8RM7
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![BU of 8rm7 by Molmil](/molmil-images/mine/8rm7) | Crystal Structure of Human Androgen Receptor DNA Binding Domain Bound to its Response Element: MMTV-177 GRE/ARE | 分子名称: | Isoform 2 of Androgen receptor, MMTV-177 GRE/ARE Chain C, MMTV-177 GRE/ARE, ... | 著者 | Lee, X.Y, Helsen, C, Van Eynde, W, Voet, A, Claessens, F. | 登録日 | 2024-01-05 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural mechanism underlying variations in DNA binding by the androgen receptor. J.Steroid Biochem.Mol.Biol., 241, 2024
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8RM6
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![BU of 8rm6 by Molmil](/molmil-images/mine/8rm6) | Crystal Structure of Human Androgen Receptor DNA Binding Domain Bound to its Response Element: C3(1)ARE | 分子名称: | C3(1)ARE_Chain C, C3(1)ARE_Chain D, Isoform 2 of Androgen receptor, ... | 著者 | Lee, X.Y, Helsen, C, Van Eynde, W, Voet, A, Claessens, F. | 登録日 | 2024-01-05 | 公開日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural mechanism underlying variations in DNA binding by the androgen receptor. J.Steroid Biochem.Mol.Biol., 241, 2024
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5NSD
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![BU of 5nsd by Molmil](/molmil-images/mine/5nsd) | Co-crystal structure of NAMPT dimer with KPT-9274 | 分子名称: | (~{E})-3-(6-azanylpyridin-3-yl)-~{N}-[[5-[4-[4,4-bis(fluoranyl)piperidin-1-yl]carbonylphenyl]-7-(4-fluorophenyl)-1-benzofuran-2-yl]methyl]prop-2-enamide, GLYCEROL, Nicotinamide phosphoribosyltransferase, ... | 著者 | Neggers, J.E, Kwanten, B, Dierckx, T, Noguchi, H, Voet, A, Vercruysse, T, Baloglu, E, Senapedis, W, Jacquemyn, M, Daelemans, D. | 登録日 | 2017-04-26 | 公開日 | 2018-02-14 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.046 Å) | 主引用文献 | Target identification of small molecules using large-scale CRISPR-Cas mutagenesis scanning of essential genes. Nat Commun, 9, 2018
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3LPU
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![BU of 3lpu by Molmil](/molmil-images/mine/3lpu) | HIV integrase | 分子名称: | (2S)-2-(6-chloro-2-methyl-4-phenylquinolin-3-yl)pentanoic acid, 2-[3-[3-(2-hydroxyethoxy)propoxy]propoxy]ethanol, CALCIUM ION, ... | 著者 | Nicolet, S, Christ, F, Voet, A, Marchand, A, Strelkov, S.V, de Maeyer, M, Chaltin, P, Debyzer, Z. | 登録日 | 2010-02-06 | 公開日 | 2010-05-12 | 最終更新日 | 2021-11-10 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication. Nat.Chem.Biol., 6, 2010
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3LPT
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![BU of 3lpt by Molmil](/molmil-images/mine/3lpt) | HIV integrase | 分子名称: | (6-chloro-2-oxo-4-phenyl-1,2-dihydroquinolin-3-yl)acetic acid, 2-[3-[3-(2-hydroxyethoxy)propoxy]propoxy]ethanol, CALCIUM ION, ... | 著者 | Nicolet, S, Christ, F, Voet, A, Marchand, A, Strelkov, S.V, de Maeyer, M, Chaltin, P, Debyzer, Z. | 登録日 | 2010-02-05 | 公開日 | 2010-05-12 | 最終更新日 | 2021-11-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication. Nat.Chem.Biol., 6, 2010
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5Z5E
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![BU of 5z5e by Molmil](/molmil-images/mine/5z5e) | |
6F0Q
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![BU of 6f0q by Molmil](/molmil-images/mine/6f0q) | |
6F0S
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![BU of 6f0s by Molmil](/molmil-images/mine/6f0s) | |
6F0T
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![BU of 6f0t by Molmil](/molmil-images/mine/6f0t) | Crystal structure of Pizza6-SFW | 分子名称: | GLYCEROL, Pizza6-SFW | 著者 | Noguchi, H, De Zitter, E, Van Meervelt, L, Voet, A.R.D. | 登録日 | 2017-11-20 | 公開日 | 2018-03-21 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Design of tryptophan-containing mutants of the symmetrical Pizza protein for biophysical studies. Biochem. Biophys. Res. Commun., 497, 2018
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3L1Q
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![BU of 3l1q by Molmil](/molmil-images/mine/3l1q) | The crystal structure of the undecamer d(TGGCCTTAAGG) | 分子名称: | 5'-D(*TP*GP*GP*CP*CP*TP*TP*AP*AP*GP*G)-3' | 著者 | Van Hecke, K. | 登録日 | 2009-12-14 | 公開日 | 2010-10-27 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Designing Triple Helical Fragments: The Crystal Structure of the Undecamer d(TGGCCTTAAGG) Mimicking T·AT Base Triplets Cryst.Growth Des., 10, 2010
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