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1MUI
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BU of 1mui by Molmil
Crystal structure of HIV-1 protease complexed with Lopinavir.
分子名称: N-{1-BENZYL-4-[2-(2,6-DIMETHYL-PHENOXY)-ACETYLAMINO]-3-HYDROXY-5-PHENYL-PENTYL}-3-METHYL-2-(2-OXO-TETRAHYDRO-PYRIMIDIN-1-YL)-BUTYRAMIDE, protease
著者Stoll, V, Qin, W, Stewart, K.D, Jakob, C, Park, C, Walter, K, Simmer, R.L, Helfrich, R, Bussiere, D, Kao, J, Kempf, D, Sham, H.L, Norbeck, D.W.
登録日2002-09-23
公開日2002-10-23
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献X-ray Crystallographic Structure of ABT-378 (Lopinavir) Bound to HIV-1 Protease
BIOORG.MED.CHEM., 10, 2002
1YUB
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BU of 1yub by Molmil
SOLUTION STRUCTURE OF AN RRNA METHYLTRANSFERASE (ERMAM) THAT CONFERS MACROLIDE-LINCOSAMIDE-STREPTOGRAMIN ANTIBIOTIC RESISTANCE, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: RRNA METHYLTRANSFERASE
著者Yu, L, Petros, A.M, Schnuchel, A, Zhong, P, Severin, J.M, Walter, K, Holzman, T.F, Fesik, S.W.
登録日1997-03-04
公開日1998-03-04
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of an rRNA methyltransferase (ErmAM) that confers macrolide-lincosamide-streptogramin antibiotic resistance.
Nat.Struct.Biol., 4, 1997
1DHM
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BU of 1dhm by Molmil
DNA-BINDING DOMAIN OF E2 FROM HUMAN PAPILLOMAVIRUS-31, NMR, MINIMIZED AVERAGE STRUCTURE
分子名称: E2 PROTEIN
著者Liang, H, Petros, A.P, Meadows, R.P, Yoon, H.S, Egan, D.A, Walter, K, Holzman, T.F, Robins, T, Fesik, S.W.
登録日1995-08-15
公開日1996-12-07
最終更新日2024-04-10
実験手法SOLUTION NMR
主引用文献Solution structure of the DNA-binding domain of a human papillomavirus E2 protein: evidence for flexible DNA-binding regions.
Biochemistry, 35, 1996
2K39
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BU of 2k39 by Molmil
Recognition dynamics up to microseconds revealed from RDC derived ubiquitin ensemble in solution
分子名称: Ubiquitin
著者Lange, O.F, Lakomek, N.A, Fares, C, Schroder, G, Walter, K, Becker, S, Meiler, J, Grubmuller, H, Griesinger, C, de Groot, B.L.
登録日2008-04-25
公開日2008-06-24
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Recognition dynamics up to microseconds revealed from an RDC-derived ubiquitin ensemble in solution.
Science, 320, 2008
5IRS
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BU of 5irs by Molmil
crystal structure of the proteasomal Rpn13 PRU-domain
分子名称: 2,3-DIHYDROXY-1,4-DITHIOBUTANE, Proteasomal ubiquitin receptor ADRM1
著者Chen, X, Shi, K, Walters, K, Aihara, H.
登録日2016-03-14
公開日2016-07-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.796 Å)
主引用文献Structures of Rpn1 T1:Rad23 and hRpn13:hPLIC2 Reveal Distinct Binding Mechanisms between Substrate Receptors and Shuttle Factors of the Proteasome.
Structure, 24, 2016
2KP8
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BU of 2kp8 by Molmil
Ligand bound to a model peptide that mimics the open fusogenic form
分子名称: 5-{[(4'-methoxybiphenyl-4-yl)methyl][(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl}benzene-1,2,4-tricarboxylic acid, Model peptide
著者Olejniczak, E.T.
登録日2009-10-09
公開日2010-01-19
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Non-peptide entry inhibitors of HIV-1 that target the gp41 coiled coil pocket.
Bioorg.Med.Chem.Lett., 20, 2010
1A7G
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BU of 1a7g by Molmil
THE CRYSTAL STRUCTURE OF THE E2 DNA-BINDING DOMAIN FROM HUMAN PAPILLOMAVIRUS AT 2.4 ANGSTROMS
分子名称: REGULATORY PROTEIN E2, SULFATE ION
著者Bussiere, D.E, Giranda, V.L.
登録日1998-03-13
公開日1999-04-27
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of the E2 DNA-binding domain from human papillomavirus serotype 31 at 2.4 A.
Acta Crystallogr.,Sect.D, 54, 1998
1ZP5
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BU of 1zp5 by Molmil
Crystal structure of the complex between MMP-8 and a N-hydroxyurea inhibitor
分子名称: CALCIUM ION, N-{2-[(4'-CYANO-1,1'-BIPHENYL-4-YL)OXY]ETHYL}-N'-HYDROXY-N-METHYLUREA, Neutrophil collagenase, ...
著者Campestre, C, Agamennone, M, Tortorella, P, Preziuso, S, Biasone, A, Gavuzzo, E, Pochetti, G, Mazza, F, Tschesche, H, Gallina, C.
登録日2005-05-16
公開日2005-12-06
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献N-Hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: Mode of binding in a complex with MMP-8.
Bioorg.Med.Chem.Lett., 16, 2006
2N12
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BU of 2n12 by Molmil
Solution structure of human Myosin VI isoform3 (1050-1131)
分子名称: Unconventional myosin-VI
著者He, F, Walters, K.
登録日2015-03-20
公開日2016-03-02
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Diverse functions of myosin VI elucidated by an isoform-specific alpha-helix domain.
Nat.Struct.Mol.Biol., 23, 2016
2R2Y
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BU of 2r2y by Molmil
Crystal structure of the proteasomal Rpn13 PRU-domain
分子名称: Protein ADRM1
著者Groll, M, Walters, K, Dikic, I, Finley, D.
登録日2007-08-28
公開日2008-05-13
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Ubiquitin docking at the proteasome through a novel pleckstrin-homology domain interaction.
Nature, 453, 2008
2N0Z
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BU of 2n0z by Molmil
Solution structure of MyUb (1080-1122) of human Myosin VI
分子名称: Unconventional myosin-VI
著者He, F, Walters, K.
登録日2015-03-20
公開日2016-03-09
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Myosin VI Contains a Compact Structural Motif that Binds to Ubiquitin Chains.
Cell Rep, 14, 2016
2N10
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BU of 2n10 by Molmil
Solution structure of MyUb (1080-1131) of human Myosin VI
分子名称: Unconventional myosin-VI
著者He, F, Ehlinger, A, Walters, K.
登録日2015-03-20
公開日2016-03-09
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Myosin VI Contains a Compact Structural Motif that Binds to Ubiquitin Chains.
Cell Rep, 14, 2016
2N11
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BU of 2n11 by Molmil
Solution structure of human Myosin VI isoform3 (998-1071)
分子名称: Unconventional myosin-VI
著者He, F, Walters, K.
登録日2015-03-20
公開日2016-03-09
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Myosin VI Contains a Compact Structural Motif that Binds to Ubiquitin Chains.
Cell Rep, 14, 2016
2N13
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BU of 2n13 by Molmil
Complex structure of MyUb (1080-1122) of human Myosin VI with K63-diUb
分子名称: Ubiquitin, Unconventional myosin-VI
著者He, F, Walters, K.
登録日2015-03-20
公開日2016-03-09
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Myosin VI Contains a Compact Structural Motif that Binds to Ubiquitin Chains.
Cell Rep, 14, 2016

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件を2024-07-17に公開中

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