolate reductase-thymidylate synthase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | Authors: | Vanichtanankul, J, Vitsupakorn, D. | Deposit date: | 2019-11-27 | Release date: | 2020-12-02 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (2.644 Å) | Cite: | Flexible diaminodihydrotriazine inhibitors of Plasmodium falciparum dihydrofolate reductase: Binding strengths, modes of binding and their antimalarial activities. Eur.J.Med.Chem., 195, 2020
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6KPR
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![BU of 6kpr by Molmil](/molmil-images/mine/6kpr) | |