5F17
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![BU of 5f17 by Molmil](/molmil-images/mine/5f17) | |
8IFU
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![BU of 8ifu by Molmil](/molmil-images/mine/8ifu) | HcCCR in NaCl | 分子名称: | (1S)-2-{[(S)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-1-[(octadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, HcCCR, RETINAL, ... | 著者 | Zhang, M.F. | 登録日 | 2023-02-19 | 公開日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (2.37 Å) | 主引用文献 | Structure of HcCCR To Be Published
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8IO5
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![BU of 8io5 by Molmil](/molmil-images/mine/8io5) | Herg1a-herg1b closed state 2 | 分子名称: | Potassium voltage-gated channel subfamily H member 2 | 著者 | Zhang, M.F. | 登録日 | 2023-03-10 | 公開日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Structure of Herg1a-herg1b open state To Be Published
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8IOB
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![BU of 8iob by Molmil](/molmil-images/mine/8iob) | Herg1a-herg1b closed state 1 | 分子名称: | Potassium voltage-gated channel subfamily H member 2 | 著者 | Zhang, M.F. | 登録日 | 2023-03-10 | 公開日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | Structure of Herg1a-herg1b closed state 1 To Be Published
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8IO4
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![BU of 8io4 by Molmil](/molmil-images/mine/8io4) | Herg1a-herg1b open state | 分子名称: | Potassium voltage-gated channel subfamily H member 2 | 著者 | Zhang, M.F. | 登録日 | 2023-03-10 | 公開日 | 2024-03-13 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structure of Herg1a-herg1b open state To Be Published
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7XTK
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![BU of 7xtk by Molmil](/molmil-images/mine/7xtk) | |
7XYM
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![BU of 7xym by Molmil](/molmil-images/mine/7xym) | |
5EYI
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![BU of 5eyi by Molmil](/molmil-images/mine/5eyi) | Structure of PRRSV apo-NSP11 at 2.16A | 分子名称: | 2-(2-METHOXYETHOXY)ETHANOL, CHLORIDE ION, Non-structural protein 11, ... | 著者 | Zhang, M.F, Chen, Z. | 登録日 | 2015-11-25 | 公開日 | 2016-10-12 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Structural Biology of the Arterivirus nsp11 Endoribonucleases. J. Virol., 91, 2017
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7V1U
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![BU of 7v1u by Molmil](/molmil-images/mine/7v1u) | Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor ZJ12 | 分子名称: | 1,2-ETHANEDIOL, Bromodomain-containing protein 4, ~{N}-(3-ethyl-6-methoxy-1,2-benzoxazol-5-yl)-2-methoxy-benzenesulfonamide | 著者 | Zhang, M, Wang, C, Zhang, C, Zhang, Y, Xu, Y. | 登録日 | 2021-08-06 | 公開日 | 2022-08-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Design, synthesis and pharmacological characterization of N-(3-ethylbenzo[d]isoxazol-5-yl) sulfonamide derivatives as BRD4 inhibitors against acute myeloid leukemia. Acta Pharmacol.Sin., 43, 2022
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7V2J
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![BU of 7v2j by Molmil](/molmil-images/mine/7v2j) | Crystal Structure of the first bromodomain of human BRD4 in complex with the inhibitor 33 | 分子名称: | Bromodomain-containing protein 4, ~{N}-(3-ethyl-6-methoxy-1,2-benzoxazol-5-yl)-4-methoxy-benzenesulfonamide | 著者 | Zhang, M, Wang, C, Zhang, C, Zhang, Y, Xu, Y. | 登録日 | 2021-08-09 | 公開日 | 2022-08-17 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.24 Å) | 主引用文献 | Design, synthesis and pharmacological characterization of N-(3-ethylbenzo[d]isoxazol-5-yl) sulfonamide derivatives as BRD4 inhibitors against acute myeloid leukemia. Acta Pharmacol.Sin., 43, 2022
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5HC1
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5HBZ
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![BU of 5hbz by Molmil](/molmil-images/mine/5hbz) | |
7YJ0
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7YIG
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![BU of 7yig by Molmil](/molmil-images/mine/7yig) | Human KCNH5 pre-open state 2 | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5 | 著者 | Zhang, M.F. | 登録日 | 2022-07-16 | 公開日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel. Nat Commun, 14, 2023
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7YIE
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![BU of 7yie by Molmil](/molmil-images/mine/7yie) | Human KCNH5-closed state 2 | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5 | 著者 | Zhang, M.F. | 登録日 | 2022-07-16 | 公開日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel. Nat Commun, 14, 2023
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7YIH
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![BU of 7yih by Molmil](/molmil-images/mine/7yih) | Human KCNH5 open state | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5 | 著者 | Zhang, M.F. | 登録日 | 2022-07-16 | 公開日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel. Nat Commun, 14, 2023
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7YIF
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![BU of 7yif by Molmil](/molmil-images/mine/7yif) | Human KCNH5 pre-open state 1 | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5 | 著者 | Zhang, M.F. | 登録日 | 2022-07-16 | 公開日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel. Nat Commun, 14, 2023
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7YID
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![BU of 7yid by Molmil](/molmil-images/mine/7yid) | Human KCNH5 closed state 1 | 分子名称: | POTASSIUM ION, Potassium voltage-gated channel subfamily H member 5 | 著者 | Zhang, M.F. | 登録日 | 2022-07-16 | 公開日 | 2023-04-05 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Mechanism underlying delayed rectifying in human voltage-mediated activation Eag2 channel. Nat Commun, 14, 2023
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7YIJ
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8GRS
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![BU of 8grs by Molmil](/molmil-images/mine/8grs) | human TMEM63A | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, CSC1-like protein 1 | 著者 | Zhang, M.F. | 登録日 | 2022-09-02 | 公開日 | 2023-06-14 | 最終更新日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | A mechanical-coupling mechanism in OSCA/TMEM63 channel mechanosensitivity. Nat Commun, 14, 2023
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8GRN
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![BU of 8grn by Molmil](/molmil-images/mine/8grn) | AtOSCA1.1 extended state | 分子名称: | Protein OSCA1, [1-MYRISTOYL-GLYCEROL-3-YL]PHOSPHONYLCHOLINE | 著者 | Zhang, M.F. | 登録日 | 2022-09-02 | 公開日 | 2023-06-14 | 最終更新日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | A mechanical-coupling mechanism in OSCA/TMEM63 channel mechanosensitivity. Nat Commun, 14, 2023
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8GSO
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![BU of 8gso by Molmil](/molmil-images/mine/8gso) | AtOSCA3.1 channel extended state | 分子名称: | CSC1-like protein ERD4 | 著者 | Zhang, M.F. | 登録日 | 2022-09-06 | 公開日 | 2023-06-14 | 最終更新日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | A mechanical-coupling mechanism in OSCA/TMEM63 channel mechanosensitivity. Nat Commun, 14, 2023
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8GRO
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![BU of 8gro by Molmil](/molmil-images/mine/8gro) | AtOSCA3.1 contracted state | 分子名称: | CSC1-like protein ERD4 | 著者 | Zhang, M.F. | 登録日 | 2022-09-02 | 公開日 | 2023-06-14 | 最終更新日 | 2023-07-26 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | A mechanical-coupling mechanism in OSCA/TMEM63 channel mechanosensitivity. Nat Commun, 14, 2023
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7DHS
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![BU of 7dhs by Molmil](/molmil-images/mine/7dhs) | Crystal Structure Analysis of the BRD4 | 分子名称: | 6-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[(1R)-1-phenylethyl]benzo[cd]indol-2-one, Bromodomain-containing protein 4 | 著者 | Wu, T, Xiang, Q, Wang, C, Wu, C, Zhang, C, Zhang, M, Liu, Z, Zhang, Y, Xiao, L, Xu, Y. | 登録日 | 2020-11-17 | 公開日 | 2021-09-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Y06014 is a selective BET inhibitor for the treatment of prostate cancer. Acta Pharmacol.Sin., 42, 2021
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