7KP9
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![BU of 7kp9 by Molmil](/molmil-images/mine/7kp9) | asymmetric hTNF-alpha | Descriptor: | 1-{[2-(difluoromethoxy)phenyl]methyl}-2-methyl-6-[6-(piperazin-1-yl)pyridin-3-yl]-1H-benzimidazole, Tumor necrosis factor | Authors: | Arakaki, T.L, Abendroth, J, Fairman, J.W, Foley, A, Ceska, T. | Deposit date: | 2020-11-10 | Release date: | 2021-01-13 | Last modified: | 2024-04-03 | Method: | X-RAY DIFFRACTION (2.15 Å) | Cite: | Structural insights into the disruption of TNF-TNFR1 signalling by small molecules stabilising a distorted TNF. Nat Commun, 12, 2021
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3MYB
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![BU of 3myb by Molmil](/molmil-images/mine/3myb) | |
3OI9
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![BU of 3oi9 by Molmil](/molmil-images/mine/3oi9) | |
3QYR
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![BU of 3qyr by Molmil](/molmil-images/mine/3qyr) | |
3R4T
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![BU of 3r4t by Molmil](/molmil-images/mine/3r4t) | |
3R9P
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![BU of 3r9p by Molmil](/molmil-images/mine/3r9p) | |
7JWL
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![BU of 7jwl by Molmil](/molmil-images/mine/7jwl) | Crystal Structure of Pseudomonas aeruginosa Penicillin Binding Protein 3 (PAE-PBP3) bound to ETX0462 | Descriptor: | CHLORIDE ION, ETX0462 (Bound form), Peptidoglycan D,D-transpeptidase FtsI | Authors: | Mayclin, S.J, Abendroth, J, Horanyi, P.S, Sylvester, M, Wu, X, Shapiro, A, Moussa, S, Durand-Reville, T.F. | Deposit date: | 2020-08-25 | Release date: | 2021-05-26 | Last modified: | 2023-10-18 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Rational design of a new antibiotic class for drug-resistant infections. Nature, 597, 2021
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3HZG
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![BU of 3hzg by Molmil](/molmil-images/mine/3hzg) | Crystal structure of mycobacterium tuberculosis thymidylate synthase X bound with FAD | Descriptor: | FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, PHOSPHATE ION, ... | Authors: | Staker, B.L, Rathod, P, Hunter, J, Seattle Structural Genomics Center for Infectious Disease (SSGCID) | Deposit date: | 2009-06-23 | Release date: | 2009-07-07 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.45 Å) | Cite: | Increasing the structural coverage of tuberculosis drug targets. Tuberculosis (Edinb), 95, 2015
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3PE8
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![BU of 3pe8 by Molmil](/molmil-images/mine/3pe8) | |
3R9S
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![BU of 3r9s by Molmil](/molmil-images/mine/3r9s) | |
3R0O
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![BU of 3r0o by Molmil](/molmil-images/mine/3r0o) | |
3MMT
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![BU of 3mmt by Molmil](/molmil-images/mine/3mmt) | |
1K5G
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![BU of 1k5g by Molmil](/molmil-images/mine/1k5g) | Crystal structure of Ran-GDP-AlFx-RanBP1-RanGAP complex | Descriptor: | ALUMINUM FLUORIDE, GTP-binding nuclear protein RAN, GUANOSINE-5'-DIPHOSPHATE, ... | Authors: | Seewald, M.J, Koerner, C, Wittinghofer, A, Vetter, I.R. | Deposit date: | 2001-10-10 | Release date: | 2002-02-13 | Last modified: | 2023-08-16 | Method: | X-RAY DIFFRACTION (3.1 Å) | Cite: | RanGAP mediates GTP hydrolysis without an arginine finger. Nature, 415, 2002
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3PK0
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![BU of 3pk0 by Molmil](/molmil-images/mine/3pk0) | |
3RSI
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![BU of 3rsi by Molmil](/molmil-images/mine/3rsi) | |
3R9Q
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![BU of 3r9q by Molmil](/molmil-images/mine/3r9q) | |
3RR6
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![BU of 3rr6 by Molmil](/molmil-images/mine/3rr6) | |
3QHA
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![BU of 3qha by Molmil](/molmil-images/mine/3qha) | |
3RR2
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![BU of 3rr2 by Molmil](/molmil-images/mine/3rr2) | |
6C99
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![BU of 6c99 by Molmil](/molmil-images/mine/6c99) | Crystal structure of FcRn bound to UCB-303 | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-2-microglobulin, CITRIC ACID, ... | Authors: | Fox III, D, Abendroth, J, Porter, J, Deboves, H. | Deposit date: | 2018-01-25 | Release date: | 2018-05-30 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Insight into small molecule binding to the neonatal Fc receptor by X-ray crystallography and 100 kHz magic-angle-spinning NMR. PLoS Biol., 16, 2018
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3R2N
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![BU of 3r2n by Molmil](/molmil-images/mine/3r2n) | |
3R9T
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![BU of 3r9t by Molmil](/molmil-images/mine/3r9t) | |
3RFQ
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![BU of 3rfq by Molmil](/molmil-images/mine/3rfq) | |
3RRV
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![BU of 3rrv by Molmil](/molmil-images/mine/3rrv) | |
4G50
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![BU of 4g50 by Molmil](/molmil-images/mine/4g50) | |