8Q1N
| Cyclic peptide binder of the WBM-site of WDR5 | 分子名称: | Cyclic peptide inhibitor, WD repeat-containing protein 5 | 著者 | Schmeing, S, Chang, J.Y, t Hart, P, Gasper, R. | 登録日 | 2023-08-01 | 公開日 | 2023-09-06 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.843 Å) | 主引用文献 | Macrocyclic peptides as inhibitors of WDR5-lncRNA interactions. Chem.Commun.(Camb.), 59, 2023
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7BOC
| Crystal structure of the PRMT5 TIM barrel domain in complex with RioK1 peptide | 分子名称: | Protein arginine N-methyltransferase 5, peptide | 著者 | Krzyzanowski, A, t Hart, P, Waldmann, H, Gasper, R. | 登録日 | 2021-01-25 | 公開日 | 2021-09-15 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Biochemical Investigation of the Interaction of pICln, RioK1 and COPR5 with the PRMT5-MEP50 Complex. Chembiochem, 22, 2021
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8BWF
| PTBP1 RRM1 bound to an allosteric inhibitor | 分子名称: | AMINO GROUP, GLYCEROL, Ligand, ... | 著者 | Schmeing, S, Vetter, I, t Hart, P, Gasper, R. | 登録日 | 2022-12-06 | 公開日 | 2023-10-11 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Rationally designed stapled peptides allosterically inhibit PTBP1-RNA-binding. Chem Sci, 14, 2023
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